Target Details
| UniProt AC | P05106 |
|---|---|
| Gene Symbol | ITGB3 |
| Protein Name | Integrin beta-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07974 (EGF_2) PF23105 (EGF_integrin) PF18372 (I-EGF_1) PF08725 (Integrin_b_cyt) PF07965 (Integrin_B_tail) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 2,474
- Clinical molecules 0
- Avg pChEMBL 7.74
KEGG Pathways (26)
- Arrhythmogenic right ventricular cardiomyopathy
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Efferocytosis
- Fluid shear stress and atherosclerosis
- Focal adhesion
- Hematopoietic cell lineage
- Herpes simplex virus 1 infection
- Hormone signaling
- Human cytomegalovirus infection
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- MicroRNAs in cancer
- Neutrophil extracellular trap formation
- Osteoclast differentiation
- PI3K-Akt signaling pathway
- Phagosome
- Platelet activation
- Proteoglycans in cancer
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Thyroid hormone signaling pathway
- Virion - Herpesvirus
Associated Diseases (6)
Active Molecules (2,474)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MFXDNMBOOLLKDW
|
8.7 | Ki | 2 | — | |
MHOGEKRNTRTBND
|
8.7 | IC50 | 2 | — | |
MKIGTYOZNUPATH
|
8.7 | IC50 | 2 | — | |
NUQYRSCTGCUBSM
|
8.7 | IC50 | 2 | — | |
OBOJFQICXTYCRY
|
8.7 | IC50 | 8 | — | |
PVNQAXDNDZYXIW
|
8.7 | Ki | 2 | — | |
RIURMXCCOAPSBY
|
8.7 | IC50 | 2 | — | |
SEQAMEBLAGCPKC
|
8.7 | IC50 | 2 | — | |
SILCDNIUFOQMNJ
|
8.7 | Ki | 2 | — | |
UAYIUFJSMAVZPH
|
8.7 | Ki | 2 | — | |
VKOQXUDGMWQFAJ
|
8.7 | IC50 | 2 | — | |
VSLCOPYIMSFOEG
|
8.7 | IC50 | 2 | — | |
WHVHLBHOPFCDHJ
|
8.7 | IC50 | 2 | — | |
WSAQSLNUSGZKRH
|
8.7 | IC50 | 3 | — | |
XSDMZRDIJUIWTH
|
8.7 | Ki | 2 | — | |
XZIITQXUTRLVIH
|
8.7 | Ki | 2 | — | |
YJHIZJHDJXPOAG
|
8.7 | IC50 | 2 | — | |
YLEXAKYOIPPMHL
|
8.7 | IC50 | 3 | — | |
ZHCINJQZDFCSEL
|
8.7 | IC50 | 2 | — | |
ZPRQEMGTRXGZPE
|
8.7 | IC50 | 5 | — | |
ZPUDEDYAGNPIDY
|
8.7 | Ki | 2 | — | |
LOLMVTRGQZKBHS
|
8.7 | IC50 | 2 | — | |
AFBPNQXAQLFHKE
|
8.7 | IC50 | 2 | — | |
ASSOJPJBNSNTEH
|
8.7 | IC50 | 2 | — | |
CTOPQASYIWIPDN
|
8.7 | IC50 | 3 | — | |
FLABGAZLPSNUBD
|
8.7 | IC50 | 3 | — | |
IACRPVCXCCKFSE
|
8.7 | Ki | 2 | — | |
JMPYJQPICLIXCK
|
8.7 | IC50 | 3 | — | |
LCNAIFMSOWTUTF
|
8.7 | IC50 | 2 | — | |
UAPVZXWNLBOZAW
|
8.7 | Ki | 2 | — | |
UEIWSFUOMHYAMK
|
8.7 | IC50 | 4 | — | |
VSANDTNNMCAWJM
|
8.7 | Kd | 2 | — | |
GJZSXEXGYRGEQC
|
8.7 | IC50 | 3 | — | |
HOXLTGNIFJUOIA
|
8.7 | IC50 | 6 | — | |
NAHSXOFCCYXMHP
|
8.7 | IC50 | 2 | — | |
UVRKETLYFWGQPV
|
8.7 | IC50 | 2 | — | |
VRLVARCYYMQMEO
|
8.7 | IC50 | 2 | — | |
BWAUVRFZNDRMLY
|
8.6 | IC50 | 8 | — | |
CICPWOGAFQCAEW
|
8.6 | IC50 | 2 | — | |
DBFQYQDMGSZHES
|
8.6 | IC50 | 2 | — | |
UQSXTDKNKMCKEM
|
8.6 | IC50 | 3 | — | |
WEGLNNBXKMBXSR
|
8.6 | Ki | 2 | — | |
XEMTYGFOVBXDLG
|
8.6 | IC50 | 2 | — | |
YITSCMGHJOGUNC
|
8.6 | Ki | 2 | — | |
YUFKABYHWCRYRX
|
8.6 | IC50 | 2 | — | |
ZWPCJINLOLYZBQ
|
8.6 | IC50 | 4 | — | |
CGSLGBRMSMBNMX
|
8.6 | IC50 | 6 | — | |
DAFKTUSUEPQPBU
|
8.6 | IC50 | 3 | — | |
ITGKMDQIQJNXCY
|
8.6 | IC50 | 3 | — | |
JYENEFWTARBUPP
|
8.6 | IC50 | 2 | — |