Target Details
| UniProt AC | P04632 |
|---|---|
| Gene Symbol | CAPNS1 |
| Protein Name | Calpain small subunit 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
Summary
- Multi-target molecules 56
- Clinical molecules 2
- Avg pChEMBL 6.92
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (56)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XGJGWYRHLPSMLW
|
8.3 | IC50 | 2 | — | |
YTSRZPGVQKOFFF
|
8.1 | IC50 | 2 | — | |
UNCOFUQMWOIDMS
|
8.1 | Ki | 3 | — | |
WQBLPTWYDVNJDE
|
7.7 | IC50 | 2 | — | |
DSYDMMPAZVEHMK
|
7.6 | IC50 | 2 | — | |
SMHWTXZVZOFOFA
|
7.6 | IC50 | 2 | — | |
VXFRMVRMWOZAFZ
|
7.5 | IC50 | 2 | — | |
CSKGFHNQMOIAFM
|
7.5 | IC50 | 4 | Yes | |
WNILNJHVHCOVFU
|
7.4 | IC50 | 2 | — | |
NGBKFLTYGSREKK
|
7.4 | IC50 | 6 | Yes | |
NGBKFLTYGSREKK
|
7.4 | IC50 | 4 | — | |
BPDWJQKYAHEPMF
|
7.3 | IC50 | 2 | — | |
BQWHGKILBWBBEZ
|
7.3 | Ki | 3 | — | |
HHNHYEDODWWQEY
|
7.3 | IC50 | 2 | — | |
XUZYDWHWSIJZRS
|
7.3 | IC50 | 2 | — | |
GLNKVXFQBYGNDP
|
7.2 | Ki | 3 | — | |
GLEMPIVMKMAASA
|
7.1 | Ki | 3 | — | |
NTZYOTXUVHBKSM
|
7.1 | IC50 | 2 | — | |
SEANAGCTCGCPQM
|
7.1 | Ki | 3 | — | |
OIXYHRZFKWJACP
|
7.1 | IC50 | 2 | — | |
NWUVYAAEXDXAHP
|
7.0 | IC50 | 2 | — | |
BJVLXPNAIXTDOW
|
7.0 | Ki | 3 | — | |
BYUMFTKUIXAFNT
|
7.0 | IC50 | 2 | — | |
OFDVDFSINZOAMJ
|
7.0 | IC50 | 2 | — | |
OITJHBJCHPRBCI
|
7.0 | IC50 | 2 | — | |
ORFNBDAQQVIIPT
|
7.0 | IC50 | 2 | — | |
RFLQJGASGWLMCH
|
7.0 | Ki | 3 | — | |
FYLLWVNXHDSOBP
|
7.0 | IC50 | 2 | — | |
IZOVMLGFODKHHH
|
6.9 | Ki | 2 | — | |
AHEDBTSELMBNTN
|
6.9 | IC50 | 2 | — | |
BSQXGCSIDWZSHW
|
6.8 | IC50 | 2 | — | |
AYSDUNWXRUGZRO
|
6.8 | IC50 | 2 | — | |
ZOBGGAIYJYPPGQ
|
6.8 | IC50 | 2 | — | |
PRVNMMSXHWFZAQ
|
6.8 | Ki | 3 | — | |
GOYRCQFAGVGQLH
|
6.7 | Ki | 3 | — | |
QDIFXVWJRNFSAW
|
6.7 | Ki | 3 | — | |
QFMKANIDVYDNPI
|
6.7 | Ki | 3 | — | |
WJDCRUSBRSNMME
|
6.7 | Ki | 3 | — | |
VZPAOLJPGFQEEK
|
6.7 | Ki | 3 | — | |
ODVBWVUZXJFGFP
|
6.7 | IC50 | 2 | — | |
LKVFZCXXFXGYDC
|
6.6 | Ki | 3 | — | |
XUFBOUSMDJZDOA
|
6.6 | IC50 | 2 | — | |
YLELJBQQWFIURX
|
6.5 | Ki | 3 | — | |
BALDEWOSOSUCAN
|
6.5 | Ki | 3 | — | |
NDHXUSGFCSYNLZ
|
6.5 | Ki | 2 | — | |
XJZJHBWBHUESJD
|
6.5 | Ki | 3 | — | |
ZEPJUNYIGZQROD
|
6.5 | IC50 | 2 | — | |
OIKITZBTDSAJQH
|
6.4 | IC50 | 4 | — | |
BOLCGBQAKSTBLH
|
6.3 | IC50 | 2 | — | |
VLHHFIURJMMQSU
|
6.3 | Ki | 3 | — |