Target Details
| UniProt AC | P04629 |
|---|---|
| Gene Symbol | NTRK1 |
| Protein Name | High affinity nerve growth factor receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF13855 (LRR_8) PF16920 (LRRCT_2) PF07714 (PK_Tyr_Ser-Thr) PF18613 (TrkA_TMD) |
Summary
- Multi-target molecules 1,127
- Clinical molecules 52
- Avg pChEMBL 7.65
KEGG Pathways (11)
Associated Diseases (4)
Active Molecules (1,127)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MTCHBJMHQSHCIK
|
8.7 | IC50 | 3 | — | |
PHKCNLPGORPBKO
|
8.7 | IC50 | 3 | — | |
RPNUUULYRBUSBJ
|
8.7 | IC50 | 3 | — | |
WDZMQMMLPZNCPU
|
8.7 | IC50 | 3 | — | |
BCNBASJWOYJQGY
|
8.7 | IC50 | 2 | — | |
DGVVSWFLMBWPNY
|
8.7 | IC50 | 2 | — | |
FZBVNCFBCNXULH
|
8.7 | IC50 | 18 | — | |
MCGUMEZGZDHGBX
|
8.7 | IC50 | 2 | — | |
QTJHBCKEZSYXTG
|
8.7 | IC50 | 3 | — | |
WAAWHVXSMHHZCZ
|
8.7 | IC50 | 2 | — | |
WAHDCQYLZWQRBB
|
8.7 | IC50 | 2 | — | |
WUOOWFKJQHKXHK
|
8.7 | IC50 | 4 | — | |
YISMQBFJYDFMAL
|
8.7 | IC50 | 46 | — | |
YTPXNCADDOOFPA
|
8.7 | Kd | 2 | — | |
WUASJGDLFRRAKD
|
8.7 | IC50 | 2 | — | |
FPPLXTGCMYMFDI
|
8.7 | IC50 | 2 | — | |
ISCJKTYZQXHEBM
|
8.7 | IC50 | 2 | — | |
MJTXQVLFZPHAOU
|
8.7 | IC50 | 2 | — | |
OTCSCPHWCZZRDC
|
8.7 | IC50 | 2 | — | |
RFOHHTZHDHDNPM
|
8.7 | IC50 | 3 | — | |
UEHKWTJSMNTTCC
|
8.7 | IC50 | 2 | — | |
IFTKTMZJBXEOCK
|
8.7 | IC50 | 2 | — | |
LQRYCJFXMJIIPW
|
8.7 | IC50 | 2 | — | |
RSFALMGMTQBFJZ
|
8.6 | Kd | 9 | — | |
WSTUJEXAPHIEIM
|
8.6 | IC50 | 10 | — | |
XWDLDVQSUXONBG
|
8.6 | IC50 | 2 | — | |
LJJBCTSKXBRDPV
|
8.6 | IC50 | 2 | — | |
OXVCBPXLNVQEGM
|
8.6 | IC50 | 2 | — | |
QXTPBRKTCUTGBZ
|
8.6 | IC50 | 2 | — | |
RFSSOUGNOQIPBG
|
8.6 | IC50 | 3 | — | |
RZRSOLZCLWVUTL
|
8.6 | IC50 | 2 | — | |
UEHKWTJSMNTTCC
|
8.6 | IC50 | 2 | — | |
UMZFBMAHLWQSBF
|
8.6 | IC50 | 4 | — | |
CWZWSPLRRXTDRE
|
8.6 | IC50 | 2 | — | |
IVHDXWQQZJTUMV
|
8.6 | IC50 | 2 | — | |
KKYPRNBBPBRJQX
|
8.6 | Ki | 40 | — | |
OJEYPUNKJUVVID
|
8.6 | IC50 | 2 | — | |
STZNSTWBJYAKHQ
|
8.6 | IC50 | 3 | — | |
UYIANZRYPSGDFM
|
8.6 | IC50 | 2 | — | |
AUTGNDRENPBZKA
|
8.6 | Kd | 3 | — | |
CXTZBLHNTGMZDF
|
8.6 | IC50 | 2 | — | |
XSWLSCPOLAJGJH
|
8.6 | IC50 | 2 | — | |
SNEMCZIOBDJWLQ
|
8.6 | IC50 | 3 | — | |
IAJVWMAWMQNCEM
|
8.6 | IC50 | 2 | — | |
IYYCEJNOEXGZEZ
|
8.6 | IC50 | 3 | — | |
KDFREDAEEQQCFD
|
8.6 | IC50 | 3 | — | |
LBVKEEFIPBQIMD
|
8.6 | IC50 | 4 | — | |
MLJKSWPNIQXPCX
|
8.6 | IC50 | 2 | — | |
ZPDUZRKQTNYYQZ
|
8.6 | IC50 | 2 | — | |
GCAJYDBNZMKHTH
|
8.6 | IC50 | 3 | — |