Target Details
| UniProt AC | P05067 |
|---|---|
| Gene Symbol | APP |
| Protein Name | Amyloid-beta precursor protein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10515 (APP_amyloid) PF12924 (APP_Cu_bd) PF12925 (APP_E2) PF02177 (APP_N) PF03494 (Beta-APP) PF00014 (Kunitz_BPTI) |
Summary
- Multi-target molecules 345
- Clinical molecules 2
- Avg pChEMBL 7.64
KEGG Pathways (4)
Associated Diseases (2)
Active Molecules (345)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PGKOVKXDONQGMH
|
7.8 | IC50 | 2 | — | |
WPIVAKLBMCTDCK
|
7.8 | IC50 | 2 | — | |
LPTYIZIFEMAJPK
|
7.8 | IC50 | 2 | — | |
LTKKMSORNDRROD
|
7.8 | IC50 | 7 | — | |
MTRPAEDXTYGACS
|
7.8 | IC50 | 2 | — | |
PKBFNKHRNBOEGL
|
7.8 | IC50 | 2 | — | |
ROJZGNGSPMMZLM
|
7.8 | IC50 | 2 | — | |
OJULZIHGKOEUGD
|
7.8 | IC50 | 2 | — | |
DGKJKZFNUCFCQA
|
7.8 | IC50 | 3 | — | |
FGCFYPLYGHWAIM
|
7.8 | IC50 | 2 | — | |
HALWMQVNBCAXRZ
|
7.8 | IC50 | 2 | — | |
HBGNURMASUAQFL
|
7.8 | Kd | 3 | — | |
OAMAZEDOCLMRJG
|
7.8 | IC50 | 2 | — | |
MQZGUSZHWAGWJN
|
7.8 | IC50 | 2 | — | |
CYYGGALMMNBOPQ
|
7.8 | Ki | 2 | — | |
VEZYROFGIDSNEB
|
7.7 | IC50 | 2 | — | |
GEFZXXPGNGYLMH
|
7.7 | IC50 | 2 | — | |
GNNDIRZJLBDRCO
|
7.7 | IC50 | 3 | — | |
PPPNFACLMPPXHQ
|
7.7 | IC50 | 2 | — | |
RJIJEEIOHDLRFZ
|
7.7 | IC50 | 2 | — | |
VHAUFUROQRJMRS
|
7.7 | IC50 | 2 | — | |
ITDYKITUTOFAKT
|
7.7 | Ki | 2 | — | |
NVGBNEWLPGDDDO
|
7.7 | IC50 | 2 | — | |
VIKJQTTZBYWMNX
|
7.7 | Ki | 2 | — | |
LFRZWTUDQUJIOZ
|
7.7 | IC50 | 3 | — | |
PDZMLCFMZBYPNH
|
7.7 | Kd | 3 | — | |
QVNUOJRVQDGJQW
|
7.7 | IC50 | 8 | — | |
XXUKTXRJOFQHLP
|
7.7 | IC50 | 4 | — | |
YMEVFLBOXWRPCH
|
7.7 | IC50 | 2 | — | |
AMGGIBWEIGCKRZ
|
7.6 | Ki | 2 | — | |
JCRFLTOHIUBPBI
|
7.6 | IC50 | 2 | — | |
MAUWSMJVVWTKNC
|
7.6 | IC50 | 2 | — | |
RVZQCFAUGDSGAA
|
7.6 | IC50 | 2 | — | |
OLJWGKMQUSBBIA
|
7.6 | IC50 | 7 | — | |
OLJWGKMQUSBBIA
|
7.6 | IC50 | 2 | — | |
DOJQNRYLSRMQDA
|
7.6 | IC50 | 4 | — | |
FGYNZFHVGOFCMD
|
7.6 | Ki | 2 | — | |
KGNLPACQRCXMGM
|
7.6 | IC50 | 2 | — | |
KSZDQDUDHWUQCJ
|
7.6 | IC50 | 3 | — | |
LWCYPSYNLAAESS
|
7.6 | IC50 | 2 | — | |
BGQRAIICKIPHAT
|
7.6 | Ki | 2 | — | |
HUQALVJHHCENTE
|
7.6 | IC50 | 4 | — | |
RDBWLFGMGXLTQD
|
7.6 | IC50 | 7 | — | |
TULNEWNRYDONGE
|
7.6 | Ki | 2 | — | |
LOLRSSGXRIPFCB
|
7.6 | IC50 | 3 | — | |
MZAPDYQWIGAEQO
|
7.6 | IC50 | 8 | — | |
GEFZXXPGNGYLMH
|
7.6 | IC50 | 2 | — | |
FMYPBFZNJZIDKT
|
7.5 | IC50 | 3 | — | |
RNLNFTQJIYFRSH
|
7.5 | IC50 | 3 | — | |
CLWLYGJCKORDAK
|
7.5 | IC50 | 2 | — |