Target Details
| UniProt AC | P04629 |
|---|---|
| Gene Symbol | NTRK1 |
| Protein Name | High affinity nerve growth factor receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF13855 (LRR_8) PF16920 (LRRCT_2) PF07714 (PK_Tyr_Ser-Thr) PF18613 (TrkA_TMD) |
Summary
- Multi-target molecules 1,127
- Clinical molecules 52
- Avg pChEMBL 7.65
KEGG Pathways (11)
Associated Diseases (4)
Active Molecules (1,127)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VWMOKEZPLSLTCC
|
8.5 | IC50 | 2 | — | |
ZGPOATYOAANSTK
|
8.5 | IC50 | 2 | — | |
LWMPTEZPBQOOSS
|
8.5 | IC50 | 3 | — | |
CDDGGDMFHAHNMC
|
8.5 | IC50 | 2 | — | |
KKDAOAYKDHBBPF
|
8.5 | IC50 | 2 | — | |
VELQWDIGSWMICE
|
8.5 | IC50 | 3 | — | |
COJJJJKXTCQCLW
|
8.4 | IC50 | 2 | — | |
GLRHZMRFCNDDIZ
|
8.4 | IC50 | 3 | — | |
HYUGTGGDEAGXJP
|
8.4 | IC50 | 11 | — | |
OPRRDZXAVINFQM
|
8.4 | IC50 | 2 | — | |
RKUGDCZKRYDCFQ
|
8.4 | IC50 | 2 | — | |
QTSGFRRREQFWGK
|
8.4 | IC50 | 3 | — | |
CXQHYVUVSFXTMY
|
8.4 | IC50 | 154 | — | |
FYNQXKHYYDAGJQ
|
8.4 | IC50 | 2 | — | |
MGUOEMOYOJLRIK
|
8.4 | IC50 | 2 | — | |
SQQPRORGDVPLSI
|
8.4 | IC50 | 4 | — | |
CNWIKXJNZAJWKF
|
8.4 | IC50 | 2 | — | |
HLAYAPGHRGSWFL
|
8.4 | IC50 | 2 | — | |
NYNZQNWKBKUAII
|
8.4 | IC50 | 3 | — | |
OMWFIVWGJYQGKO
|
8.4 | IC50 | 2 | — | |
WGPVINKDZIUGSE
|
8.4 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
8.4 | Kd | 213 | — | |
JJSRRCSUDKCPDQ
|
8.4 | Kd | 2 | — | |
LBVKEEFIPBQIMD
|
8.4 | Ki | 27 | — | |
ONSKSKMJNHEONW
|
8.4 | IC50 | 3 | Yes | |
ONSKSKMJNHEONW
|
8.4 | IC50 | 3 | Yes | |
QSGGLLCPVRJDDE
|
8.4 | IC50 | 4 | — | |
QTGGPQXZCLZMSN
|
8.4 | IC50 | 2 | — | |
WOXZGVPKIRNQQA
|
8.4 | IC50 | 3 | — | |
XIXBPLMTEROWPD
|
8.4 | IC50 | 3 | — | |
XYWFZNZTTHKFPM
|
8.4 | IC50 | 3 | — | |
ZSFJFWHLJJYXII
|
8.4 | IC50 | 2 | — | |
CCPZQDBNLBNUMF
|
8.4 | IC50 | 2 | — | |
LTWRCYLYOAZNPD
|
8.4 | IC50 | 2 | — | |
SXFVRQSCLPLRFN
|
8.4 | IC50 | 2 | — | |
BNPMMVDYMYENIM
|
8.4 | IC50 | 4 | — | |
RSRCBHDMPNBSTN
|
8.4 | IC50 | 2 | — | |
SSEZULRYZRTZPF
|
8.4 | IC50 | 3 | — | |
CTGZXMASDOJLIY
|
8.3 | IC50 | 2 | — | |
HFDYFIJWKPLZKI
|
8.3 | IC50 | 4 | — | |
JAKWBQOCOJPWEX
|
8.3 | IC50 | 2 | — | |
XZXHXSATPCNXJR
|
8.3 | Kd | 165 | Yes | |
AGHGCWANYKXNGS
|
8.3 | IC50 | 3 | — | |
IVHDXWQQZJTUMV
|
8.3 | IC50 | 2 | — | |
ZJGWNGRVSUFGBL
|
8.3 | IC50 | 3 | — | |
FDBFUEIJFKHRQU
|
8.3 | IC50 | 2 | — | |
VFYYBFAGANQTES
|
8.3 | IC50 | 2 | — | |
XXOVDEACMYYQHV
|
8.3 | IC50 | 3 | — | |
GYPXDOPFEWTHRF
|
8.3 | IC50 | 2 | — | |
LDKFMROXBKEDTL
|
8.3 | IC50 | 2 | — |