Target Details
| UniProt AC | P04629 |
|---|---|
| Gene Symbol | NTRK1 |
| Protein Name | High affinity nerve growth factor receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF13855 (LRR_8) PF16920 (LRRCT_2) PF07714 (PK_Tyr_Ser-Thr) PF18613 (TrkA_TMD) |
Summary
- Multi-target molecules 1,127
- Clinical molecules 52
- Avg pChEMBL 7.65
KEGG Pathways (11)
Associated Diseases (4)
Active Molecules (1,127)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZXDAOGSITPXTJV
|
9.2 | IC50 | 2 | — | |
IEBZBPYYZNDTMO
|
9.2 | IC50 | 4 | — | |
MPTHHGRJSLVPSX
|
9.2 | IC50 | 2 | — | |
HACQCZAUTIOAKZ
|
9.2 | IC50 | 2 | — | |
LEOYYKMTNGOPRD
|
9.2 | IC50 | 2 | — | |
RFCPQXPQIFCVHE
|
9.2 | IC50 | 3 | — | |
RWWNIGJTZLTACI
|
9.2 | IC50 | 2 | — | |
WPQQNUFDOKQHRQ
|
9.2 | IC50 | 2 | — | |
XDTRTPIHJGKMHO
|
9.2 | IC50 | 2 | — | |
XJIIVPVOGYFVME
|
9.2 | Kd | 3 | — | |
NFVNVIQUEXSEFR
|
9.1 | IC50 | 4 | — | |
IXJWJBUYPZPUQB
|
9.1 | IC50 | 2 | — | |
BLGCSOKKBWHJMB
|
9.1 | Kd | 2 | — | |
GNNDEPIMDAZHRQ
|
9.1 | IC50 | 6 | — | |
IBWUYNSLISMPFY
|
9.1 | IC50 | 4 | — | |
INNUOJBTOZECFW
|
9.1 | Kd | 2 | — | |
BCFGWXGYMCPFQX
|
9.1 | IC50 | 2 | — | |
GSCBTVAYMDWDTL
|
9.1 | IC50 | 2 | — | |
TWRNOCZDGWHEGC
|
9.1 | IC50 | 3 | — | |
WDEZXSKNKVBRGN
|
9.1 | IC50 | 2 | — | |
WRXZQYJJPXFOIB
|
9.1 | IC50 | 3 | — | |
DJADXHQZNZDUAO
|
9.0 | IC50 | 2 | — | |
KUSZMPYJQONYEI
|
9.0 | IC50 | 2 | — | |
RDRCKVYUJKQGJL
|
9.0 | IC50 | 2 | — | |
CFVOAVDAPUQRNK
|
9.0 | IC50 | 4 | Yes | |
CFVOAVDAPUQRNK
|
9.0 | IC50 | 5 | Yes | |
CXVBPWYIUWZVJO
|
9.0 | IC50 | 4 | — | |
FWANKJAOTQAHHR
|
9.0 | Kd | 2 | — | |
HAYYBYPASCDWEQ
|
9.0 | IC50 | 47 | — | |
HIKKZNRTRHJLST
|
9.0 | IC50 | 3 | — | |
LJJBCTSKXBRDPV
|
9.0 | IC50 | 2 | — | |
PXPRXTYAUNNAHY
|
9.0 | IC50 | 3 | — | |
UQKLTKAHTNLXPA
|
9.0 | IC50 | 5 | — | |
WAIWXFGIIWQVMF
|
9.0 | IC50 | 2 | — | |
XEWYVOAMYRLGMQ
|
9.0 | IC50 | 3 | — | |
MBZCRLUONJJYJU
|
9.0 | IC50 | 2 | — | |
AKARKHHDGYZKIF
|
9.0 | IC50 | 5 | — | |
BKQWHAVIQWXFBE
|
9.0 | IC50 | 2 | — | |
GGJNWRFNZLJBRQ
|
9.0 | IC50 | 2 | — | |
PWCNVYNJXOVGLO
|
9.0 | IC50 | 4 | — | |
RJWUXXDSPBTHTI
|
9.0 | IC50 | 2 | — | |
RJWUXXDSPBTHTI
|
9.0 | IC50 | 2 | — | |
VTUVGNKQBUVKIW
|
9.0 | IC50 | 2 | — | |
XCBGRHHBQFJBBF
|
9.0 | IC50 | 2 | — | |
LRJJEMRURFIKDD
|
8.9 | IC50 | 6 | — | |
XHJBITNPWPZMGB
|
8.9 | IC50 | 2 | — | |
XHJBITNPWPZMGB
|
8.9 | IC50 | 2 | — | |
ISGDOVGHVRHZFY
|
8.9 | IC50 | 2 | — | |
KOZFSFOOLUUIGY
|
8.9 | IC50 | 15 | Yes | |
SGCBBVKTBTZXBX
|
8.9 | IC50 | 2 | — |