Target Details
| UniProt AC | P04629 |
|---|---|
| Gene Symbol | NTRK1 |
| Protein Name | High affinity nerve growth factor receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF13855 (LRR_8) PF16920 (LRRCT_2) PF07714 (PK_Tyr_Ser-Thr) PF18613 (TrkA_TMD) |
Summary
- Multi-target molecules 1,127
- Clinical molecules 52
- Avg pChEMBL 7.65
KEGG Pathways (11)
Associated Diseases (4)
Active Molecules (1,127)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NRFLPOVNIIJIDX
|
8.1 | IC50 | 3 | — | |
NVTUEJKEIISOPJ
|
8.1 | IC50 | 3 | — | |
NWDUSAJTSMCLKW
|
8.1 | IC50 | 3 | — | |
RONLQWJKAFWDOO
|
8.1 | IC50 | 3 | — | |
SOWTUSBRJBRQBT
|
8.1 | IC50 | 3 | — | |
SUZGZTADNRRPLU
|
8.1 | IC50 | 3 | — | |
XAJRDFVVIXWATE
|
8.1 | IC50 | 2 | — | |
XURYENAZODILKN
|
8.1 | IC50 | 2 | — | |
YNXUIZMRPVCJTM
|
8.1 | IC50 | 3 | — | |
FXIGRQYWRMUBFO
|
8.1 | IC50 | 3 | — | |
GCYXEGSPUDSZJY
|
8.1 | IC50 | 17 | Yes | |
HRXHRVGEOCMYJD
|
8.1 | IC50 | 2 | — | |
ITGKPZIBLXMPGK
|
8.1 | IC50 | 2 | — | |
NRXYESAXZCGGAF
|
8.1 | IC50 | 2 | — | |
SIPNIVSCAYGONU
|
8.1 | IC50 | 3 | — | |
UGNXBDMIUNXKPM
|
8.1 | IC50 | 3 | — | |
WABINVADIAZJHY
|
8.0 | IC50 | 3 | — | |
BXQLLJDNLWFKET
|
8.0 | IC50 | 2 | — | |
CPLYGSUKEOEHTJ
|
8.0 | IC50 | 2 | — | |
FQQIJMFIYQPLDE
|
8.0 | IC50 | 2 | — | |
KTEIFNKAUNYNJU
|
8.0 | IC50 | 114 | — | |
YYDUWLSETXNJJT
|
8.0 | IC50 | 5 | — | |
WAILKVZLYWOKPO
|
8.0 | IC50 | 3 | — | |
HAPDPSKWHISKDX
|
8.0 | IC50 | 2 | — | |
NXDRKVFQQJUBOG
|
8.0 | IC50 | 2 | — | |
OSIRKNSRCSGLDC
|
8.0 | IC50 | 2 | — | |
PTVPBWWDGZSEAF
|
8.0 | Ki | 63 | — | |
UAZRNUYGVNUMRW
|
8.0 | IC50 | 3 | — | |
XOOAAYRIVATZNM
|
8.0 | Ki | 55 | — | |
KMEGQNKGSCVGJZ
|
8.0 | IC50 | 3 | — | |
NGFHESZMOOWBCG
|
8.0 | IC50 | 2 | — | |
RMCCHANPQRKRIO
|
8.0 | IC50 | 3 | — | |
ZWVGJPGEHUORGV
|
8.0 | IC50 | 3 | — | |
BOGXBCHXRCHFDS
|
8.0 | IC50 | 2 | — | |
CABSRBXIZHPYSN
|
8.0 | IC50 | 2 | — | |
XBJCMGUGQRINQY
|
8.0 | IC50 | 2 | — | |
AGTCXVHPFWVGDM
|
8.0 | IC50 | 2 | — | |
CHLFFSKXUJQLQO
|
8.0 | IC50 | 7 | — | |
GNHQMDGKASSYQR
|
8.0 | IC50 | 2 | — | |
KZFPHKZQVCYHEZ
|
8.0 | IC50 | 3 | — | |
OVSWBIYHLZFTTJ
|
8.0 | IC50 | 2 | — | |
DXPSQKSTVIVZLV
|
8.0 | IC50 | 6 | Yes | |
MIWWARHIDNFXAZ
|
8.0 | IC50 | 6 | — | |
MYNCTXHNZVXWKX
|
8.0 | IC50 | 3 | — | |
WAVGXEMZTAFUCY
|
8.0 | IC50 | 2 | — | |
AMUDMWQYJMAZGP
|
8.0 | IC50 | 2 | — | |
HNJJBTOZBLOWTO
|
8.0 | IC50 | 2 | — | |
KUMKUBXRGRIPEY
|
8.0 | IC50 | 2 | — | |
PURCTPVNRDSZSF
|
8.0 | IC50 | 2 | — | |
OBIPEYBSOQNLDE
|
7.9 | IC50 | 3 | — |