Target Details
| UniProt AC | P05067 |
|---|---|
| Gene Symbol | APP |
| Protein Name | Amyloid-beta precursor protein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10515 (APP_amyloid) PF12924 (APP_Cu_bd) PF12925 (APP_E2) PF02177 (APP_N) PF03494 (Beta-APP) PF00014 (Kunitz_BPTI) |
Summary
- Multi-target molecules 345
- Clinical molecules 2
- Avg pChEMBL 7.64
KEGG Pathways (4)
Associated Diseases (2)
Active Molecules (345)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JQBMPLUGJXSJPF
|
8.6 | IC50 | 2 | — | |
PPPNFACLMPPXHQ
|
8.6 | IC50 | 2 | — | |
WEHAHFRWAHYPCU
|
8.6 | IC50 | 2 | — | |
AMWCDMOOTAVMSV
|
8.6 | IC50 | 2 | — | |
GJVWSAKHBXGRHV
|
8.6 | IC50 | 2 | — | |
YNWCSWFGCSURHN
|
8.6 | IC50 | 2 | — | |
GSAVHMBMISQPPR
|
8.6 | IC50 | 2 | — | |
ULDMQHGBWVBBMN
|
8.5 | IC50 | 2 | — | |
AWWAZUFXKKZKCD
|
8.5 | IC50 | 2 | — | |
BQFHTVUWPJXLOW
|
8.5 | IC50 | 3 | — | |
BSTQSBRVJGRBPC
|
8.5 | IC50 | 2 | — | |
LHTZVIDMVHFLLF
|
8.5 | IC50 | 4 | — | |
MTNQDQUYJFDVLS
|
8.5 | IC50 | 4 | — | |
PSBBWFNMHDUTRH
|
8.5 | IC50 | 4 | — | |
RZBPWVNRIHVDBR
|
8.5 | IC50 | 2 | — | |
OEJPKPVOWLAKLD
|
8.5 | Kd | 2 | — | |
RDZDAKHZWXGMEB
|
8.5 | IC50 | 2 | — | |
PEYUKFMDCGZLQN
|
8.5 | IC50 | 3 | — | |
GYYFFSAIGLHSCV
|
8.5 | IC50 | 2 | — | |
HRDQJFPXQGWLSV
|
8.4 | IC50 | 2 | — | |
KVNVGAUWCHPHOE
|
8.4 | Kd | 3 | — | |
YMBXEBSSLRFPOM
|
8.4 | IC50 | 3 | — | |
JJEORDNWHQBLEW
|
8.4 | IC50 | 2 | — | |
FSIYTVBWWROBPT
|
8.4 | IC50 | 2 | — | |
HYRSOCCYHCESGJ
|
8.4 | IC50 | 3 | — | |
KBPMBBOBMLYWBG
|
8.4 | IC50 | 2 | — | |
XGBNYYCTJVZIKG
|
8.4 | IC50 | 3 | — | |
DIYNYEGNVUSOIR
|
8.4 | IC50 | 7 | — | |
FSPVOBOVPOEPEV
|
8.4 | IC50 | 2 | — | |
IQIVZKLXTXCLSL
|
8.4 | IC50 | 2 | — | |
SPYYWCDGZNJHNH
|
8.4 | Kd | 2 | — | |
MZMGBLWHPUKZKF
|
8.4 | IC50 | 2 | — | |
QRKMJBIQBFXXFC
|
8.4 | IC50 | 2 | — | |
YTYDNLGBBFZDFG
|
8.4 | IC50 | 2 | — | |
RDZDAKHZWXGMEB
|
8.3 | IC50 | 2 | — | |
WXWZQOAPXMLOGN
|
8.3 | IC50 | 2 | — | |
VDXFKYHWRXWVOF
|
8.3 | IC50 | 3 | — | |
WNIDBJOQKWEFFV
|
8.3 | IC50 | 2 | — | |
YGUANPLEQMZXTA
|
8.3 | IC50 | 2 | — | |
CSWYTFLVWXTIPC
|
8.3 | Kd | 3 | — | |
MONBOQDZSLNZSN
|
8.3 | IC50 | 3 | — | |
MWIIPGZITGHTPU
|
8.3 | IC50 | 4 | — | |
CFGDZHHUKZKWPM
|
8.3 | IC50 | 2 | — | |
CDKNJSXTOTWFRF
|
8.3 | IC50 | 7 | — | |
HKXVZYVBKHNCOB
|
8.3 | IC50 | 2 | — | |
ZQAQXZBSGZUUNL
|
8.2 | Ki | 2 | — | |
NGPXAOWJBUFQFX
|
8.2 | IC50 | 3 | — | |
UCYVFUSXGNJNEO
|
8.2 | IC50 | 2 | — | |
KEJARRYEPKQENB
|
8.2 | IC50 | 2 | — | |
HZHGVFUZMFVSNM
|
8.2 | IC50 | 2 | — |