Target Details
| UniProt AC | P05107 |
|---|---|
| Gene Symbol | ITGB2 |
| Protein Name | Integrin beta-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF23105 (EGF_integrin) PF08725 (Integrin_b_cyt) PF07965 (Integrin_B_tail) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 373
- Clinical molecules 0
- Avg pChEMBL 7.14
KEGG Pathways (21)
- Amoebiasis
- Cell adhesion molecule (CAM) interaction
- Complement and coagulation cascades
- Hippo signaling pathway
- Human T-cell leukemia virus 1 infection
- IgSF CAM signaling
- Integrin signaling
- Legionellosis
- Leishmaniasis
- Leukocyte transendothelial migration
- Malaria
- Natural killer cell mediated cytotoxicity
- Neutrophil extracellular trap formation
- Pertussis
- Phagosome
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Rheumatoid arthritis
- Staphylococcus aureus infection
- Tuberculosis
- Viral myocarditis
Associated Diseases (1)
Active Molecules (373)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MVRMZEXFMDYXCV
|
7.2 | IC50 | 3 | — | |
SSUCZPFAHCENOP
|
7.2 | IC50 | 3 | — | |
WGYZXTCUEIZSAP
|
7.2 | IC50 | 3 | — | |
WZKOECKNEHAVJL
|
7.2 | IC50 | 3 | — | |
XWTGFUGJJCIZRY
|
7.2 | IC50 | 3 | — | |
ZIHNRIDMLOHFPP
|
7.2 | IC50 | 3 | — | |
MDLWTUYIAFVKGK
|
7.2 | IC50 | 3 | — | |
OCQSLVRRSSLDCT
|
7.2 | IC50 | 3 | — | |
PBWGNAKIFNSLLR
|
7.2 | IC50 | 3 | — | |
XHNFQBYXWHWBKQ
|
7.2 | IC50 | 3 | — | |
BMLUKZUMDLIBNN
|
7.2 | IC50 | 3 | — | |
CEPHCBHONKERLG
|
7.2 | Kd | 3 | — | |
COVPLULNDBDXTN
|
7.2 | IC50 | 3 | — | |
LGJZQZFSGWSQNO
|
7.2 | IC50 | 3 | — | |
OQGNIEVOYVXSHE
|
7.2 | IC50 | 3 | — | |
RINLDUKDNNFJSS
|
7.2 | IC50 | 3 | — | |
UODMRUIEPLWYGA
|
7.2 | Kd | 3 | — | |
KMZGVJHSOHMQRG
|
7.1 | IC50 | 3 | — | |
ACJAZSQRMWXCLM
|
7.1 | IC50 | 3 | — | |
KQGLUKKEGLGGPO
|
7.1 | IC50 | 3 | — | |
QSJHFUJBHHSDHO
|
7.1 | IC50 | 3 | — | |
DLXSYTAQBCLTQI
|
7.1 | IC50 | 3 | — | |
ROCDTGHUIQLNBL
|
7.1 | IC50 | 3 | — | |
DIRSGZLYFCLEDL
|
7.1 | IC50 | 3 | — | |
RLTHAIWBVZSQOO
|
7.1 | IC50 | 3 | — | |
VHDWIPLMGLQQHO
|
7.1 | IC50 | 3 | — | |
FXYDXLJEJBXFBD
|
7.1 | IC50 | 6 | — | |
KRXBQXJYEYDJNX
|
7.1 | IC50 | 3 | — | |
LRABRYURWMXYGU
|
7.1 | IC50 | 3 | — | |
ZBALKPBJFFDXAB
|
7.1 | IC50 | 3 | — | |
BVXBVMYTIQBMPV
|
7.0 | IC50 | 3 | — | |
KRGAECPDXVSJPY
|
7.0 | IC50 | 3 | — | |
OCUFGCYPFDLREE
|
7.0 | IC50 | 3 | — | |
VOAJYNCTUMVQQJ
|
7.0 | IC50 | 3 | — | |
VQVVXSALLAVZRC
|
7.0 | IC50 | 3 | — | |
LUQRKXJPRPZZOI
|
7.0 | IC50 | 3 | — | |
ASEPTZPIYTWOSV
|
7.0 | IC50 | 3 | — | |
DOTRUZSRWNXWJD
|
7.0 | IC50 | 3 | — | |
IOORAGVPEMUXSU
|
7.0 | IC50 | 3 | — | |
LNUHEJIWTOBAQF
|
7.0 | IC50 | 3 | — | |
PODGAZYUFOSBKT
|
7.0 | IC50 | 3 | — | |
XOXBNFKSIDCMFB
|
7.0 | IC50 | 3 | — | |
YSCQEWQIIQUHAR
|
7.0 | IC50 | 3 | — | |
BKXTXBYRPWNSJQ
|
7.0 | IC50 | 3 | — | |
AYCHCVUKHOSWTG
|
7.0 | Kd | 3 | — | |
MGBNIQZDOXDPDU
|
7.0 | IC50 | 3 | — | |
MRALGEXHJHNARS
|
7.0 | IC50 | 3 | — | |
RNOQFAVOZIQTQB
|
7.0 | IC50 | 3 | — | |
RXCDHJANJVJLRC
|
7.0 | IC50 | 3 | — | |
VMYQJXMFOGNDIJ
|
7.0 | IC50 | 3 | — |