Target Details
| UniProt AC | P05067 |
|---|---|
| Gene Symbol | APP |
| Protein Name | Amyloid-beta precursor protein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10515 (APP_amyloid) PF12924 (APP_Cu_bd) PF12925 (APP_E2) PF02177 (APP_N) PF03494 (Beta-APP) PF00014 (Kunitz_BPTI) |
Summary
- Multi-target molecules 345
- Clinical molecules 2
- Avg pChEMBL 7.64
KEGG Pathways (4)
Associated Diseases (2)
Active Molecules (345)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RDZDAKHZWXGMEB
|
7.0 | IC50 | 2 | — | |
UMMCMVOJRYIPSD
|
7.0 | IC50 | 2 | — | |
CLOXVWLCRWFUQF
|
7.0 | IC50 | 2 | — | |
VAFUDQUXHDFJQT
|
7.0 | IC50 | 4 | — | |
REPAOSCPUIWQRP
|
7.0 | Ki | 2 | — | |
MDZDVNVGBBGHLD
|
7.0 | IC50 | 3 | — | |
QTMYFSCQEGCHIT
|
7.0 | Ki | 2 | — | |
NOZXPLNYHOGSHE
|
7.0 | Ki | 3 | — | |
IRXWYHUQSSDRPD
|
6.9 | Ki | 2 | — | |
RRXNKIRFKWHJJD
|
6.9 | Ki | 2 | — | |
OMBWPONBVQEDHK
|
6.9 | IC50 | 2 | — | |
VWRHRENEJPEKGV
|
6.9 | IC50 | 2 | — | |
AOIUAVCQCDCNFO
|
6.9 | Ki | 3 | — | |
BOLLXFUEVRCEAN
|
6.9 | Ki | 2 | — | |
IXZCGAMHPOYBCA
|
6.9 | Ki | 3 | — | |
OSPFSPHQIOAXEW
|
6.9 | Ki | 3 | — | |
BHTCXYKONZVALL
|
6.9 | Ki | 3 | — | |
BHTCXYKONZVALL
|
6.9 | Ki | 3 | — | |
MRBBFOWSPXHYQT
|
6.9 | IC50 | 2 | — | |
AOIUAVCQCDCNFO
|
6.8 | Ki | 3 | — | |
WVFHQWCQXOAIHG
|
6.8 | IC50 | 2 | — | |
YUFMOSSQCPKPCP
|
6.8 | IC50 | 2 | — | |
RYPGTHOZCUSFLF
|
6.8 | IC50 | 2 | — | |
OWDYFPYKCCMOHX
|
6.8 | IC50 | 2 | — | |
ZTBPTRRMAKYTAR
|
6.8 | IC50 | 2 | — | |
ULLKDRHZBXMQBC
|
6.8 | IC50 | 2 | — | |
IBJMVRAGTMDAFC
|
6.8 | IC50 | 2 | — | |
PZHFCAIXAVDQAK
|
6.8 | IC50 | 2 | — | |
WSDJYMPBPPNFDL
|
6.8 | IC50 | 2 | — | |
FPIPGXGPPPQFEQ
|
6.7 | IC50 | 3 | — | |
MKLSHCVZEOAEFB
|
6.7 | IC50 | 2 | — | |
NCYCYZXNIZJOKI
|
6.7 | IC50 | 2 | — | |
OJKVNSOZHYKLQR
|
6.7 | IC50 | 2 | — | |
SHGAZHPCJJPHSC
|
6.7 | IC50 | 13 | — | |
YJPIAQRBQQFOPC
|
6.7 | IC50 | 3 | — | |
HODYOYXOWRKLLU
|
6.7 | IC50 | 2 | — | |
KDXWOKQTAHIJMK
|
6.7 | Ki | 2 | — | |
LVRLSYPNFFBYCZ
|
6.7 | IC50 | 3 | — | |
WICQDDCNCVTFDX
|
6.7 | IC50 | 16 | Yes | |
AQOPKQZDRIMOPX
|
6.7 | Ki | 3 | — | |
MJQOUOQLEXOUFE
|
6.7 | IC50 | 2 | — | |
RZZDAMQILXHFNA
|
6.7 | IC50 | 2 | — | |
AZSDCDNUQDIYHT
|
6.6 | IC50 | 7 | — | |
AQOPKQZDRIMOPX
|
6.6 | Ki | 3 | — | |
ILYFUIFSMHDPKE
|
6.6 | Ki | 2 | — | |
SYFKAGCUUZFBGJ
|
6.6 | IC50 | 2 | — | |
CRCWUBLTFGOMDD
|
6.6 | Ki | 2 | — | |
FLQJNXIYQVZXEY
|
6.6 | IC50 | 2 | — | |
NOZXPLNYHOGSHE
|
6.6 | Ki | 3 | — | |
AOIUAVCQCDCNFO
|
6.6 | Kd | 3 | — |