Target Details
| UniProt AC | P05106 |
|---|---|
| Gene Symbol | ITGB3 |
| Protein Name | Integrin beta-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07974 (EGF_2) PF23105 (EGF_integrin) PF18372 (I-EGF_1) PF08725 (Integrin_b_cyt) PF07965 (Integrin_B_tail) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 2,474
- Clinical molecules 0
- Avg pChEMBL 7.74
KEGG Pathways (26)
- Arrhythmogenic right ventricular cardiomyopathy
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Efferocytosis
- Fluid shear stress and atherosclerosis
- Focal adhesion
- Hematopoietic cell lineage
- Herpes simplex virus 1 infection
- Hormone signaling
- Human cytomegalovirus infection
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- MicroRNAs in cancer
- Neutrophil extracellular trap formation
- Osteoclast differentiation
- PI3K-Akt signaling pathway
- Phagosome
- Platelet activation
- Proteoglycans in cancer
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Thyroid hormone signaling pathway
- Virion - Herpesvirus
Associated Diseases (6)
Active Molecules (2,474)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OQLMEWQXUAYOHO
|
10.5 | IC50 | 2 | — | |
IPLLAQOFEDGGKD
|
10.4 | IC50 | 4 | — | |
LEEJTINVSSJMDG
|
10.4 | IC50 | 2 | — | |
LEEJTINVSSJMDG
|
10.4 | IC50 | 3 | — | |
UJAJKKVATBUTAU
|
10.4 | IC50 | 2 | — | |
KBFHSTNZWSMOOM
|
10.3 | IC50 | 2 | — | |
JGRADSKQVRSSDT
|
10.2 | IC50 | 2 | — | |
HAMNCHGAVJSNBY
|
10.2 | IC50 | 3 | — | |
MUWWGBUXCFRNCO
|
10.2 | IC50 | 2 | — | |
DMDDFJFCCZFCKL
|
10.2 | IC50 | 2 | — | |
VGNHZMRKYBWPOO
|
10.2 | IC50 | 3 | — | |
FFYHCEWZIRARDA
|
10.1 | IC50 | 2 | — | |
NCUDSCWWOMSIFO
|
10.1 | IC50 | 2 | — | |
NJDBZBVQIMZWPP
|
10.1 | IC50 | 2 | — | |
CFHPIPZTEAYFIR
|
10.1 | IC50 | 2 | — | |
SVESXPIJWQQCBW
|
10.0 | IC50 | 2 | — | |
LOLMVTRGQZKBHS
|
10.0 | IC50 | 2 | — | |
BGDLLUWAZFBMGD
|
10.0 | IC50 | 2 | — | |
CYKYNQSFAYHHEZ
|
10.0 | IC50 | 2 | — | |
CYKYNQSFAYHHEZ
|
10.0 | IC50 | 3 | — | |
DRZSFOQHHTVBQV
|
10.0 | Ki | 2 | — | |
FGJKSKYLEOZELA
|
10.0 | IC50 | 3 | — | |
FWYCIUUIVROTKO
|
10.0 | Ki | 2 | — | |
LRJXQAWFNQBGLZ
|
10.0 | IC50 | 5 | — | |
QFKUDHXQVSUGKR
|
10.0 | IC50 | 2 | — | |
UFJUFUWNIIBKKK
|
10.0 | IC50 | 2 | — | |
WHDDGMQNGFSWHS
|
10.0 | IC50 | 2 | — | |
WURWJPCCHUZQHY
|
10.0 | IC50 | 2 | — | |
HTJMDVDUBVVYKB
|
10.0 | IC50 | 2 | — | |
KKEMGRLKOQAUBU
|
10.0 | IC50 | 2 | — | |
KSQUEZUEYFZRQY
|
10.0 | IC50 | 2 | — | |
YXLLXCYQWYHDOI
|
10.0 | IC50 | 2 | — | |
HFXICNGRABOTIL
|
9.9 | IC50 | 2 | — | |
UBJJRHHGGWEKRK
|
9.9 | IC50 | 2 | — | |
BDFMVIGZRRIXCL
|
9.9 | IC50 | 5 | — | |
BZNWTXRYYZHACY
|
9.9 | IC50 | 2 | — | |
CQHDUHCWSJOZFD
|
9.9 | IC50 | 2 | — | |
ILIAIJBQDWEDLF
|
9.9 | IC50 | 2 | — | |
QRGILGTYGXRRFJ
|
9.9 | IC50 | 2 | — | |
RFJPNVAPTYAFSN
|
9.9 | IC50 | 2 | — | |
AQNSLCJLLMFYBT
|
9.8 | IC50 | 2 | — | |
XIUUVOUXDREGQI
|
9.8 | IC50 | 2 | — | |
ABNXKGFLZFSILK
|
9.8 | IC50 | 2 | — | |
FXUNUOYKSJCHND
|
9.8 | IC50 | 3 | — | |
YSLIZGZENLHKBF
|
9.8 | IC50 | 2 | — | |
CFXVNDHCOWFOSR
|
9.8 | IC50 | 3 | — | |
DOULIFPELQSYIR
|
9.8 | IC50 | 2 | — | |
MCDJJGKLMCJYFS
|
9.8 | IC50 | 2 | — | |
OVLTXZRGJNTGSK
|
9.8 | IC50 | 2 | — | |
QAFIKBJSAZTLCJ
|
9.8 | IC50 | 2 | — |