Target Details
| UniProt AC | P04629 |
|---|---|
| Gene Symbol | NTRK1 |
| Protein Name | High affinity nerve growth factor receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF13855 (LRR_8) PF16920 (LRRCT_2) PF07714 (PK_Tyr_Ser-Thr) PF18613 (TrkA_TMD) |
Summary
- Multi-target molecules 1,127
- Clinical molecules 52
- Avg pChEMBL 7.65
KEGG Pathways (11)
Associated Diseases (4)
Active Molecules (1,127)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKTKCWHAQWAVOW
|
8.6 | IC50 | 5 | — | |
HYHRGQAQGDRQRW
|
8.6 | IC50 | 2 | — | |
LNOMNJXKSIKMEZ
|
8.6 | IC50 | 2 | — | |
LTPMGUPHSVPNRT
|
8.6 | IC50 | 3 | — | |
NXPHBBCDRJWBHG
|
8.6 | IC50 | 3 | — | |
OUBJSHKDVMRZQJ
|
8.6 | IC50 | 5 | — | |
POXSFRWIBWNONT
|
8.6 | IC50 | 3 | — | |
QPQWYASIHZVVSO
|
8.6 | IC50 | 2 | — | |
QRMNFHGVKRGQBQ
|
8.6 | IC50 | 3 | — | |
RFPOGGXYJDJURU
|
8.6 | IC50 | 2 | — | |
RLHGMHDDJDTUOF
|
8.6 | IC50 | 3 | — | |
SCHLJLHHIALWBK
|
8.6 | IC50 | 5 | — | |
SXRLSRMWBAVNFG
|
8.6 | IC50 | 3 | — | |
VROSTPWCFHKXPW
|
8.6 | IC50 | 4 | — | |
WHODNMAIHAPRJL
|
8.6 | IC50 | 3 | — | |
WJAQYAUNJKXATP
|
8.6 | IC50 | 3 | — | |
XNIIBBGPPVUEJT
|
8.6 | IC50 | 2 | — | |
ISCJKTYZQXHEBM
|
8.6 | IC50 | 2 | — | |
MCGUMEZGZDHGBX
|
8.6 | IC50 | 2 | — | |
PJFDUIVXIFHGSE
|
8.6 | IC50 | 3 | — | |
VQFKVNURGWYBCE
|
8.6 | IC50 | 2 | — | |
ZBTADFYRGPHVEO
|
8.6 | IC50 | 2 | — | |
ZRFDOJZJWLQZJB
|
8.6 | IC50 | 2 | — | |
HRNZKBRSPYYSBU
|
8.5 | IC50 | 2 | — | |
OTBHAYAYGBSHCF
|
8.5 | Kd | 2 | — | |
VBDSRXYVIRRJJF
|
8.5 | IC50 | 2 | — | |
AYEUXZLSMOOOKC
|
8.5 | IC50 | 2 | — | |
COGWCSCPIYIKOV
|
8.5 | IC50 | 3 | — | |
DIGOSQFGMNNGOP
|
8.5 | IC50 | 3 | — | |
FOORTUZRHZKYIF
|
8.5 | IC50 | 3 | — | |
GUYRCSVNTIHWAI
|
8.5 | IC50 | 3 | — | |
HIHOEGPXVVKJPP
|
8.5 | IC50 | 10 | — | |
HKSZLNNOFSGOKW
|
8.5 | IC50 | 118 | — | |
HNLSVESOKZTLCF
|
8.5 | IC50 | 2 | — | |
HXGMCPSJILOUIU
|
8.5 | IC50 | 2 | — | |
KKQVKLFNDUPHNK
|
8.5 | IC50 | 2 | — | |
OQULCJFCULISIS
|
8.5 | IC50 | 3 | — | |
PDOQBOJDRPLBQU
|
8.5 | IC50 | 21 | — | |
RKERQEKFTWWCEY
|
8.5 | IC50 | 4 | — | |
VEJZPSCYDZCQLW
|
8.5 | IC50 | 2 | — | |
VFWZEMIPXRZJDU
|
8.5 | IC50 | 2 | — | |
GZISOCBRRUTHKW
|
8.5 | IC50 | 2 | — | |
GZISOCBRRUTHKW
|
8.5 | IC50 | 2 | — | |
WIVNLRJLMBFTMY
|
8.5 | IC50 | 3 | — | |
QONPPIZSNSSCSK
|
8.5 | Ki | 45 | Yes | |
HRNZKBRSPYYSBU
|
8.5 | IC50 | 2 | — | |
MEHIPRLZSVZRLS
|
8.5 | IC50 | 3 | — | |
UEWLKIVHINNLJX
|
8.5 | IC50 | 2 | — | |
OBXXVELGHXKSST
|
8.5 | IC50 | 3 | — | |
VQFPMVKAMVDQNA
|
8.5 | IC50 | 2 | — |