Target Details
| UniProt AC | P05106 |
|---|---|
| Gene Symbol | ITGB3 |
| Protein Name | Integrin beta-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07974 (EGF_2) PF23105 (EGF_integrin) PF18372 (I-EGF_1) PF08725 (Integrin_b_cyt) PF07965 (Integrin_B_tail) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 2,474
- Clinical molecules 0
- Avg pChEMBL 7.74
KEGG Pathways (26)
- Arrhythmogenic right ventricular cardiomyopathy
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Efferocytosis
- Fluid shear stress and atherosclerosis
- Focal adhesion
- Hematopoietic cell lineage
- Herpes simplex virus 1 infection
- Hormone signaling
- Human cytomegalovirus infection
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- MicroRNAs in cancer
- Neutrophil extracellular trap formation
- Osteoclast differentiation
- PI3K-Akt signaling pathway
- Phagosome
- Platelet activation
- Proteoglycans in cancer
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Thyroid hormone signaling pathway
- Virion - Herpesvirus
Associated Diseases (6)
Active Molecules (2,474)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MSGZVCWOFQOMDA
|
8.9 | IC50 | 2 | — | |
NYFWULSTXJLATO
|
8.9 | IC50 | 3 | — | |
ZSYFEFOBOJYQCG
|
8.9 | IC50 | 2 | — | |
KAMSHMVKMNHYHX
|
8.9 | IC50 | 3 | — | |
LWCKRBHIZLBAFM
|
8.9 | IC50 | 2 | — | |
BHDLQEOXHBGVFT
|
8.9 | IC50 | 2 | — | |
DTNKZZXZAPCYPT
|
8.9 | IC50 | 3 | — | |
FQTMTTZENZSMQU
|
8.9 | IC50 | 2 | — | |
HUIGGCYPYURGFA
|
8.9 | Ki | 2 | — | |
MHGHYXQIIPLSCN
|
8.9 | Ki | 2 | — | |
XFNZYXKVDFJAFI
|
8.9 | IC50 | 6 | — | |
ZEEBGVAVQWCFLT
|
8.9 | IC50 | 3 | — | |
ZXCIVKBMKMAQIS
|
8.9 | Kd | 2 | — | |
RTHTZKFWJRGDKZ
|
8.9 | IC50 | 4 | — | |
YVGFDNFQFUSINK
|
8.9 | IC50 | 3 | — | |
AEFPUSNNPXBSKD
|
8.8 | IC50 | 3 | — | |
CDIQJJMJTFHODD
|
8.8 | IC50 | 2 | — | |
DKCBOEVMYBPSHB
|
8.8 | Ki | 2 | — | |
IJIQSYZFWKZVHL
|
8.8 | Ki | 2 | — | |
PLPDPJUYPOKPOK
|
8.8 | IC50 | 2 | — | |
QKCFDPUKGKJIML
|
8.8 | IC50 | 7 | — | |
RGPCXWUHNLAAMX
|
8.8 | IC50 | 2 | — | |
SBROZGGPOIEKJM
|
8.8 | IC50 | 2 | — | |
UHIXYIGWNOLNHI
|
8.8 | IC50 | 2 | — | |
VYKRADAUJUCJRE
|
8.8 | Kd | 2 | — | |
XHPZRPHYLGZLTO
|
8.8 | IC50 | 5 | — | |
XKXMEMPIHRKAQX
|
8.8 | IC50 | 5 | — | |
YTKGKCKBCJZBIX
|
8.8 | IC50 | 4 | — | |
YWCFKVFIEXQDJL
|
8.8 | IC50 | 3 | — | |
DRAZWXSJTKLZTP
|
8.8 | IC50 | 2 | — | |
XNBNFFZMGGWODG
|
8.8 | IC50 | 4 | — | |
AQDWTTAFCBSSHY
|
8.8 | Ki | 2 | — | |
ASDVCZXKBVVZII
|
8.8 | Ki | 2 | — | |
CJDLVBMPCKYVJE
|
8.8 | IC50 | 2 | — | |
FLHQMWMGVZBTDD
|
8.8 | IC50 | 2 | — | |
FZBGGWKHCWPGOF
|
8.8 | IC50 | 2 | — | |
GARROJJZLJSGSW
|
8.8 | IC50 | 4 | — | |
HRJYJLGVTFNBBO
|
8.8 | IC50 | 2 | — | |
IXYJRFZTWSBREE
|
8.8 | IC50 | 2 | — | |
JARATYKMRJHXBN
|
8.8 | IC50 | 2 | — | |
JTQSBYUBJLIDAK
|
8.8 | IC50 | 5 | — | |
NMCRMSDRKRSKLI
|
8.8 | Ki | 2 | — | |
OPDQGEZDVZHFLO
|
8.8 | Ki | 2 | — | |
RIDAEANAMCADNQ
|
8.8 | Ki | 2 | — | |
UJAJKKVATBUTAU
|
8.8 | IC50 | 2 | — | |
VMCREQBBFYDYNW
|
8.8 | Ki | 2 | — | |
ZMNAHKMVEDGEFB
|
8.8 | IC50 | 2 | — | |
DGHLGBHZIKLZQQ
|
8.8 | IC50 | 2 | — | |
FNKFUBZIIVXPMV
|
8.8 | IC50 | 2 | — | |
UBSZHEXPLSECRR
|
8.8 | IC50 | 3 | — |