Target Details
| UniProt AC | P05106 |
|---|---|
| Gene Symbol | ITGB3 |
| Protein Name | Integrin beta-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07974 (EGF_2) PF23105 (EGF_integrin) PF18372 (I-EGF_1) PF08725 (Integrin_b_cyt) PF07965 (Integrin_B_tail) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 2,474
- Clinical molecules 0
- Avg pChEMBL 7.74
KEGG Pathways (26)
- Arrhythmogenic right ventricular cardiomyopathy
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Efferocytosis
- Fluid shear stress and atherosclerosis
- Focal adhesion
- Hematopoietic cell lineage
- Herpes simplex virus 1 infection
- Hormone signaling
- Human cytomegalovirus infection
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- MicroRNAs in cancer
- Neutrophil extracellular trap formation
- Osteoclast differentiation
- PI3K-Akt signaling pathway
- Phagosome
- Platelet activation
- Proteoglycans in cancer
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Thyroid hormone signaling pathway
- Virion - Herpesvirus
Associated Diseases (6)
Active Molecules (2,474)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XPIJPDHIAQUTCT
|
8.8 | IC50 | 2 | — | |
DSVRSYVZAMHQET
|
8.8 | IC50 | 2 | — | |
QYKHSZCOMAXNCJ
|
8.8 | IC50 | 6 | — | |
UMSKKXXFLOGWFX
|
8.8 | IC50 | 4 | — | |
WCZAIWWFRSMLCO
|
8.8 | Ki | 2 | — | |
WFYXHJWMKRUJRV
|
8.8 | IC50 | 2 | — | |
YJVQTPGCEVENKR
|
8.8 | IC50 | 4 | — | |
GFBIYISHVPCCGE
|
8.8 | Ki | 2 | — | |
HNJOHJBYQFWLOL
|
8.8 | IC50 | 2 | — | |
HRDIZOQCGGRTPM
|
8.8 | IC50 | 2 | — | |
IALCADUNFMACEG
|
8.8 | IC50 | 3 | — | |
KNVMGBKMZYKHLR
|
8.8 | IC50 | 5 | — | |
LDHLQPMIUKAPSY
|
8.8 | IC50 | 5 | — | |
LPWSHOGTPIIOBC
|
8.8 | IC50 | 5 | — | |
MDAJFZIQBMXEKL
|
8.8 | IC50 | 2 | — | |
OCFMIMLTAYUZOV
|
8.8 | IC50 | 2 | — | |
PEFBVOAICYLSAF
|
8.8 | IC50 | 8 | — | |
PMZAMOSBWUCNBG
|
8.8 | IC50 | 5 | — | |
RRYMQSFBOJUJEI
|
8.8 | IC50 | 2 | — | |
YRIJMZJTWNXHBY
|
8.8 | IC50 | 2 | — | |
MXSJSHDIEDILST
|
8.8 | IC50 | 4 | — | |
OLQOZUUGUUUOMF
|
8.8 | IC50 | 3 | — | |
FXBDPMBWPSLDQZ
|
8.7 | Kd | 2 | — | |
LAKQAEHCCWPUIS
|
8.7 | IC50 | 3 | — | |
LMFGOELGOHYQNF
|
8.7 | IC50 | 2 | — | |
QTPSIFSNODGQLH
|
8.7 | IC50 | 2 | — | |
URUQCDJWYNLAGR
|
8.7 | IC50 | 2 | — | |
ZMVBGJMBSDZOLI
|
8.7 | IC50 | 2 | — | |
BDICDHJCLYIIQR
|
8.7 | IC50 | 2 | — | |
BIIVGTIHIPJAHG
|
8.7 | Ki | 2 | — | |
HOXCYDQJLHZQJW
|
8.7 | IC50 | 2 | — | |
MDGSJXNNVZDXCV
|
8.7 | IC50 | 2 | — | |
XGBKKOOTEJXBQX
|
8.7 | IC50 | 2 | — | |
XIDSVQGXAGLHHT
|
8.7 | IC50 | 2 | — | |
ZPRQEMGTRXGZPE
|
8.7 | IC50 | 4 | — | |
LTTIHWWYCLBIKC
|
8.7 | IC50 | 3 | — | |
CGSCSHWTEZCGFQ
|
8.7 | IC50 | 2 | — | |
CQUBDSKDQMDXPM
|
8.7 | Ki | 2 | — | |
CUWCAWQFVBJCMK
|
8.7 | IC50 | 2 | — | |
CVAFKDVZZYLXCZ
|
8.7 | IC50 | 6 | — | |
DTLIDYQJLOBQPK
|
8.7 | IC50 | 2 | — | |
FUKBQDRZNSNAOO
|
8.7 | IC50 | 2 | — | |
GITHMVUAHBUYNI
|
8.7 | IC50 | 2 | — | |
HLCQRNGEUFKGFI
|
8.7 | IC50 | 3 | — | |
IEPGKKVDERKGDN
|
8.7 | IC50 | 2 | — | |
JCZHWFZLHYLGEG
|
8.7 | Ki | 2 | — | |
JKEXIYXWHPGQLX
|
8.7 | IC50 | 2 | — | |
JUCUUAVAOJAIHU
|
8.7 | Ki | 2 | — | |
JWDZKECSZGMGRE
|
8.7 | IC50 | 2 | — | |
LZPPYUNNJYIBTG
|
8.7 | IC50 | 2 | — |