Target Details
| UniProt AC | P05067 |
|---|---|
| Gene Symbol | APP |
| Protein Name | Amyloid-beta precursor protein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10515 (APP_amyloid) PF12924 (APP_Cu_bd) PF12925 (APP_E2) PF02177 (APP_N) PF03494 (Beta-APP) PF00014 (Kunitz_BPTI) |
Summary
- Multi-target molecules 345
- Clinical molecules 2
- Avg pChEMBL 7.64
KEGG Pathways (4)
Associated Diseases (2)
Active Molecules (345)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UDNMOPIWQUAQRD
|
8.2 | IC50 | 7 | — | |
ISXCJKRNXUQSFB
|
8.2 | IC50 | 3 | — | |
JLPMGOFESRTFLV
|
8.2 | IC50 | 2 | — | |
VZKPBWICQCZMIB
|
8.2 | IC50 | 3 | — | |
WNIDBJOQKWEFFV
|
8.1 | IC50 | 2 | — | |
UTPYURSIXIVBEJ
|
8.1 | IC50 | 7 | — | |
JXMIZSIVCHFRDW
|
8.1 | IC50 | 2 | — | |
FIQQLONWDXAKPQ
|
8.1 | Kd | 3 | — | |
HEZJDRFUHMYWFH
|
8.1 | IC50 | 2 | — | |
XZRLHXIFWZKMCO
|
8.1 | IC50 | 3 | — | |
GQLYTFBOIYIDOU
|
8.1 | IC50 | 7 | — | |
OLLCSNPRGPMBHT
|
8.1 | IC50 | 7 | — | |
MBVITGGTLKHHQT
|
8.1 | IC50 | 2 | — | |
SMKLPOGYVJHNSP
|
8.1 | IC50 | 2 | — | |
QQULQSVUDLAXCV
|
8.1 | IC50 | 2 | — | |
TWKUHRBKUHLJDI
|
8.1 | IC50 | 3 | — | |
WAZXJCCRJQZNHV
|
8.1 | IC50 | 3 | — | |
WUJRLQGOZRVKDS
|
8.0 | IC50 | 2 | — | |
GBNJNJPEBSZUOQ
|
8.0 | IC50 | 2 | — | |
DRKAFGKWERJHKK
|
8.0 | IC50 | 4 | — | |
IBGZXUPONLUVLS
|
8.0 | IC50 | 2 | — | |
LUDSHWAKEHVLGG
|
8.0 | IC50 | 2 | — | |
OHQWUKZYZSMZAC
|
8.0 | IC50 | 7 | — | |
UNTHRMMZVRJKBA
|
8.0 | IC50 | 7 | — | |
FSPVOBOVPOEPEV
|
8.0 | IC50 | 2 | — | |
MJLRPASHEJEXBJ
|
8.0 | IC50 | 7 | — | |
POIRYFHGYWLALK
|
8.0 | IC50 | 2 | — | |
RTQLEDFPONJSDB
|
8.0 | Ki | 2 | — | |
BQEOVNOSRGLHCK
|
8.0 | IC50 | 2 | — | |
QUSFOPKCQPEPCC
|
8.0 | Ki | 2 | — | |
QUDGAPHVUAEHFA
|
8.0 | IC50 | 2 | — | |
YNDIAUKFXKEXSV
|
8.0 | Ki | 3 | — | |
HJMCUUCUCMHIEU
|
7.9 | IC50 | 2 | — | |
GOOGDNLQKOSOJY
|
7.9 | IC50 | 2 | — | |
CGFNKFZCIRBOAD
|
7.9 | IC50 | 3 | — | |
DJWUDIFTUQYCIR
|
7.9 | IC50 | 8 | — | |
USRBCCHTSUIKOF
|
7.9 | IC50 | 2 | — | |
YLJREFDVOIBQDA
|
7.9 | IC50 | 7 | — | |
KWUKMYMZASNCGG
|
7.9 | IC50 | 2 | — | |
PDOPEKODNLOZRJ
|
7.9 | IC50 | 2 | — | |
PUANGZKWYIUWGX
|
7.9 | IC50 | 3 | — | |
UDZQLDSLTPDOSW
|
7.9 | Ki | 2 | — | |
VABJLQOQMZEOHJ
|
7.9 | IC50 | 2 | — | |
XWRREAIVFZDEEK
|
7.9 | IC50 | 2 | — | |
BABSGYNDJJCRAD
|
7.9 | IC50 | 2 | — | |
LWHLEVWRUZVAKD
|
7.9 | IC50 | 7 | — | |
LWHLEVWRUZVAKD
|
7.9 | IC50 | 2 | — | |
ZWUWGLTVWPXQQS
|
7.8 | IC50 | 3 | — | |
AEEPSMNZRMEZBF
|
7.8 | IC50 | 2 | — | |
GGFYWXBSNMOKOK
|
7.8 | Ki | 2 | — |