Target Details
| UniProt AC | P05107 |
|---|---|
| Gene Symbol | ITGB2 |
| Protein Name | Integrin beta-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF23105 (EGF_integrin) PF08725 (Integrin_b_cyt) PF07965 (Integrin_B_tail) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 373
- Clinical molecules 0
- Avg pChEMBL 7.14
KEGG Pathways (21)
- Amoebiasis
- Cell adhesion molecule (CAM) interaction
- Complement and coagulation cascades
- Hippo signaling pathway
- Human T-cell leukemia virus 1 infection
- IgSF CAM signaling
- Integrin signaling
- Legionellosis
- Leishmaniasis
- Leukocyte transendothelial migration
- Malaria
- Natural killer cell mediated cytotoxicity
- Neutrophil extracellular trap formation
- Pertussis
- Phagosome
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Rheumatoid arthritis
- Staphylococcus aureus infection
- Tuberculosis
- Viral myocarditis
Associated Diseases (1)
Active Molecules (373)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PKSKMDBFTLPBGD
|
8.0 | IC50 | 3 | — | |
GKORLDUEXWMZDW
|
8.0 | IC50 | 3 | — | |
LXPIKCWBQUZGHG
|
8.0 | IC50 | 3 | — | |
OISQKZHMDXVZKJ
|
8.0 | Kd | 3 | — | |
QQSAZMAJLFVCGT
|
8.0 | IC50 | 3 | — | |
TZLWATKWJLUXTA
|
8.0 | Kd | 3 | — | |
UHTHCCFWRKLUOC
|
8.0 | IC50 | 3 | — | |
UQFJJELMTYQZLF
|
8.0 | Kd | 3 | — | |
ZFUSMHKFXKIZTH
|
8.0 | IC50 | 3 | — | |
PXWKZXMPCCTSLZ
|
8.0 | IC50 | 3 | — | |
PQEXIWGLHFOPDT
|
8.0 | IC50 | 3 | — | |
HCVGIQGOPCGGPD
|
7.9 | IC50 | 3 | — | |
LYDRSMBADUZQIU
|
7.9 | IC50 | 3 | — | |
YIIHVSKSGPYBER
|
7.9 | IC50 | 3 | — | |
MEMSOGHDJLMQDL
|
7.9 | IC50 | 3 | — | |
OHELAVHWEMILBF
|
7.9 | IC50 | 3 | — | |
UNSPTWPYUISLGN
|
7.8 | IC50 | 3 | — | |
WZWKDGGJAXYHLC
|
7.8 | IC50 | 3 | — | |
XYVGXDQZIPFLPB
|
7.8 | IC50 | 3 | — | |
UAGCAOFGPDUCEN
|
7.8 | IC50 | 3 | — | |
IAAIGCGTGAJLIA
|
7.8 | IC50 | 3 | — | |
WBSXKVRTVMHGNY
|
7.8 | IC50 | 3 | — | |
GKGJFUXSTSUKPB
|
7.7 | Kd | 2 | — | |
HXFLTJZCIRRAHJ
|
7.7 | IC50 | 3 | — | |
NPMNYUOXEKFFIQ
|
7.7 | IC50 | 3 | — | |
QIHAPYRUKBWYGW
|
7.7 | IC50 | 3 | — | |
BODOXPRBLCFXNR
|
7.7 | IC50 | 3 | — | |
CWQGLTCXNRXUQD
|
7.7 | Kd | 3 | — | |
FOXOPJJICTTZEU
|
7.7 | IC50 | 3 | — | |
FVEAFWBHBUVJQZ
|
7.7 | IC50 | 3 | — | |
MLYREBCRTPGARB
|
7.7 | Kd | 3 | — | |
MYIHWAVPLWUTSA
|
7.7 | Kd | 3 | — | |
SWIQOJQBTDWCRB
|
7.7 | IC50 | 3 | — | |
WVCQICGGXLHQQZ
|
7.7 | IC50 | 3 | — | |
NXNKJLOEGWSJGI
|
7.7 | IC50 | 3 | — | |
LBFPLUWTLKUUCU
|
7.7 | IC50 | 3 | — | |
OSHCCAHIHYVBQE
|
7.7 | IC50 | 3 | — | |
FJNJHZQMQRVZEE
|
7.6 | IC50 | 3 | — | |
ZTKAYKYKKPDCAJ
|
7.6 | IC50 | 3 | — | |
AQMLUIURUPLBCR
|
7.6 | IC50 | 3 | — | |
MWKSRKSEWLRPBL
|
7.6 | Kd | 1075 | — | |
WVKIRPXFXBGIEJ
|
7.6 | IC50 | 3 | — | |
UIQHPJBLRPBJON
|
7.6 | IC50 | 3 | — | |
QNPSGQWAWDUUBG
|
7.6 | IC50 | 3 | — | |
WHGBQVUQKROPLI
|
7.6 | IC50 | 3 | — | |
XEKXLTGSRAVVJK
|
7.6 | IC50 | 3 | — | |
JFOZKMSJYSPYLN
|
7.6 | IC50 | 3 | — | |
GWKUQIDUBUTSSN
|
7.6 | IC50 | 3 | — | |
WMECQBYXSNEKHN
|
7.6 | IC50 | 3 | — | |
CYHYOQQJILLXPV
|
7.6 | IC50 | 3 | — |