Target Details
| UniProt AC | P05107 |
|---|---|
| Gene Symbol | ITGB2 |
| Protein Name | Integrin beta-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF23105 (EGF_integrin) PF08725 (Integrin_b_cyt) PF07965 (Integrin_B_tail) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 373
- Clinical molecules 0
- Avg pChEMBL 7.14
KEGG Pathways (21)
- Amoebiasis
- Cell adhesion molecule (CAM) interaction
- Complement and coagulation cascades
- Hippo signaling pathway
- Human T-cell leukemia virus 1 infection
- IgSF CAM signaling
- Integrin signaling
- Legionellosis
- Leishmaniasis
- Leukocyte transendothelial migration
- Malaria
- Natural killer cell mediated cytotoxicity
- Neutrophil extracellular trap formation
- Pertussis
- Phagosome
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Rheumatoid arthritis
- Staphylococcus aureus infection
- Tuberculosis
- Viral myocarditis
Associated Diseases (1)
Active Molecules (373)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XYTRSSKMVCVZQA
|
7.5 | IC50 | 3 | — | |
ZTROBKLFMPLYHQ
|
7.5 | IC50 | 3 | — | |
WVTSKZKNRPBXCK
|
7.5 | IC50 | 3 | — | |
DPOIZQRENSINPW
|
7.5 | IC50 | 3 | — | |
GLGFUMDYDHOFDP
|
7.5 | IC50 | 3 | — | |
IJHCQZSIRPACKX
|
7.5 | Kd | 3 | — | |
MRWGXKWDMVKCMX
|
7.5 | IC50 | 3 | — | |
CVXOYGQYPVWPFZ
|
7.5 | IC50 | 3 | — | |
YJOIYUZQCBNKOU
|
7.5 | IC50 | 3 | — | |
GVXLMTNNCFPRBM
|
7.5 | IC50 | 3 | — | |
AMEPXQRZUIVGBX
|
7.5 | IC50 | 3 | — | |
VNBHPAJREIIVSS
|
7.5 | IC50 | 3 | — | |
SKCJPAKVOZQNSP
|
7.4 | IC50 | 3 | — | |
GOOVDGYHZXZDFB
|
7.4 | IC50 | 3 | — | |
AIMBUGRSRLAWJW
|
7.4 | IC50 | 3 | — | |
HANCDWQKPIEEQU
|
7.4 | IC50 | 3 | — | |
PZJWSJORJOUILO
|
7.4 | IC50 | 3 | — | |
RGCAVHSBAFLEJX
|
7.4 | Kd | 3 | — | |
TUIWCAJBTHNBBI
|
7.4 | IC50 | 3 | — | |
YPXGDBHQKAJSNY
|
7.4 | Kd | 3 | — | |
QUGRAPNUWRECOX
|
7.4 | IC50 | 3 | — | |
FFZPSNRNURGDLB
|
7.4 | IC50 | 3 | — | |
HTGGAYLWTDOFDK
|
7.4 | IC50 | 3 | — | |
UYUMTQVAGHXLJZ
|
7.4 | IC50 | 3 | — | |
GPGCGKYPWDTDDC
|
7.3 | IC50 | 3 | — | |
HPLNGZWRFIAXQN
|
7.3 | IC50 | 3 | — | |
LQONBFLCEHNJJY
|
7.3 | IC50 | 3 | — | |
VKDICKOLJZIYGR
|
7.3 | IC50 | 3 | — | |
BHEGQCULFWMOJE
|
7.3 | IC50 | 3 | — | |
FMBLPFSVDXVCAX
|
7.3 | Kd | 3 | — | |
UTAAVKMLQCWSFT
|
7.3 | IC50 | 3 | — | |
QIUVOSJLYMTVAE
|
7.3 | IC50 | 5 | — | |
RDDGVDXVIDYSSC
|
7.3 | IC50 | 3 | — | |
UODMRUIEPLWYGA
|
7.3 | Kd | 3 | — | |
VTZOJHBFLMFAIP
|
7.3 | Kd | 3 | — | |
XGCZRGJUCNQVCO
|
7.3 | IC50 | 2 | — | |
IAAIGCGTGAJLIA
|
7.3 | IC50 | 3 | — | |
JBBDDNUWYXTKTL
|
7.3 | IC50 | 3 | — | |
JLATZOOYNDMRMO
|
7.3 | IC50 | 3 | — | |
LAGKCZDXFAJYPU
|
7.3 | IC50 | 3 | — | |
ZKMPUIRFXLMIMW
|
7.3 | IC50 | 3 | — | |
LUWQOLUBBVTNCZ
|
7.3 | IC50 | 3 | — | |
CMVMPRRSIRJGRR
|
7.3 | IC50 | 3 | — | |
CYUHNCVDNNTABN
|
7.3 | Kd | 3 | — | |
VEUANACROFZFPI
|
7.3 | IC50 | 3 | — | |
ZZSDJBZHPJZXBL
|
7.3 | IC50 | 3 | — | |
DEABNERZBCCLOD
|
7.2 | IC50 | 3 | — | |
GRRUUHVYLVKVPJ
|
7.2 | IC50 | 3 | — | |
JDKJXMPWWOENAF
|
7.2 | IC50 | 3 | — | |
JOGGIPBFAFXTJX
|
7.2 | IC50 | 3 | — |