Target Details
| UniProt AC | P05067 |
|---|---|
| Gene Symbol | APP |
| Protein Name | Amyloid-beta precursor protein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10515 (APP_amyloid) PF12924 (APP_Cu_bd) PF12925 (APP_E2) PF02177 (APP_N) PF03494 (Beta-APP) PF00014 (Kunitz_BPTI) |
Summary
- Multi-target molecules 345
- Clinical molecules 2
- Avg pChEMBL 7.64
KEGG Pathways (4)
Associated Diseases (2)
Active Molecules (345)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MREAOFDYHRBSRT
|
6.6 | Ki | 3 | — | |
FKENLPZVPNVYQW
|
6.5 | IC50 | 3 | — | |
BRXHNDFMYDDAFF
|
6.5 | IC50 | 2 | — | |
BTQYJGMMVLMRIM
|
6.5 | IC50 | 2 | — | |
GEYFZFDMDJIWCM
|
6.5 | IC50 | 2 | — | |
XJKFPLBHLHQERY
|
6.5 | Ki | 2 | — | |
WPZSQSSOBHCYOZ
|
6.5 | Ki | 3 | — | |
UAEMPXBCTYCXDD
|
6.5 | IC50 | 2 | — | |
BGVASHDMRXAQIW
|
6.5 | IC50 | 2 | — | |
WPEMUUFTBABGBW
|
6.4 | IC50 | 2 | — | |
LWEBLWPFYINVNF
|
6.4 | Kd | 2 | — | |
GDKGAYIPAAQPCP
|
6.4 | IC50 | 2 | — | |
SIABTKWBOMYBGS
|
6.4 | IC50 | 2 | — | |
UACJAEPUZXTOBN
|
6.4 | Kd | 2 | — | |
FKUWIXCLOXGDMB
|
6.4 | IC50 | 3 | — | |
WPZSQSSOBHCYOZ
|
6.4 | Ki | 3 | — | |
NCAGWNFSRXNJDL
|
6.3 | IC50 | 3 | — | |
APPRVPLQWUIXSC
|
6.3 | IC50 | 4 | — | |
OZMOZYSNNYCTFH
|
6.3 | Ki | 2 | — | |
ZKOUORMEQBYWEC
|
6.3 | IC50 | 2 | — | |
HTVUCPUQMUSURS
|
6.3 | IC50 | 2 | — | |
LKLASFRCXLTNMY
|
6.3 | IC50 | 4 | Yes | |
RBTBFTRPCNLSDE
|
6.3 | IC50 | 5 | — | |
UJXWJWJKWZNYSW
|
6.3 | IC50 | 2 | — | |
UQOZNVGULYNSJW
|
6.3 | IC50 | 2 | — | |
YGKQMZYHQKDGRZ
|
6.3 | IC50 | 2 | — | |
QVRAESASNNQBSC
|
6.2 | IC50 | 2 | — | |
LTIOGWHOZDPVCK
|
6.2 | IC50 | 2 | — | |
MNDLUTPGUCHDRU
|
6.2 | IC50 | 2 | — | |
KBPMBBOBMLYWBG
|
6.2 | IC50 | 2 | — | |
VVUQQLRXQSHPIF
|
6.2 | IC50 | 7 | — | |
OZMOZYSNNYCTFH
|
6.2 | Ki | 2 | — | |
VELVOYXHSYTAQT
|
6.2 | Ki | 3 | — | |
FCHFJDXLCKNCCS
|
6.1 | IC50 | 2 | — | |
MWVBEWBNSOHPSD
|
6.1 | IC50 | 2 | — | |
PPISZIMXPLLQGN
|
6.1 | Ki | 3 | — | |
JCRQLFDPHZWIEQ
|
6.1 | IC50 | 2 | — | |
CEOCITIVLDEXBN
|
6.1 | IC50 | 3 | — | |
CFUZORHXMOWNMN
|
6.1 | IC50 | 4 | — | |
VFLDPWHFBUODDF
|
6.1 | IC50 | 25 | — | |
VFLDPWHFBUODDF
|
6.1 | IC50 | 6 | — | |
BENIBYVETVNODM
|
6.1 | IC50 | 2 | — | |
XNFNZERRRUIVBJ
|
6.1 | IC50 | 2 | — | |
QAOTWNNTGAUPFL
|
6.0 | IC50 | 2 | — | |
YBQUWVFHSNRTQF
|
6.0 | Ki | 3 | — |