Target Details
| UniProt AC | P05106 |
|---|---|
| Gene Symbol | ITGB3 |
| Protein Name | Integrin beta-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07974 (EGF_2) PF23105 (EGF_integrin) PF18372 (I-EGF_1) PF08725 (Integrin_b_cyt) PF07965 (Integrin_B_tail) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 2,474
- Clinical molecules 0
- Avg pChEMBL 7.74
KEGG Pathways (26)
- Arrhythmogenic right ventricular cardiomyopathy
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Efferocytosis
- Fluid shear stress and atherosclerosis
- Focal adhesion
- Hematopoietic cell lineage
- Herpes simplex virus 1 infection
- Hormone signaling
- Human cytomegalovirus infection
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- MicroRNAs in cancer
- Neutrophil extracellular trap formation
- Osteoclast differentiation
- PI3K-Akt signaling pathway
- Phagosome
- Platelet activation
- Proteoglycans in cancer
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Thyroid hormone signaling pathway
- Virion - Herpesvirus
Associated Diseases (6)
Active Molecules (2,474)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XAHWDFRDQNVXQX
|
9.1 | IC50 | 2 | — | |
YCBAFTWBMGUKQE
|
9.1 | IC50 | 2 | — | |
AHZHHMWUUGETMN
|
9.1 | IC50 | 3 | — | |
KEYWFOSYJDAKCT
|
9.1 | IC50 | 2 | — | |
PSZYZEZKPQGGPA
|
9.1 | IC50 | 6 | — | |
LDHLQPMIUKAPSY
|
9.1 | IC50 | 4 | — | |
AIBKMZWFGWJRQW
|
9.1 | IC50 | 3 | — | |
BOPPVVPCLIACBR
|
9.1 | IC50 | 2 | — | |
BPFSDEAWEWNYMO
|
9.1 | IC50 | 2 | — | |
POHCCPZJODTAKF
|
9.1 | IC50 | 3 | — | |
QHSKOAKVMQHGPS
|
9.1 | IC50 | 3 | — | |
VWXQFGQQZYTQPI
|
9.1 | IC50 | 2 | — | |
WVOZQEYNBBHACY
|
9.1 | IC50 | 2 | — | |
XCTHUNKHDUMJGV
|
9.1 | IC50 | 2 | — | |
BPBHTITUTUZWBT
|
9.0 | IC50 | 3 | — | |
KAVRMLREXXGTPY
|
9.0 | IC50 | 3 | — | |
KNVMGBKMZYKHLR
|
9.0 | IC50 | 4 | — | |
QYKHSZCOMAXNCJ
|
9.0 | IC50 | 5 | — | |
RZYRWEAZPQSSKX
|
9.0 | IC50 | 5 | — | |
ZQAQMOMRTYIDJU
|
9.0 | IC50 | 4 | — | |
AFEBUYQIVROWSL
|
9.0 | IC50 | 3 | — | |
NRXYMNJDCGQEHP
|
9.0 | IC50 | 2 | — | |
PCSAMHIZFOPKDJ
|
9.0 | IC50 | 3 | — | |
VJTDBRLHPYYFBZ
|
9.0 | IC50 | 2 | — | |
FCUCMIIVLCLREX
|
9.0 | IC50 | 3 | — | |
NIGWPUUZRHIDKJ
|
9.0 | IC50 | 3 | — | |
IFUROQAKNZUNFY
|
9.0 | IC50 | 5 | — | |
UMFVUEYVEGNPTM
|
9.0 | IC50 | 3 | — | |
ANCHZQJTSKHDFM
|
9.0 | IC50 | 2 | — | |
BEOOWKDNVJKISL
|
9.0 | IC50 | 3 | — | |
BGZXFBKQLANYBE
|
9.0 | IC50 | 2 | — | |
BNTMUQHWJSORQO
|
9.0 | IC50 | 3 | — | |
BSNWAPOUYOPCPS
|
9.0 | IC50 | 2 | — | |
CNNXQMKKHGGQNP
|
9.0 | Ki | 2 | — | |
CYIAZAFUQCTLTE
|
9.0 | IC50 | 2 | — | |
DKSFLHZSAWZIDR
|
9.0 | IC50 | 2 | — | |
DXNCFWHJVOGGRD
|
9.0 | IC50 | 2 | — | |
GDEQKRGKHZOXGD
|
9.0 | IC50 | 8 | — | |
IFDIAYNOLNAOOF
|
9.0 | Ki | 2 | — | |
JTGRZJZVZNGYOK
|
9.0 | IC50 | 2 | — | |
MXVQXMBMRJIIHT
|
9.0 | IC50 | 2 | — | |
OCNALRIBAIFGLP
|
9.0 | IC50 | 3 | — | |
OSKMUZRGKURIOY
|
9.0 | Ki | 2 | — | |
PSWDFAPCKFYFPG
|
9.0 | IC50 | 2 | — | |
PTZKOSOAVVRMBX
|
9.0 | IC50 | 2 | — | |
PZAMXSCMHJPGFV
|
9.0 | IC50 | 3 | — | |
QFUAOXPDMSSGEO
|
9.0 | IC50 | 3 | — | |
QGOXLUXYLLZODC
|
9.0 | IC50 | 3 | — | |
QJTMDUFVKLGAAJ
|
9.0 | IC50 | 2 | — | |
QTBFGJFGHGTDRF
|
9.0 | IC50 | 8 | — |