Target Details
| UniProt AC | P05106 |
|---|---|
| Gene Symbol | ITGB3 |
| Protein Name | Integrin beta-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07974 (EGF_2) PF23105 (EGF_integrin) PF18372 (I-EGF_1) PF08725 (Integrin_b_cyt) PF07965 (Integrin_B_tail) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 2,474
- Clinical molecules 0
- Avg pChEMBL 7.74
KEGG Pathways (26)
- Arrhythmogenic right ventricular cardiomyopathy
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Efferocytosis
- Fluid shear stress and atherosclerosis
- Focal adhesion
- Hematopoietic cell lineage
- Herpes simplex virus 1 infection
- Hormone signaling
- Human cytomegalovirus infection
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- MicroRNAs in cancer
- Neutrophil extracellular trap formation
- Osteoclast differentiation
- PI3K-Akt signaling pathway
- Phagosome
- Platelet activation
- Proteoglycans in cancer
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Thyroid hormone signaling pathway
- Virion - Herpesvirus
Associated Diseases (6)
Active Molecules (2,474)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NGLDQEAARWHFFU
|
8.5 | IC50 | 4 | — | |
ONCDSJSLWNCDLA
|
8.5 | IC50 | 2 | — | |
ZNBWKHIYCLLIHV
|
8.5 | IC50 | 2 | — | |
ABNXKGFLZFSILK
|
8.5 | IC50 | 2 | — | |
BQYBIJDRTDZCAJ
|
8.5 | IC50 | 8 | — | |
CIAFFIODVHLWSG
|
8.5 | IC50 | 2 | — | |
CJFKBQRLRONQOT
|
8.5 | IC50 | 7 | — | |
CQERSJFWLNZCJI
|
8.5 | IC50 | 2 | — | |
CVAFKDVZZYLXCZ
|
8.5 | IC50 | 2 | — | |
DPVUQQDISRAKFA
|
8.5 | IC50 | 2 | — | |
DPVUQQDISRAKFA
|
8.5 | IC50 | 3 | — | |
DPVUQQDISRAKFA
|
8.5 | IC50 | 3 | — | |
FHDYMEIDWKIBAW
|
8.5 | IC50 | 2 | — | |
GUTGOHPTMQPGTD
|
8.5 | IC50 | 3 | — | |
HIKDGFUZLZJZCB
|
8.5 | IC50 | 8 | — | |
JXVVEFIKDDVLOS
|
8.5 | IC50 | 8 | — | |
KARPAMIZBMUJBW
|
8.5 | IC50 | 2 | — | |
KWKNIANILQEFIG
|
8.5 | IC50 | 2 | — | |
LOTOEFNCKZSRAC
|
8.5 | IC50 | 2 | — | |
MWLPKZBBCRIXMO
|
8.5 | IC50 | 4 | — | |
POPLTANACXUDAZ
|
8.5 | IC50 | 2 | — | |
QVTQDWZYXPQJCE
|
8.5 | IC50 | 2 | — | |
RGUNIWOXWSKLJL
|
8.5 | IC50 | 2 | — | |
RTYLRDWEJUNBLU
|
8.5 | IC50 | 8 | — | |
RUFGUKZOARQZPD
|
8.5 | Ki | 2 | — | |
RWGBUALVFDFMJM
|
8.5 | IC50 | 2 | — | |
RWYVJJKDFYFYFO
|
8.5 | Ki | 2 | — | |
SAFNKDHVPKIPDD
|
8.5 | IC50 | 2 | — | |
SQQTTWBLXRVPQZ
|
8.5 | IC50 | 2 | — | |
SXOQOLFXGFPPBI
|
8.5 | IC50 | 2 | — | |
VPPZGLXMAAPXBC
|
8.5 | Ki | 2 | — | |
WDTHWJIIRVVYRP
|
8.5 | IC50 | 2 | — | |
WIQNHDTZROVWEI
|
8.5 | IC50 | 2 | — | |
WIZNRUGPDHNTSZ
|
8.5 | IC50 | 2 | — | |
WNVOEBNTIMVWEQ
|
8.5 | IC50 | 2 | — | |
WWDVDVKEFFDGFA
|
8.5 | IC50 | 3 | — | |
XKLZVTVODPFBIC
|
8.5 | IC50 | 2 | — | |
XMXSNMYAHVBHCD
|
8.5 | IC50 | 2 | — | |
XNQTZNPDLAFJJK
|
8.5 | IC50 | 2 | — | |
XSXPFCDFDWOKST
|
8.5 | IC50 | 2 | — | |
YPAMHQMVIMQKOR
|
8.5 | IC50 | 8 | — | |
ZCBCTVUDWUBKKH
|
8.5 | IC50 | 2 | — | |
SGUTWRZFDXCOLS
|
8.5 | IC50 | 2 | — | |
CLZGDNHRVKJUHQ
|
8.5 | IC50 | 3 | — | |
JISIOTUNOILQBW
|
8.5 | IC50 | 3 | — | |
XKFYFSNOQRUIAO
|
8.5 | Kd | 2 | — | |
YSHCUQUSNSOANU
|
8.5 | IC50 | 3 | — | |
CECDTIOXBMVUGI
|
8.5 | Ki | 2 | — | |
FHNGIQUASOHITF
|
8.5 | IC50 | 3 | — | |
FSKOAKSLUAJDDL
|
8.5 | IC50 | 3 | — |