Target Details
| UniProt AC | P05106 |
|---|---|
| Gene Symbol | ITGB3 |
| Protein Name | Integrin beta-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07974 (EGF_2) PF23105 (EGF_integrin) PF18372 (I-EGF_1) PF08725 (Integrin_b_cyt) PF07965 (Integrin_B_tail) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 2,474
- Clinical molecules 0
- Avg pChEMBL 7.74
KEGG Pathways (26)
- Arrhythmogenic right ventricular cardiomyopathy
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Efferocytosis
- Fluid shear stress and atherosclerosis
- Focal adhesion
- Hematopoietic cell lineage
- Herpes simplex virus 1 infection
- Hormone signaling
- Human cytomegalovirus infection
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- MicroRNAs in cancer
- Neutrophil extracellular trap formation
- Osteoclast differentiation
- PI3K-Akt signaling pathway
- Phagosome
- Platelet activation
- Proteoglycans in cancer
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Thyroid hormone signaling pathway
- Virion - Herpesvirus
Associated Diseases (6)
Active Molecules (2,474)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SLTMEZLQPRTTBL
|
9.2 | IC50 | 3 | — | |
VYTWTVISEPFYEI
|
9.2 | IC50 | 2 | — | |
NEEFZJDFXACOOY
|
9.2 | IC50 | 4 | — | |
OKEKRFLAQTYOCR
|
9.2 | IC50 | 3 | — | |
OSWCPUORIOBICX
|
9.2 | IC50 | 2 | — | |
SQIDFFKYMURYAR
|
9.2 | IC50 | 2 | — | |
HIASMCVWLMTBEO
|
9.2 | IC50 | 2 | — | |
UQEWVVUNGPKKKR
|
9.2 | IC50 | 6 | — | |
YYMWWKGGQOZSCP
|
9.2 | IC50 | 2 | — | |
DKCBOEVMYBPSHB
|
9.2 | Ki | 2 | — | |
DRZSFOQHHTVBQV
|
9.2 | Ki | 2 | — | |
HUIVUZCGJQLTSS
|
9.2 | IC50 | 3 | — | |
HWQHXIKXIJDPTP
|
9.2 | IC50 | 2 | — | |
IKALVLPAIVXDBO
|
9.2 | IC50 | 3 | — | |
KCPZTHQHJHVUCK
|
9.2 | IC50 | 3 | — | |
KZUKILQARHOBHB
|
9.2 | IC50 | 2 | — | |
LIFIBSDQAZPDID
|
9.2 | IC50 | 4 | — | |
NXFFLBNDPLJURV
|
9.2 | IC50 | 2 | — | |
OHKIVHLQMSGSHE
|
9.2 | IC50 | 2 | — | |
OSNKDBJRGIQKQV
|
9.2 | IC50 | 3 | — | |
PUNZTUWXCLUSNO
|
9.2 | IC50 | 2 | — | |
XAULKEKKUDCLCD
|
9.2 | IC50 | 2 | — | |
YGPMFNZQEVAKBT
|
9.2 | IC50 | 2 | — | |
FPSTULSQRYACMJ
|
9.1 | IC50 | 3 | — | |
HOWZBTKZCUTFCU
|
9.1 | IC50 | 2 | — | |
HSACVEKFGJAKFH
|
9.1 | IC50 | 3 | — | |
ZIYZOTDZIZBOGY
|
9.1 | IC50 | 2 | — | |
CKABJNNBXOFZHJ
|
9.1 | IC50 | 2 | — | |
FUBVRQRCBDJFQQ
|
9.1 | IC50 | 6 | — | |
LJKWPNDKPDWWIA
|
9.1 | IC50 | 4 | — | |
ZCECQUACUYXKTJ
|
9.1 | IC50 | 2 | — | |
LWHWQLNSWIQIMG
|
9.1 | IC50 | 4 | — | |
NGWFKQKKCNUAJQ
|
9.1 | IC50 | 3 | — | |
AKOSSGWXDCGWFL
|
9.1 | IC50 | 4 | — | |
BRCOMQAFGDHUIK
|
9.1 | IC50 | 2 | — | |
BZPNVJGCQPADST
|
9.1 | IC50 | 3 | — | |
CKSXICJFAQGSNU
|
9.1 | IC50 | 2 | — | |
GSUDEEPNSDSFMO
|
9.1 | IC50 | 2 | — | |
HVLKUEZLWREEFF
|
9.1 | IC50 | 2 | — | |
ISFSENBRVGRPMH
|
9.1 | IC50 | 2 | — | |
NXLUFIUFDMMQQF
|
9.1 | IC50 | 3 | — | |
PTLBVOXYOSUBEO
|
9.1 | IC50 | 2 | — | |
QCJUNYWAVPPVAY
|
9.1 | IC50 | 3 | — | |
SDUQEHZORCVRMT
|
9.1 | IC50 | 2 | — | |
VHKHAQYPTPVIAP
|
9.1 | IC50 | 3 | — | |
VSGFRHHVICROBS
|
9.1 | IC50 | 2 | — | |
YDHAGPCZRFQPOI
|
9.1 | IC50 | 6 | — | |
YSHCUQUSNSOANU
|
9.1 | IC50 | 3 | — | |
ZMKLPAJURKFWIQ
|
9.1 | IC50 | 5 | — | |
FIEWTBHPTPMJPY
|
9.1 | IC50 | 2 | — |