Target Details
| UniProt AC | P05106 |
|---|---|
| Gene Symbol | ITGB3 |
| Protein Name | Integrin beta-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07974 (EGF_2) PF23105 (EGF_integrin) PF18372 (I-EGF_1) PF08725 (Integrin_b_cyt) PF07965 (Integrin_B_tail) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 2,474
- Clinical molecules 0
- Avg pChEMBL 7.74
KEGG Pathways (26)
- Arrhythmogenic right ventricular cardiomyopathy
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Efferocytosis
- Fluid shear stress and atherosclerosis
- Focal adhesion
- Hematopoietic cell lineage
- Herpes simplex virus 1 infection
- Hormone signaling
- Human cytomegalovirus infection
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- MicroRNAs in cancer
- Neutrophil extracellular trap formation
- Osteoclast differentiation
- PI3K-Akt signaling pathway
- Phagosome
- Platelet activation
- Proteoglycans in cancer
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Thyroid hormone signaling pathway
- Virion - Herpesvirus
Associated Diseases (6)
Active Molecules (2,474)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RWBOWRDCKZVMOU
|
8.6 | Ki | 2 | — | |
XXBNSEBYSGKBAQ
|
8.6 | IC50 | 4 | — | |
ZNFLNPHHAFFHFM
|
8.6 | IC50 | 2 | — | |
JRVUMBDCNCWNEP
|
8.6 | IC50 | 3 | — | |
AJVBWPQQXWRZHQ
|
8.6 | IC50 | 3 | — | |
DIMDWQUSJSWNOO
|
8.6 | IC50 | 5 | — | |
FTNKTQMIRUQUMO
|
8.6 | Ki | 2 | — | |
HYYAOBWADPQLAZ
|
8.6 | Ki | 2 | — | |
JFGWITIVJGEHEK
|
8.6 | Ki | 2 | — | |
KUZMKJHBJRIPSL
|
8.6 | Ki | 4 | — | |
PYZOVVQJTLOHDG
|
8.6 | Ki | 2 | — | |
STLNBQRXIPETRC
|
8.6 | Ki | 2 | — | |
XCDCCVHZPSJDBH
|
8.6 | IC50 | 3 | — | |
YYQUWEHEBOMRPH
|
8.6 | IC50 | 2 | — | |
BSTGKAROMCRBDW
|
8.6 | IC50 | 2 | — | |
BSTGKAROMCRBDW
|
8.6 | IC50 | 3 | — | |
BXMOZMWEVJVYFV
|
8.6 | IC50 | 2 | — | |
KIOBNTPONYOMJE
|
8.6 | IC50 | 4 | — | |
KRAZOLZZRSRPAE
|
8.6 | IC50 | 4 | — | |
LOLMVTRGQZKBHS
|
8.6 | IC50 | 2 | — | |
NVHPXYIRNJFKTE
|
8.6 | IC50 | 6 | — | |
TYTHBXMTSPUPRQ
|
8.6 | IC50 | 2 | — | |
VUDQMHAFTAQNOM
|
8.6 | IC50 | 4 | — | |
XOCAITJQZBYGFQ
|
8.6 | IC50 | 5 | — | |
RIJYZNGFJGMMPF
|
8.6 | IC50 | 4 | — | |
CJRDXSVCUSRJDR
|
8.6 | IC50 | 8 | — | |
FRCHUTQNZCVLPJ
|
8.6 | IC50 | 2 | — | |
HXARURWAKJJNNF
|
8.6 | IC50 | 3 | — | |
LJRNCZFZZOWSEH
|
8.6 | IC50 | 5 | — | |
LKTCUFLNSKQNFZ
|
8.6 | IC50 | 2 | — | |
LQHWNHQINCFOIZ
|
8.6 | IC50 | 2 | — | |
NQIOUHXNYUMMLV
|
8.6 | IC50 | 4 | — | |
YIJHNENQTDBNGG
|
8.6 | IC50 | 2 | — | |
GFNRURIBKUNSSG
|
8.6 | IC50 | 2 | — | |
AQAUYHNXROATLO
|
8.6 | IC50 | 3 | — | |
CTCHISHHHJCIRE
|
8.6 | IC50 | 2 | — | |
IRAXRQFCCSHQDX
|
8.6 | Kd | 2 | — | |
JNEZPOFKGHMQAC
|
8.6 | IC50 | 3 | — | |
JRIGXBQWNCXPOG
|
8.6 | IC50 | 2 | — | |
JUCUUAVAOJAIHU
|
8.6 | Ki | 2 | — | |
JYJNRUFKUMSRIN
|
8.6 | IC50 | 6 | — | |
MYSBVCKSODARFZ
|
8.6 | IC50 | 3 | — | |
UVNKAYDKTALKMK
|
8.6 | IC50 | 3 | — | |
XRXSSPOFDFFALK
|
8.6 | IC50 | 8 | — | |
ZNERAUDQUULBOO
|
8.6 | IC50 | 3 | — | |
ACEBGKIPKRNNIW
|
8.5 | IC50 | 2 | — | |
GPYWNBXZBJVOHR
|
8.5 | Ki | 2 | — | |
JFZKVQANYRYBMC
|
8.5 | Ki | 2 | — | |
LAROZEWEPNAWMD
|
8.5 | IC50 | 2 | — | |
NGLDQEAARWHFFU
|
8.5 | IC50 | 3 | — |