Target Details
| UniProt AC | P05107 |
|---|---|
| Gene Symbol | ITGB2 |
| Protein Name | Integrin beta-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF23105 (EGF_integrin) PF08725 (Integrin_b_cyt) PF07965 (Integrin_B_tail) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 373
- Clinical molecules 0
- Avg pChEMBL 7.14
KEGG Pathways (21)
- Amoebiasis
- Cell adhesion molecule (CAM) interaction
- Complement and coagulation cascades
- Hippo signaling pathway
- Human T-cell leukemia virus 1 infection
- IgSF CAM signaling
- Integrin signaling
- Legionellosis
- Leishmaniasis
- Leukocyte transendothelial migration
- Malaria
- Natural killer cell mediated cytotoxicity
- Neutrophil extracellular trap formation
- Pertussis
- Phagosome
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Rheumatoid arthritis
- Staphylococcus aureus infection
- Tuberculosis
- Viral myocarditis
Associated Diseases (1)
Active Molecules (373)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZRGQDLKQXUUCDI
|
6.8 | IC50 | 3 | — | |
DZDHPEOBDDCTPU
|
6.8 | IC50 | 3 | — | |
MORWDGMDJBERJV
|
6.8 | IC50 | 3 | — | |
FYCLIBMUEUKVCF
|
6.8 | IC50 | 3 | — | |
LOKMFEWDWMYUHX
|
6.8 | IC50 | 3 | — | |
RPDQFVCWMZSDOT
|
6.8 | Kd | 3 | — | |
SUZAUKCYSQZDMS
|
6.7 | IC50 | 3 | — | |
JVFGBZRFEBWUBQ
|
6.7 | IC50 | 3 | — | |
MXCAAVRZKWSUKO
|
6.7 | Kd | 3 | — | |
HPSCLHCEPQQJNB
|
6.7 | IC50 | 3 | — | |
OCTRODWZSNQUGG
|
6.7 | IC50 | 3 | — | |
ULKWCLJACWMJSJ
|
6.7 | IC50 | 3 | — | |
WPVRNXUYVXQXPY
|
6.7 | IC50 | 2 | — | |
HQRUSYULBHQARY
|
6.7 | IC50 | 3 | — | |
UDJIFGWLUPATRA
|
6.7 | IC50 | 3 | — | |
XGPHRJBZYZFMFD
|
6.7 | IC50 | 3 | — | |
HSSYLIYWARWUTA
|
6.6 | IC50 | 3 | — | |
JNPJONSHMIUCKC
|
6.6 | IC50 | 3 | — | |
OVVILUUFUJVIDC
|
6.6 | IC50 | 3 | — | |
UVMBLBJOESBFLX
|
6.6 | IC50 | 3 | — | |
XFAPJIVRXVFTKU
|
6.6 | IC50 | 3 | — | |
NFHXWCPPKPQNOC
|
6.6 | IC50 | 3 | — | |
SVCPLCNUNAMBAM
|
6.6 | Kd | 3 | — | |
KHHMGBVQNFVSEB
|
6.6 | IC50 | 3 | — | |
PLFIJQUNUOVBHD
|
6.6 | IC50 | 3 | — | |
ROTGVBIACJDGCI
|
6.6 | IC50 | 3 | — | |
YAPIRWIJBXRQKZ
|
6.6 | IC50 | 3 | — | |
WEHCGVXGVWPFOC
|
6.6 | IC50 | 3 | — | |
FYSXJZQLBHIUOG
|
6.6 | IC50 | 3 | — | |
GHKRMXUUEFNJHM
|
6.6 | IC50 | 3 | — | |
KRXBQXJYEYDJNX
|
6.6 | IC50 | 3 | — | |
UDMVPCPDQWLIDT
|
6.5 | IC50 | 3 | — | |
VULGNLPSROSBRU
|
6.5 | Kd | 3 | — | |
XAYVDATZADKPFK
|
6.5 | IC50 | 3 | — | |
JYSZXOVIWSXAMG
|
6.5 | IC50 | 3 | — | |
ONGTUAKQYUOWAL
|
6.5 | IC50 | 3 | — | |
JHAUMXZLLWOYET
|
6.5 | IC50 | 3 | — | |
KBTNUFQFWHMFFZ
|
6.5 | IC50 | 3 | — | |
NXNKJLOEGWSJGI
|
6.5 | IC50 | 3 | — | |
DIXVQCDOAZRZLS
|
6.5 | IC50 | 3 | — | |
WUFSAKWUUGHJKE
|
6.5 | IC50 | 3 | — | |
JCZHZSQAEMZHAT
|
6.5 | Kd | 3 | — | |
LNXNIMOXVDAPMR
|
6.5 | IC50 | 3 | — | |
YDZZFBICTXOYAW
|
6.5 | IC50 | 3 | — | |
HBXVNIDHYGUGIY
|
6.5 | IC50 | 3 | — | |
XIHFTDUKDIRRKY
|
6.5 | IC50 | 3 | — | |
HHDURAOHKSUNTC
|
6.4 | Kd | 3 | — | |
ZFKSCQNGJJUYMW
|
6.4 | IC50 | 3 | — | |
TZLWATKWJLUXTA
|
6.4 | Kd | 3 | — | |
HYBFJADVMPQZEV
|
6.4 | IC50 | 3 | — |