Target Details
| UniProt AC | P05067 |
|---|---|
| Gene Symbol | APP |
| Protein Name | Amyloid-beta precursor protein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10515 (APP_amyloid) PF12924 (APP_Cu_bd) PF12925 (APP_E2) PF02177 (APP_N) PF03494 (Beta-APP) PF00014 (Kunitz_BPTI) |
Summary
- Multi-target molecules 345
- Clinical molecules 2
- Avg pChEMBL 7.64
KEGG Pathways (4)
Associated Diseases (2)
Active Molecules (345)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WKDNQONLGXOZRG
|
9.5 | IC50 | 2 | — | |
WKDNQONLGXOZRG
|
9.4 | IC50 | 3 | — | |
SKNSXIIPICYXKY
|
9.3 | IC50 | 2 | — | |
BQDUISPSAOQZDJ
|
9.2 | IC50 | 2 | — | |
WDZVWDXOIGQJIO
|
9.2 | IC50 | 3 | — | |
FMNVIPHETSINMI
|
9.2 | IC50 | 2 | — | |
MQWMIBOBCNOFGX
|
9.2 | IC50 | 2 | — | |
JJEORDNWHQBLEW
|
9.2 | IC50 | 2 | — | |
LWCYPSYNLAAESS
|
9.2 | IC50 | 2 | — | |
AGTQGRFUNIAYJX
|
9.1 | IC50 | 2 | — | |
DDHXRMBHBIIYGG
|
9.1 | IC50 | 2 | — | |
DSCREMQTOOAGKC
|
9.1 | IC50 | 2 | — | |
BCPJXJSUDZCZSL
|
9.0 | IC50 | 2 | — | |
JXQACBKQPQKDBW
|
9.0 | IC50 | 2 | — | |
NVGRJZRZTUKQGI
|
9.0 | IC50 | 2 | — | |
OOYVWTJLOZOKAU
|
9.0 | IC50 | 2 | — | |
PQYGXBUKYSOKJA
|
9.0 | IC50 | 2 | — | |
DZGFZIMDVXHKMA
|
9.0 | IC50 | 2 | — | |
XSPYGYYSPGDIRH
|
9.0 | IC50 | 2 | — | |
UMCUVZSSUIPNCL
|
9.0 | IC50 | 2 | — | |
JJDMMVKGGCIWNE
|
9.0 | IC50 | 2 | — | |
SKNSXIIPICYXKY
|
8.9 | IC50 | 2 | — | |
VYVMTNNUVNSRBD
|
8.9 | Kd | 3 | — | |
ZXRHVPQEUUVSBF
|
8.9 | IC50 | 2 | — | |
CGJQMXWLLKPNOI
|
8.9 | IC50 | 2 | — | |
ITBUOSMBIYYJMH
|
8.9 | IC50 | 3 | — | |
WHKFJZYBRJHBJY
|
8.9 | IC50 | 2 | — | |
XWVPZETUJYENCA
|
8.9 | IC50 | 2 | — | |
BHCDFMZEDWIROP
|
8.9 | IC50 | 2 | — | |
OYVJXWZSTBCONR
|
8.9 | IC50 | 2 | — | |
CIGIICMKOOPQKH
|
8.8 | IC50 | 2 | — | |
XTQZDTBINKMEKZ
|
8.8 | IC50 | 2 | — | |
XHPVFJGGOWNHQR
|
8.8 | IC50 | 2 | — | |
XWVPZETUJYENCA
|
8.8 | IC50 | 2 | — | |
DSCREMQTOOAGKC
|
8.8 | IC50 | 2 | — | |
LWCYPSYNLAAESS
|
8.8 | IC50 | 2 | — | |
MJQOUOQLEXOUFE
|
8.8 | IC50 | 2 | — | |
PYCHQFOZUGUMBW
|
8.8 | IC50 | 2 | — | |
WOFHTRRBXQUHFJ
|
8.8 | IC50 | 2 | — | |
DDHXRMBHBIIYGG
|
8.8 | IC50 | 2 | — | |
HZHGVFUZMFVSNM
|
8.7 | IC50 | 2 | — | |
WBYPVXZFTBKPDX
|
8.7 | Ki | 2 | — | |
HZHGVFUZMFVSNM
|
8.7 | IC50 | 2 | — | |
QSYNDUROVMEDHR
|
8.6 | IC50 | 2 | — | |
ZTHSMBOBTMQWJX
|
8.6 | IC50 | 2 | — | |
CLOXVWLCRWFUQF
|
8.6 | IC50 | 2 | — | |
GHKDKBMFJNPSBF
|
8.6 | IC50 | 2 | — | |
KKKLWLSGVSXCDO
|
8.6 | IC50 | 8 | — | |
MUPBWXCOUHZWEH
|
8.6 | IC50 | 2 | — | |
RMFCYJGEXZDLRL
|
8.6 | IC50 | 2 | — |