Target Details
| UniProt AC | P05106 |
|---|---|
| Gene Symbol | ITGB3 |
| Protein Name | Integrin beta-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07974 (EGF_2) PF23105 (EGF_integrin) PF18372 (I-EGF_1) PF08725 (Integrin_b_cyt) PF07965 (Integrin_B_tail) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 2,474
- Clinical molecules 0
- Avg pChEMBL 7.74
KEGG Pathways (26)
- Arrhythmogenic right ventricular cardiomyopathy
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Efferocytosis
- Fluid shear stress and atherosclerosis
- Focal adhesion
- Hematopoietic cell lineage
- Herpes simplex virus 1 infection
- Hormone signaling
- Human cytomegalovirus infection
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- MicroRNAs in cancer
- Neutrophil extracellular trap formation
- Osteoclast differentiation
- PI3K-Akt signaling pathway
- Phagosome
- Platelet activation
- Proteoglycans in cancer
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Thyroid hormone signaling pathway
- Virion - Herpesvirus
Associated Diseases (6)
Active Molecules (2,474)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HIKCELHIZSKMGI
|
8.5 | IC50 | 5 | — | |
KGUBGGAILPYTIW
|
8.5 | IC50 | 2 | — | |
NYIZCWIYRUTEKV
|
8.5 | IC50 | 5 | — | |
ZYPBXFINEXHXPV
|
8.5 | IC50 | 4 | — | |
BLIAKAQPONHNOO
|
8.5 | IC50 | 2 | — | |
IUXWKPVVJPFUJY
|
8.5 | IC50 | 2 | — | |
PVDGZHKJXXVONO
|
8.5 | IC50 | 2 | — | |
ROFCWWUBJHHVGZ
|
8.5 | IC50 | 6 | — | |
SVHYTSHIZOYMFB
|
8.5 | IC50 | 2 | — | |
VOZZIKGZFLWFGA
|
8.5 | IC50 | 3 | — | |
XKFYFSNOQRUIAO
|
8.5 | IC50 | 2 | — | |
YVWHUWDPZJFVCO
|
8.5 | IC50 | 2 | — | |
YVWHUWDPZJFVCO
|
8.5 | IC50 | 2 | — | |
AJZXCRQRDSKMDW
|
8.5 | Kd | 2 | — | |
CUQFEHKORVQEQE
|
8.5 | IC50 | 2 | — | |
KBBXMNQBVKMYCZ
|
8.5 | IC50 | 4 | — | |
NKIPTRIPXHQDGW
|
8.5 | IC50 | 6 | — | |
SUTFGPKMGSBIER
|
8.5 | Kd | 2 | — | |
DGSYYUPRYQBSAI
|
8.5 | IC50 | 2 | — | |
DTINBQRHDAOJQT
|
8.5 | Ki | 2 | — | |
HAWHNGUKUZPYEE
|
8.5 | IC50 | 4 | — | |
HWPUQFFXBNMTKS
|
8.5 | IC50 | 2 | — | |
NENWIXCUUFUHIH
|
8.5 | IC50 | 3 | — | |
QCZXVUVLNOHNFI
|
8.5 | IC50 | 3 | — | |
XGDVRXHWQGEVTD
|
8.5 | IC50 | 3 | — | |
YITSCMGHJOGUNC
|
8.5 | Ki | 3 | — | |
LBBYDFXRXWGQLT
|
8.4 | IC50 | 2 | — | |
AQAUYHNXROATLO
|
8.4 | IC50 | 4 | — | |
BEIUZYAXIMVQKS
|
8.4 | IC50 | 2 | — | |
DVTSXXOIRGTVES
|
8.4 | IC50 | 2 | — | |
FVGFTYFYGPWTIR
|
8.4 | Kd | 2 | — | |
GHKOZFUXJGLMAL
|
8.4 | IC50 | 2 | — | |
QYRCHDXNDRSUDT
|
8.4 | IC50 | 3 | — | |
SJZFNMIWSQZTHK
|
8.4 | IC50 | 2 | — | |
TWQKVYIVXPBLEV
|
8.4 | IC50 | 2 | — | |
VJKNTBIICLHWFT
|
8.4 | IC50 | 2 | — | |
VTLYACZOFKLVKB
|
8.4 | IC50 | 2 | — | |
CXHCNOMGODVIKB
|
8.4 | IC50 | 7 | — | |
GXEBJYPYNMZCSZ
|
8.4 | IC50 | 2 | — | |
OPMDAOWADDAQRY
|
8.4 | IC50 | 4 | — | |
RLABYQGJZRFBJA
|
8.4 | IC50 | 3 | — | |
TUBIMZBESOVRAC
|
8.4 | IC50 | 2 | — | |
VVILZPGXJJNTRY
|
8.4 | IC50 | 2 | — | |
YSBLTULPICYNEV
|
8.4 | IC50 | 2 | — | |
GNIPEZAXNSJOFR
|
8.4 | IC50 | 3 | — | |
HVRQQWLXXYKJKU
|
8.4 | IC50 | 3 | — | |
IHJDDZUSFQGHNY
|
8.4 | IC50 | 2 | — | |
MFGHNUHLUBBJOD
|
8.4 | IC50 | 2 | — | |
MYCBMOUNZVUWNJ
|
8.4 | IC50 | 2 | — | |
NLJFFXADHHBXSL
|
8.4 | IC50 | 2 | — |