Target Details
| UniProt AC | P04629 |
|---|---|
| Gene Symbol | NTRK1 |
| Protein Name | High affinity nerve growth factor receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF13855 (LRR_8) PF16920 (LRRCT_2) PF07714 (PK_Tyr_Ser-Thr) PF18613 (TrkA_TMD) |
Summary
- Multi-target molecules 1,127
- Clinical molecules 52
- Avg pChEMBL 7.65
KEGG Pathways (11)
Associated Diseases (4)
Active Molecules (1,127)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ORQCQXMGDYAIOI
|
8.3 | IC50 | 6 | — | |
SEJGTFPOEJWEGG
|
8.3 | Kd | 149 | — | |
MBWHJBDHRADERX
|
8.3 | IC50 | 4 | — | |
SHRNMJSKKQHLKT
|
8.3 | IC50 | 4 | — | |
AFEWFPBEQADGDP
|
8.3 | IC50 | 3 | — | |
BTSSYEBPODNPPC
|
8.3 | IC50 | 3 | — | |
FOLXFWBVNHRGIV
|
8.3 | IC50 | 6 | — | |
GJQVPMWSXKFICV
|
8.3 | IC50 | 3 | — | |
OSDSLNBKGDENNX
|
8.3 | IC50 | 3 | — | |
WLAVZAAODLTUSW
|
8.3 | IC50 | 7 | — | |
KOZAUWSJLNLRBA
|
8.3 | IC50 | 2 | — | |
RKVKRYPLPNWYSE
|
8.3 | IC50 | 2 | — | |
YGJUUAYGTMKZBM
|
8.3 | IC50 | 2 | — | |
YOBIWCLAYQWPPW
|
8.3 | IC50 | 23 | — | |
ZQJUUOXBTWYBJE
|
8.3 | IC50 | 2 | — | |
NZFWYKNHDNDHFJ
|
8.3 | IC50 | 2 | — | |
OHIKHZFSGQMGGD
|
8.3 | IC50 | 5 | — | |
TYZOVRSMZFTMCR
|
8.3 | IC50 | 2 | — | |
WVXNSAVVKYZVOE
|
8.3 | IC50 | 92 | — | |
WYCSRUVPJUYDGP
|
8.2 | IC50 | 6 | — | |
YCLNSIOZHCMOPZ
|
8.2 | IC50 | 3 | — | |
FTAFQADCGCSJAH
|
8.2 | Kd | 3 | — | |
HGBUMXKTCONBMP
|
8.2 | IC50 | 2 | — | |
NLXBSFDJKLDGBF
|
8.2 | IC50 | 3 | — | |
VEFAIJAFTRTKSA
|
8.2 | IC50 | 2 | — | |
NYNZQNWKBKUAII
|
8.2 | IC50 | 4 | — | |
ALKJNCZNEOTEMP
|
8.2 | Kd | 55 | — | |
BPIWZDNVMQQBQX
|
8.2 | IC50 | 5 | — | |
BVOWDAQJDDEQSR
|
8.2 | IC50 | 3 | — | |
BYKSLICDLDTYLA
|
8.2 | IC50 | 3 | — | |
DADASRPKWOGKCU
|
8.2 | IC50 | 9 | — | |
KVAUYQFSODRWMC
|
8.2 | IC50 | 3 | — | |
OZFHIGAKHHLPEF
|
8.2 | IC50 | 3 | — | |
XYLJTJTWOPEYJR
|
8.2 | Kd | 5 | — | |
ZUSOUYHYDDCGIC
|
8.2 | IC50 | 4 | — | |
HGBUMXKTCONBMP
|
8.2 | IC50 | 2 | — | |
OEBIHOVSAMBXIB
|
8.2 | IC50 | 5 | — | |
PXRHKVCFGOFIIB
|
8.2 | IC50 | 2 | — | |
QHRTXUATNCWBBL
|
8.2 | IC50 | 2 | — | |
LKQSELSKVLDVHG
|
8.2 | IC50 | 2 | — | |
RBXYGQNZRVPDNB
|
8.2 | Ki | 34 | — | |
UDXFCKQHYWOCHB
|
8.2 | IC50 | 2 | — | |
HRNZKBRSPYYSBU
|
8.2 | IC50 | 2 | — | |
KNZNJSNITSGMNY
|
8.2 | IC50 | 2 | — | |
PBBXBBSBAJKYLC
|
8.2 | Kd | 3 | — | |
RFDMZDKRTPKABF
|
8.2 | IC50 | 3 | — | |
HQCZHKJSSABUNL
|
8.2 | IC50 | 2 | — | |
WVQWVRSXVXMJSE
|
8.2 | IC50 | 2 | — | |
AROVXDKGPGGRBP
|
8.2 | IC50 | 2 | — | |
RUKGVZRSXAHREZ
|
8.2 | IC50 | 2 | — |