Target Details
| UniProt AC | P05106 |
|---|---|
| Gene Symbol | ITGB3 |
| Protein Name | Integrin beta-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07974 (EGF_2) PF23105 (EGF_integrin) PF18372 (I-EGF_1) PF08725 (Integrin_b_cyt) PF07965 (Integrin_B_tail) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 2,474
- Clinical molecules 0
- Avg pChEMBL 7.74
KEGG Pathways (26)
- Arrhythmogenic right ventricular cardiomyopathy
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Efferocytosis
- Fluid shear stress and atherosclerosis
- Focal adhesion
- Hematopoietic cell lineage
- Herpes simplex virus 1 infection
- Hormone signaling
- Human cytomegalovirus infection
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- MicroRNAs in cancer
- Neutrophil extracellular trap formation
- Osteoclast differentiation
- PI3K-Akt signaling pathway
- Phagosome
- Platelet activation
- Proteoglycans in cancer
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Thyroid hormone signaling pathway
- Virion - Herpesvirus
Associated Diseases (6)
Active Molecules (2,474)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QVMBSOXHMYDQRA
|
9.0 | IC50 | 2 | — | |
QXTJTOIUBFOZEN
|
9.0 | IC50 | 2 | — | |
UOBZVUNLYKJTSH
|
9.0 | IC50 | 2 | — | |
VIMZEKZBMIICSS
|
9.0 | IC50 | 2 | — | |
VYLURKBKHHADFJ
|
9.0 | IC50 | 2 | — | |
XJRPJRUXGLBKPY
|
9.0 | IC50 | 2 | — | |
XLDVJVWIKCPJPM
|
9.0 | IC50 | 2 | — | |
XUISHROIRBHOIM
|
9.0 | IC50 | 4 | — | |
YEEBBNWKQGDACU
|
9.0 | IC50 | 3 | — | |
YTROSQIPEKDADK
|
9.0 | IC50 | 2 | — | |
YULSCDVUYRTZCA
|
9.0 | IC50 | 2 | — | |
ZCCMELPMDDSRHL
|
9.0 | IC50 | 2 | — | |
NUWUKVFQPXUSBR
|
9.0 | IC50 | 2 | — | |
DHLKXUDAGRMGLV
|
9.0 | IC50 | 2 | — | |
GFGRBKXJVOAPLF
|
9.0 | IC50 | 3 | — | |
KIOVJZCZUNJXQB
|
9.0 | IC50 | 3 | — | |
OUOJYIATFPJDBV
|
9.0 | IC50 | 2 | — | |
PDZBKVNASRLHEK
|
9.0 | IC50 | 2 | — | |
POHCCPZJODTAKF
|
9.0 | IC50 | 3 | — | |
QJYMHIUQOMYZKT
|
9.0 | IC50 | 2 | — | |
SMMNOJYHMMCWQP
|
9.0 | IC50 | 5 | — | |
VYVQCVGITLHGKO
|
9.0 | IC50 | 2 | — | |
WPRZWONATNXRPZ
|
9.0 | IC50 | 3 | — | |
WVUZBVPGGBTRTK
|
9.0 | IC50 | 2 | — | |
XYIBYEZXQWCSGR
|
9.0 | IC50 | 2 | — | |
YLFFZEQHDMFOEC
|
9.0 | Kd | 2 | — | |
YTAHOLPCQRGOAW
|
9.0 | IC50 | 5 | — | |
YURBLSCQXZUCIK
|
9.0 | IC50 | 2 | — | |
NXKFHFCWTSGLDC
|
8.9 | IC50 | 4 | — | |
PDZPUQQVGSDNOJ
|
8.9 | IC50 | 3 | — | |
VKBWHHDLZWUCHL
|
8.9 | IC50 | 2 | — | |
BCZJAKMDVNIASQ
|
8.9 | IC50 | 3 | — | |
SFCYQXKSWPPSIX
|
8.9 | IC50 | 4 | — | |
AZPMNBDRAVVHOL
|
8.9 | IC50 | 3 | — | |
CTHYLBXDQVAGEJ
|
8.9 | IC50 | 5 | — | |
GFFKBNVAAGGGNS
|
8.9 | IC50 | 3 | — | |
IETWETOHQHTRGK
|
8.9 | IC50 | 2 | — | |
MIFZAPHWMCAHQZ
|
8.9 | IC50 | 5 | — | |
MLRWZTLJAPFEKW
|
8.9 | IC50 | 3 | — | |
MLRWZTLJAPFEKW
|
8.9 | IC50 | 2 | — | |
QXAYHAXWXRCLTG
|
8.9 | IC50 | 4 | — | |
RYILTXKXDOUWET
|
8.9 | IC50 | 2 | — | |
UQYFVSMGEHOGBU
|
8.9 | IC50 | 5 | — | |
VZYNONIAPDJFNO
|
8.9 | IC50 | 2 | — | |
YKGDXSKYOQQGRW
|
8.9 | IC50 | 3 | — | |
ZKGCNKVDPWEGNL
|
8.9 | IC50 | 3 | — | |
BIAYEWRLSABXRF
|
8.9 | IC50 | 3 | — | |
BQTUWUXJPAYSPB
|
8.9 | Ki | 2 | — | |
HAVKADYFCFXNIM
|
8.9 | IC50 | 4 | — | |
IYENZWRUEZBYIV
|
8.9 | IC50 | 2 | — |