Target Details
| UniProt AC | P05107 |
|---|---|
| Gene Symbol | ITGB2 |
| Protein Name | Integrin beta-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF23105 (EGF_integrin) PF08725 (Integrin_b_cyt) PF07965 (Integrin_B_tail) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 373
- Clinical molecules 0
- Avg pChEMBL 7.14
KEGG Pathways (21)
- Amoebiasis
- Cell adhesion molecule (CAM) interaction
- Complement and coagulation cascades
- Hippo signaling pathway
- Human T-cell leukemia virus 1 infection
- IgSF CAM signaling
- Integrin signaling
- Legionellosis
- Leishmaniasis
- Leukocyte transendothelial migration
- Malaria
- Natural killer cell mediated cytotoxicity
- Neutrophil extracellular trap formation
- Pertussis
- Phagosome
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Rheumatoid arthritis
- Staphylococcus aureus infection
- Tuberculosis
- Viral myocarditis
Associated Diseases (1)
Active Molecules (373)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SVJJYZFYKBOVBA
|
10.0 | IC50 | 3 | — | |
VORCYKUSPCBIIJ
|
9.5 | IC50 | 3 | — | |
AXSOGTWJBSDWJQ
|
9.4 | IC50 | 3 | — | |
CAESXWPQYVXWFJ
|
9.3 | IC50 | 3 | — | |
RCIAZGDKPJKNPZ
|
9.3 | IC50 | 3 | — | |
URZCVPKXOJQTLC
|
9.3 | IC50 | 3 | — | |
AXSOGTWJBSDWJQ
|
9.2 | IC50 | 3 | — | |
IVAMLBGGCGJJFO
|
9.1 | IC50 | 3 | — | |
FEEFNAKFIFJCIA
|
9.0 | IC50 | 3 | — | |
BAHKPHNZYOKPQK
|
8.8 | IC50 | 3 | — | |
DMEDNZSJTBCBCR
|
8.8 | IC50 | 3 | — | |
VDABXUWSEUQIIC
|
8.8 | IC50 | 3 | — | |
KLSZVPNVFKKIRD
|
8.8 | IC50 | 3 | — | |
DZYZAGBAGWPMOE
|
8.7 | IC50 | 3 | — | |
FZYXWDXHAVNVET
|
8.7 | IC50 | 3 | — | |
SLISYJFUVRUCKA
|
8.7 | IC50 | 3 | — | |
VEYUKVJMTNXXSF
|
8.7 | IC50 | 3 | — | |
URZCVPKXOJQTLC
|
8.6 | IC50 | 3 | — | |
VQFPBCXPBVPOKI
|
8.6 | IC50 | 3 | — | |
ZRIKDHLPCRURPX
|
8.6 | IC50 | 3 | — | |
WBSXKVRTVMHGNY
|
8.5 | IC50 | 3 | — | |
YCCWPJKUJHZBMA
|
8.5 | IC50 | 3 | — | |
DMEDNZSJTBCBCR
|
8.5 | IC50 | 3 | — | |
VHJSCKJBRABOFP
|
8.5 | IC50 | 3 | — | |
VHJSCKJBRABOFP
|
8.5 | IC50 | 3 | — | |
ONDASBAVURIEBH
|
8.4 | IC50 | 3 | — | |
LLDYORSLNIEEGL
|
8.4 | IC50 | 3 | — | |
AIXJUFNJLMLMNA
|
8.4 | IC50 | 3 | — | |
DZYZAGBAGWPMOE
|
8.4 | IC50 | 3 | — | |
LMKUPFOQNQUVLK
|
8.4 | IC50 | 3 | — | |
BWZVEDBBEOJBAG
|
8.4 | IC50 | 3 | — | |
HMHSDFNVSYBUNO
|
8.3 | IC50 | 3 | — | |
PEMCDDOYUUHYRN
|
8.3 | IC50 | 3 | — | |
QCABIGRYALYSAQ
|
8.3 | IC50 | 3 | — | |
NVVGCQABIHSJSQ
|
8.3 | IC50 | 6 | — | |
DMTPQLIVNVZBPV
|
8.3 | IC50 | 3 | — | |
BWIPTTGMQIMVBA
|
8.2 | IC50 | 3 | — | |
HSJWUDLCVCZMAZ
|
8.2 | IC50 | 3 | — | |
MCNILTQMLDZWKD
|
8.2 | IC50 | 3 | — | |
PZFCKINMYJYVSY
|
8.2 | IC50 | 3 | — | |
SYGPJZDISKKEIV
|
8.2 | IC50 | 3 | — | |
WCVPXAWSKHNQTH
|
8.2 | IC50 | 3 | — | |
ZBDUGVCGVJAVEM
|
8.2 | IC50 | 3 | — | |
GYELUVCNTNLZSS
|
8.1 | IC50 | 3 | — | |
QPWDZBBZIVDASP
|
8.1 | IC50 | 3 | — | |
XEANMEGOYUBDBY
|
8.1 | IC50 | 3 | — | |
AVUBMOWMBYBZOK
|
8.1 | Kd | 3 | — | |
FOBMOHYBRJMHEY
|
8.1 | IC50 | 3 | — | |
QOPHPRIAHZKBGU
|
8.1 | IC50 | 3 | — | |
VZSWCQOTQDDSHT
|
8.0 | IC50 | 3 | — |