Target Details
| UniProt AC | P05106 |
|---|---|
| Gene Symbol | ITGB3 |
| Protein Name | Integrin beta-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07974 (EGF_2) PF23105 (EGF_integrin) PF18372 (I-EGF_1) PF08725 (Integrin_b_cyt) PF07965 (Integrin_B_tail) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 2,474
- Clinical molecules 0
- Avg pChEMBL 7.74
KEGG Pathways (26)
- Arrhythmogenic right ventricular cardiomyopathy
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Efferocytosis
- Fluid shear stress and atherosclerosis
- Focal adhesion
- Hematopoietic cell lineage
- Herpes simplex virus 1 infection
- Hormone signaling
- Human cytomegalovirus infection
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- MicroRNAs in cancer
- Neutrophil extracellular trap formation
- Osteoclast differentiation
- PI3K-Akt signaling pathway
- Phagosome
- Platelet activation
- Proteoglycans in cancer
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Thyroid hormone signaling pathway
- Virion - Herpesvirus
Associated Diseases (6)
Active Molecules (2,474)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XRFHJLOFJUFLJB
|
9.3 | IC50 | 2 | — | |
KBRCQTXEFPMTDE
|
9.3 | IC50 | 2 | — | |
RXTBIRIYBNVLMP
|
9.3 | IC50 | 2 | — | |
YUYFHARZOUACDE
|
9.3 | IC50 | 2 | — | |
CNSDHPHNXQALLW
|
9.3 | IC50 | 2 | — | |
CPOXHOJHCZSECN
|
9.3 | Ki | 2 | — | |
KZYWKHUJTXLNJM
|
9.3 | IC50 | 5 | — | |
MLRJOXSFEYKLLF
|
9.3 | Ki | 4 | — | |
OLCXJKREUBWULJ
|
9.3 | IC50 | 2 | — | |
OMISPTOHCAHRQR
|
9.3 | IC50 | 3 | — | |
PRILHZGEUSLPLF
|
9.3 | IC50 | 2 | — | |
RBSUHEPCSZKVSP
|
9.3 | IC50 | 4 | — | |
WEXQBLSMARBRMG
|
9.3 | IC50 | 6 | — | |
WWUJBWRZVJNABY
|
9.3 | IC50 | 3 | — | |
XVIKFFNGSSURCJ
|
9.3 | IC50 | 3 | — | |
XVIKFFNGSSURCJ
|
9.3 | IC50 | 2 | — | |
YRCDKPLXZYFHKS
|
9.3 | IC50 | 2 | — | |
KRKCYEQJGKMBKL
|
9.3 | IC50 | 2 | — | |
PWDSDBVBKCIRHN
|
9.3 | IC50 | 4 | — | |
SWSSTJOKJXGDQH
|
9.3 | IC50 | 2 | — | |
SXIKNOJEFQXCPA
|
9.3 | IC50 | 4 | — | |
TZEHAFMMPSPZTD
|
9.3 | IC50 | 2 | — | |
URUQCDJWYNLAGR
|
9.3 | IC50 | 2 | — | |
WAJIHESGSSDZLV
|
9.3 | IC50 | 6 | — | |
ZJLJEWROVSZOMN
|
9.3 | IC50 | 6 | — | |
OPSRUAAFZJIVQO
|
9.3 | IC50 | 2 | — | |
WPFBXGBKFBKHDX
|
9.2 | IC50 | 3 | — | |
AMLYAMJWYAIXIA
|
9.2 | IC50 | 3 | — | |
DAAOVRXMYNJKRS
|
9.2 | IC50 | 2 | — | |
LHGHYRBRMNOGPF
|
9.2 | IC50 | 2 | — | |
YGOKSIVHHLSPET
|
9.2 | IC50 | 4 | — | |
AKXRNGZFXODFCT
|
9.2 | IC50 | 6 | — | |
BLKCXKZUJXHCGP
|
9.2 | IC50 | 4 | — | |
INPJXWNSGITHFI
|
9.2 | IC50 | 2 | — | |
QEWKBLVMROGVIO
|
9.2 | IC50 | 6 | — | |
WUEFOEAIDROUBP
|
9.2 | IC50 | 3 | — | |
XCOSALUIMNYBMA
|
9.2 | IC50 | 2 | — | |
ABVOSXLHVDENOA
|
9.2 | IC50 | 2 | — | |
AFJXMMWPBLETCO
|
9.2 | IC50 | 2 | — | |
MMTMLJZCVSAZFC
|
9.2 | IC50 | 3 | — | |
OJTBKASAMAYZRX
|
9.2 | IC50 | 2 | — | |
RQMPMSIEFFKLGD
|
9.2 | IC50 | 3 | — | |
SHCPBSMGQZIVTA
|
9.2 | IC50 | 3 | — | |
WGHOQSIOKMBZIJ
|
9.2 | IC50 | 3 | — | |
WROMAHOUFMMNHT
|
9.2 | IC50 | 2 | — | |
XPXOBWWMCFKOKQ
|
9.2 | IC50 | 2 | — | |
GTSHXMCHGDUGRQ
|
9.2 | IC50 | 4 | — | |
SXIKNOJEFQXCPA
|
9.2 | IC50 | 4 | — | |
XIHAPPZUKXNKFE
|
9.2 | IC50 | 2 | — | |
DTCHSFYIOSVBQO
|
9.2 | IC50 | 5 | — |