Target Details
| UniProt AC | P05107 |
|---|---|
| Gene Symbol | ITGB2 |
| Protein Name | Integrin beta-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF23105 (EGF_integrin) PF08725 (Integrin_b_cyt) PF07965 (Integrin_B_tail) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 373
- Clinical molecules 0
- Avg pChEMBL 7.14
KEGG Pathways (21)
- Amoebiasis
- Cell adhesion molecule (CAM) interaction
- Complement and coagulation cascades
- Hippo signaling pathway
- Human T-cell leukemia virus 1 infection
- IgSF CAM signaling
- Integrin signaling
- Legionellosis
- Leishmaniasis
- Leukocyte transendothelial migration
- Malaria
- Natural killer cell mediated cytotoxicity
- Neutrophil extracellular trap formation
- Pertussis
- Phagosome
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Rheumatoid arthritis
- Staphylococcus aureus infection
- Tuberculosis
- Viral myocarditis
Associated Diseases (1)
Active Molecules (373)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CEEYZLMHLBHWRT
|
7.0 | IC50 | 3 | — | |
JVJJYUVCAROHSN
|
7.0 | IC50 | 3 | — | |
UOPLAJAFYJNCFL
|
7.0 | IC50 | 3 | — | |
XGCZRGJUCNQVCO
|
7.0 | IC50 | 3 | — | |
FXYDXLJEJBXFBD
|
6.9 | IC50 | 5 | — | |
LFMVROPXFXRDLY
|
6.9 | IC50 | 3 | — | |
LXPIKCWBQUZGHG
|
6.9 | IC50 | 3 | — | |
ABFZFLPVUIIHIL
|
6.9 | IC50 | 3 | — | |
ACLVTPBNANYOKG
|
6.9 | IC50 | 3 | — | |
CUSLWNBCMONUNY
|
6.9 | IC50 | 3 | — | |
CVAUURCTSNKGEZ
|
6.9 | IC50 | 3 | — | |
FKFWCWLZUOSSNM
|
6.9 | IC50 | 3 | — | |
MPHIYSGHFVGRGH
|
6.9 | IC50 | 3 | — | |
SKOPXHFNQHFUFJ
|
6.9 | IC50 | 3 | — | |
BPJSFBIYRVIFEZ
|
6.9 | IC50 | 3 | — | |
OZDIXXYNNZCRMU
|
6.9 | IC50 | 3 | — | |
BZNCFMHNUSOIAG
|
6.9 | IC50 | 3 | — | |
HHWSDMCKOLNFCZ
|
6.9 | IC50 | 3 | — | |
HVZJOWMEYSKFNV
|
6.9 | IC50 | 3 | — | |
IBJIONZZKQZZDE
|
6.9 | IC50 | 3 | — | |
NCFNEGXOEYXVOP
|
6.9 | IC50 | 3 | — | |
VAATYVLSQSKJGH
|
6.9 | IC50 | 3 | — | |
YDDSCHDADLMSAK
|
6.9 | IC50 | 3 | — | |
YGQRAJLJNWTQJX
|
6.9 | IC50 | 3 | — | |
ZMYOKTHPJKLGOG
|
6.9 | IC50 | 3 | — | |
JAUMKMDGCWUQCV
|
6.8 | IC50 | 3 | — | |
JQZDFLNJNAPFDP
|
6.8 | IC50 | 3 | — | |
QMCLITAQOBPTQP
|
6.8 | IC50 | 3 | — | |
SJUIYCCLDVYYMH
|
6.8 | IC50 | 3 | — | |
STPAECMJMZUXFA
|
6.8 | Kd | 3 | — | |
WPBDKMFHMPORIP
|
6.8 | IC50 | 3 | — | |
GERAUBTWBQPHRK
|
6.8 | IC50 | 3 | — | |
FHJXPRTVVWNFEW
|
6.8 | Kd | 3 | — | |
HROSRSVATNBMRZ
|
6.8 | IC50 | 3 | — | |
MSANEFFUSIOKNH
|
6.8 | IC50 | 3 | — | |
RUJBILLSZGCLSC
|
6.8 | IC50 | 3 | — | |
KLWCZYZPAXGKGD
|
6.8 | IC50 | 3 | — | |
MPPICRKUKRZKSE
|
6.8 | IC50 | 3 | — | |
SQLPKVCMRLUBJT
|
6.8 | IC50 | 3 | — | |
ULOLQJYJZXDFCF
|
6.8 | IC50 | 3 | — | |
VJRMETDTVGHPMG
|
6.8 | IC50 | 3 | — | |
VLAKGWWGUVHWPD
|
6.8 | IC50 | 3 | — | |
FIOKSZYEWJPCQK
|
6.8 | IC50 | 3 | — | |
HKQSYXSKLFYXEZ
|
6.8 | IC50 | 3 | — | |
QPZCYDCQRGXZLP
|
6.8 | IC50 | 3 | — | |
VWDMVVKQHNPLEH
|
6.8 | IC50 | 3 | — | |
APECBVUSSLUJRS
|
6.8 | Kd | 3 | — | |
CFGADNMKHAGYEI
|
6.8 | IC50 | 3 | — | |
JMKWZXFWHSLFSK
|
6.8 | IC50 | 3 | — | |
KMZOHDKTUBGFTI
|
6.8 | IC50 | 3 | — |