Target Details
| UniProt AC | P04629 |
|---|---|
| Gene Symbol | NTRK1 |
| Protein Name | High affinity nerve growth factor receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF13855 (LRR_8) PF16920 (LRRCT_2) PF07714 (PK_Tyr_Ser-Thr) PF18613 (TrkA_TMD) |
Summary
- Multi-target molecules 1,127
- Clinical molecules 52
- Avg pChEMBL 7.65
KEGG Pathways (11)
Associated Diseases (4)
Active Molecules (1,127)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GJKJRHCPSRGVLC
|
8.2 | IC50 | 2 | — | |
MLIFTZTWMYPZAL
|
8.2 | IC50 | 2 | — | |
TZPUNPWJLMOANL
|
8.2 | IC50 | 6 | — | |
WLZVGCRFNLQBBM
|
8.2 | IC50 | 2 | — | |
WMWHVTDZNIVNIE
|
8.2 | IC50 | 9 | — | |
WMWHVTDZNIVNIE
|
8.2 | IC50 | 9 | — | |
CNSDQPQILIEBIM
|
8.2 | IC50 | 2 | — | |
HAFMFNSFPWDDBC
|
8.2 | IC50 | 5 | — | |
HMMBZLXOFKQWRQ
|
8.2 | IC50 | 2 | — | |
JCRUDKWPDBIGME
|
8.2 | IC50 | 2 | — | |
JECVRFZSSMBKTJ
|
8.2 | IC50 | 2 | — | |
SBXCJOXIBNFCBN
|
8.2 | IC50 | 3 | — | |
VXJAFFGXYYHGQN
|
8.2 | IC50 | 3 | — | |
XOTYCWCEXOJPBF
|
8.2 | IC50 | 3 | — | |
ZQGBDVIGTTVIFV
|
8.2 | IC50 | 3 | — | |
BFTXUHWRGHJJHM
|
8.1 | IC50 | 2 | — | |
JWPYZYBMSBDDCD
|
8.1 | IC50 | 2 | — | |
LQVXSNNAFNGRAH
|
8.1 | IC50 | 33 | Yes | |
ZNNDCLZKVULOKL
|
8.1 | IC50 | 3 | — | |
PMKFFRXMNWSTLH
|
8.1 | IC50 | 2 | — | |
ZBJDRRTVBWHVAP
|
8.1 | IC50 | 2 | — | |
DSZLKOXKYRREEO
|
8.1 | IC50 | 10 | — | |
WRZKZMHISIDZRI
|
8.1 | IC50 | 3 | — | |
XOWLGKWJTBNPJL
|
8.1 | IC50 | 3 | — | |
DEGILXGFBNYPQN
|
8.1 | IC50 | 3 | — | |
RUKTWERRDLRGTH
|
8.1 | IC50 | 2 | — | |
YIKVOJGIIXEFHZ
|
8.1 | IC50 | 2 | — | |
ZBSQPLKGTYVAIB
|
8.1 | IC50 | 3 | — | |
DYNHJHQFHQTFTP
|
8.1 | Kd | 38 | — | |
FQYLJBVSYHZWLT
|
8.1 | Ki | 35 | Yes | |
HGBUMXKTCONBMP
|
8.1 | IC50 | 2 | — | |
KNARVZUUCLIBGV
|
8.1 | Ki | 33 | — | |
MCCCQFAOMZMZKE
|
8.1 | Ki | 52 | — | |
NPZSESRPQGYDMI
|
8.1 | IC50 | 3 | — | |
NXRSAGDKLSDJBW
|
8.1 | IC50 | 3 | — | |
RIJBDOXTEPVDPJ
|
8.1 | IC50 | 2 | — | |
XOMSZJJKZWBVAH
|
8.1 | IC50 | 3 | — | |
ZWVZORIKUNOTCS
|
8.1 | Ki | 69 | — | |
AYQXKPMEHPZRKR
|
8.1 | IC50 | 6 | — | |
RKIKBHDFIWQGHL
|
8.1 | IC50 | 3 | — | |
UIARLYUEJFELEN
|
8.1 | Kd | 289 | Yes | |
HHFHBMCHRPJYLX
|
8.1 | IC50 | 2 | — | |
PNBULRZVGIVARS
|
8.1 | IC50 | 3 | — | |
UHXOAJSLKLIFLJ
|
8.1 | IC50 | 2 | — | |
WDCXWYXCNRUVKU
|
8.1 | IC50 | 2 | — | |
ARFSIMCXZSKBGL
|
8.1 | IC50 | 3 | — | |
IXPSNGNVZSOSLS
|
8.1 | IC50 | 2 | — | |
MMZVTNYPOASLID
|
8.1 | IC50 | 3 | — | |
MPLLJMUCCXFTPL
|
8.1 | IC50 | 3 | — | |
NQWWOVKURVMLJC
|
8.1 | IC50 | 2 | — |