Target Details
| UniProt AC | P05106 |
|---|---|
| Gene Symbol | ITGB3 |
| Protein Name | Integrin beta-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07974 (EGF_2) PF23105 (EGF_integrin) PF18372 (I-EGF_1) PF08725 (Integrin_b_cyt) PF07965 (Integrin_B_tail) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 2,474
- Clinical molecules 0
- Avg pChEMBL 7.74
KEGG Pathways (26)
- Arrhythmogenic right ventricular cardiomyopathy
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Efferocytosis
- Fluid shear stress and atherosclerosis
- Focal adhesion
- Hematopoietic cell lineage
- Herpes simplex virus 1 infection
- Hormone signaling
- Human cytomegalovirus infection
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- MicroRNAs in cancer
- Neutrophil extracellular trap formation
- Osteoclast differentiation
- PI3K-Akt signaling pathway
- Phagosome
- Platelet activation
- Proteoglycans in cancer
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Thyroid hormone signaling pathway
- Virion - Herpesvirus
Associated Diseases (6)
Active Molecules (2,474)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MKIOVSFGHYIVDB
|
9.5 | IC50 | 3 | — | |
MPAIDFBWWZPGEV
|
9.5 | IC50 | 2 | — | |
OTGFOVKWHHNDHF
|
9.5 | IC50 | 3 | — | |
SHRSEUHJTZQLRO
|
9.5 | IC50 | 8 | — | |
VSAKVGBQGGPIJH
|
9.5 | IC50 | 2 | — | |
VYPOWHUOZSVSQJ
|
9.5 | IC50 | 2 | — | |
XGZVUDGXURHWEC
|
9.5 | IC50 | 3 | — | |
ZFIVYUYYCMBCTR
|
9.5 | IC50 | 2 | — | |
FJUFYEBFJYPEFS
|
9.5 | IC50 | 2 | — | |
JZTSYGNOFKHTHM
|
9.5 | IC50 | 2 | — | |
HLXLTYRHIUOBBV
|
9.5 | IC50 | 2 | — | |
OAUKXLIBIFPGBT
|
9.5 | IC50 | 2 | — | |
PDPLWPUOLLTXCX
|
9.5 | IC50 | 2 | — | |
HDNLLSLLYCIFIU
|
9.5 | IC50 | 2 | — | |
LGMXGJOVGIKKKC
|
9.5 | IC50 | 4 | — | |
FDEYYGVHDVBTNW
|
9.5 | IC50 | 4 | — | |
QPZOEIQRDYCGMD
|
9.5 | IC50 | 5 | — | |
RGDXUISAOHECQH
|
9.5 | IC50 | 2 | — | |
VJTDBRLHPYYFBZ
|
9.5 | IC50 | 2 | — | |
VJTDBRLHPYYFBZ
|
9.5 | IC50 | 2 | — | |
ZBPWDXMZTZUZSY
|
9.5 | IC50 | 2 | — | |
WYVKIJXOPFCHFD
|
9.4 | IC50 | 4 | — | |
ABNXKGFLZFSILK
|
9.4 | IC50 | 2 | — | |
AJCAJRVJXQOQGR
|
9.4 | IC50 | 2 | — | |
BGLLQJHWAUGNSA
|
9.4 | IC50 | 3 | — | |
WWWQNOCFIMKBQL
|
9.4 | IC50 | 2 | — | |
GHKJCEINAARURY
|
9.4 | IC50 | 2 | — | |
JSXUDXGPZPGJOP
|
9.4 | IC50 | 2 | — | |
XQUJDYKAECREGU
|
9.4 | IC50 | 2 | — | |
FVYSXFUNKAIEAQ
|
9.4 | IC50 | 3 | — | |
ICALNGJCZQBZDD
|
9.4 | IC50 | 2 | — | |
MGVKLGFDHDXKFL
|
9.4 | IC50 | 2 | — | |
YWGKJZDMSJRNNY
|
9.4 | IC50 | 2 | — | |
BSNWAPOUYOPCPS
|
9.4 | IC50 | 6 | — | |
HHUNTZLKFUBXAE
|
9.4 | IC50 | 3 | — | |
PRTDUHZCDXSBIZ
|
9.4 | IC50 | 5 | — | |
RIXFBZVXQWVSQN
|
9.4 | IC50 | 2 | — | |
USYHJFFPGOCQTN
|
9.4 | IC50 | 2 | — | |
VQFZVRMJIHFIPZ
|
9.4 | IC50 | 2 | — | |
WBIUNXVKIMTWNG
|
9.4 | IC50 | 2 | — | |
WBNIBVOJNZUYKZ
|
9.4 | IC50 | 3 | — | |
WRJHOBGONWLLMD
|
9.4 | IC50 | 2 | — | |
XTHVPXDEZXVGPQ
|
9.4 | IC50 | 2 | — | |
YSUOCWJZGZEUQT
|
9.4 | IC50 | 2 | — | |
KSSPHFGIOASRDE
|
9.4 | IC50 | 2 | — | |
RIRSYRXZEYNCLO
|
9.4 | IC50 | 4 | — | |
XGMBDTKPGSGTQW
|
9.4 | IC50 | 4 | — | |
YTAHOLPCQRGOAW
|
9.4 | IC50 | 3 | — | |
MSJFRVFQMDZEFH
|
9.3 | IC50 | 2 | — | |
OTRLSMNUUKTGCC
|
9.3 | IC50 | 3 | — |