Target Details
| UniProt AC | P05067 |
|---|---|
| Gene Symbol | APP |
| Protein Name | Amyloid-beta precursor protein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10515 (APP_amyloid) PF12924 (APP_Cu_bd) PF12925 (APP_E2) PF02177 (APP_N) PF03494 (Beta-APP) PF00014 (Kunitz_BPTI) |
Summary
- Multi-target molecules 345
- Clinical molecules 2
- Avg pChEMBL 7.64
KEGG Pathways (4)
Associated Diseases (2)
Active Molecules (345)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DFOUAWOLZRCIJU
|
7.5 | IC50 | 2 | — | |
YGNDEESWZOXXLA
|
7.5 | IC50 | 2 | — | |
ROMALOVSXMWQTO
|
7.5 | IC50 | 2 | — | |
YXVXJOUZYSITLN
|
7.5 | IC50 | 7 | — | |
CPNUDRZQULAFCT
|
7.4 | Ki | 3 | — | |
YTTGJOLKFFUHCP
|
7.4 | IC50 | 2 | — | |
NKSGATNIAQTKIG
|
7.4 | Ki | 2 | — | |
PNGMSULGCSIWPT
|
7.4 | IC50 | 2 | — | |
HDIARGDXJLJVAH
|
7.4 | Ki | 2 | — | |
MWVBEWBNSOHPSD
|
7.4 | IC50 | 2 | — | |
XSIPOULVCGGORY
|
7.3 | IC50 | 3 | — | |
YZSOGWONFTWVKT
|
7.3 | IC50 | 2 | — | |
LGQYIGQUEVQRCI
|
7.3 | IC50 | 2 | — | |
LSDKOPMEZMBWQB
|
7.3 | Kd | 2 | — | |
PBZIPKGPSVOZPH
|
7.3 | IC50 | 2 | — | |
PSPGXNMAHYIESQ
|
7.3 | IC50 | 3 | — | |
VOAYXBVNQZNDJQ
|
7.3 | IC50 | 2 | — | |
VPNIQGRFZCTBEZ
|
7.3 | IC50 | 2 | — | |
CKGUJEHCLFSIPS
|
7.3 | Ki | 3 | — | |
MWVBEWBNSOHPSD
|
7.3 | IC50 | 2 | — | |
VFLOCXPTWZLDFY
|
7.3 | IC50 | 7 | — | |
HWLVLRSTFUBCSW
|
7.2 | IC50 | 7 | — | |
SNHBRHBMEDWDNF
|
7.2 | IC50 | 7 | — | |
UXWJPYCELGAIGP
|
7.2 | IC50 | 3 | — | |
XGZLGNFGLZOBER
|
7.2 | IC50 | 2 | — | |
CPNUDRZQULAFCT
|
7.2 | Ki | 3 | — | |
VJQYWRACFCYUPR
|
7.2 | IC50 | 3 | — | |
LPHMJKHHQPFBCQ
|
7.2 | IC50 | 2 | — | |
AAHNBILIYONQLX
|
7.2 | IC50 | 13 | — | |
KKFRXIHTRCQMHV
|
7.2 | IC50 | 7 | — | |
WFIZWFCJKHASMD
|
7.2 | IC50 | 3 | — | |
XDEGBKYUJYVGEV
|
7.2 | IC50 | 2 | — | |
RZPYITONBLAMAN
|
7.2 | IC50 | 2 | — | |
BABOZPFZHGSHOB
|
7.2 | Ki | 2 | — | |
BIODWENPZVUOJQ
|
7.1 | IC50 | 2 | — | |
QMFFOURMHQBKKZ
|
7.1 | Ki | 2 | — | |
XUWDIJDGYAIURP
|
7.1 | IC50 | 2 | — | |
YSSDLRQAOJLLFT
|
7.1 | IC50 | 7 | — | |
OSPFSPHQIOAXEW
|
7.1 | Ki | 3 | — | |
QYVNHRYCOVFLFE
|
7.1 | IC50 | 2 | — | |
XSQKUWZLKKUZPU
|
7.1 | IC50 | 2 | — | |
XXRXTSVWBPYSMG
|
7.1 | Kd | 2 | — | |
HTWVAHYYWZCEOA
|
7.1 | IC50 | 2 | — | |
OOYVWTJLOZOKAU
|
7.1 | IC50 | 2 | — | |
BMPSPTZUQDKEEP
|
7.1 | IC50 | 3 | — | |
QOCIHSUXWNYFHI
|
7.1 | IC50 | 3 | — | |
RMFCYJGEXZDLRL
|
7.1 | IC50 | 2 | — | |
MQFTZDVMSMFRAU
|
7.1 | IC50 | 3 | — | |
NYMXIKPEDWDOQL
|
7.1 | IC50 | 2 | — | |
XNUKXZBBFWKBDZ
|
7.1 | IC50 | 3 | — |