Target Details
| UniProt AC | P04629 |
|---|---|
| Gene Symbol | NTRK1 |
| Protein Name | High affinity nerve growth factor receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF13855 (LRR_8) PF16920 (LRRCT_2) PF07714 (PK_Tyr_Ser-Thr) PF18613 (TrkA_TMD) |
Summary
- Multi-target molecules 1,127
- Clinical molecules 52
- Avg pChEMBL 7.65
KEGG Pathways (11)
Associated Diseases (4)
Active Molecules (1,127)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PWRMINAVABZMME
|
7.4 | IC50 | 2 | — | |
AROVXDKGPGGRBP
|
7.4 | IC50 | 2 | — | |
DSYTUISCOWQTPC
|
7.4 | IC50 | 2 | — | |
GCIKSSRWRFVXBI
|
7.4 | Kd | 109 | Yes | |
GRFSXOHKPKDKRB
|
7.4 | IC50 | 2 | — | |
NJAVDBDBSBBDKS
|
7.4 | IC50 | 3 | — | |
XIWVEZNCIIVZQH
|
7.4 | IC50 | 3 | — | |
YHWLSZUFSOTFQF
|
7.4 | IC50 | 2 | — | |
OGKQRFCRLNVUPG
|
7.4 | IC50 | 3 | — | |
SOLRFWOVULTERW
|
7.4 | IC50 | 2 | — | |
QESFWVGTAWQADH
|
7.4 | IC50 | 3 | — | |
QJIVDCJIPGAKQZ
|
7.4 | Ki | 25 | — | |
YGUHZTGUYHUMMF
|
7.4 | IC50 | 3 | — | |
DWRDCEAGIMHGDA
|
7.4 | IC50 | 3 | — | |
NOWAWLXYDFVEIE
|
7.4 | IC50 | 3 | — | |
UQLJOQKYBXUIFI
|
7.4 | IC50 | 3 | — | |
DUJMHEBMAPADNS
|
7.4 | IC50 | 4 | — | |
MSDSJOCXJMWGST
|
7.4 | IC50 | 2 | — | |
QJMSOLBVHUXFJN
|
7.4 | IC50 | 3 | — | |
IYHJCLOZCBCODN
|
7.4 | IC50 | 2 | — | |
UEXYLQPMBYMXCX
|
7.4 | IC50 | 2 | — | |
NKAVBKULSDGBBI
|
7.3 | IC50 | 2 | — | |
WRBFVDOQDFYXNC
|
7.3 | IC50 | 2 | — | |
ZFESQIANWCIUCE
|
7.3 | IC50 | 2 | — | |
JGEBLDKNWBUGRZ
|
7.3 | IC50 | 20 | Yes | |
KGBCNTOGVNRFPN
|
7.3 | IC50 | 3 | — | |
LTTAHJWMYYUXHI
|
7.3 | IC50 | 2 | — | |
JSSACTCBXIXNAA
|
7.3 | IC50 | 2 | — | |
IHXVXJVXFFLYQL
|
7.3 | IC50 | 2 | — | |
ONENEBSQEBHUSO
|
7.3 | IC50 | 2 | — | |
UWWDGFCKMLJGIQ
|
7.3 | IC50 | 3 | — | |
VYCGSIVULARDLE
|
7.3 | IC50 | 2 | — | |
COXSWEZHBTXILY
|
7.3 | IC50 | 3 | — | |
FLEAYYMORDPWAJ
|
7.3 | Ki | 90 | — | |
IKENQUDOTQBCJH
|
7.3 | Kd | 18 | — | |
JREJWPGPNAQDPQ
|
7.3 | IC50 | 3 | — | |
JZORFWRZZRNPER
|
7.3 | IC50 | 3 | — | |
LYADGAGFYYXXIO
|
7.3 | IC50 | 82 | — | |
MQRDVGBWWVWMEN
|
7.3 | Ki | 47 | — | |
YUDZZEAZLCNKOZ
|
7.3 | IC50 | 3 | — | |
AUFWLXVVSPEREI
|
7.3 | IC50 | 3 | — | |
LNSSOTMJRRLINS
|
7.3 | IC50 | 2 | — | |
NFYFLWXBIHYPII
|
7.3 | IC50 | 3 | — | |
ZKDXRFMOHZVXSG
|
7.3 | IC50 | 13 | Yes | |
JLVUEKVUGINUJP
|
7.3 | IC50 | 3 | — | |
MYVXPLSILQDDFA
|
7.3 | IC50 | 2 | — | |
PEUXFCOIQKEZCE
|
7.3 | IC50 | 2 | — | |
PFNIFDHHWXBYCS
|
7.3 | IC50 | 3 | — | |
TUBXJQSNTKADJB
|
7.3 | IC50 | 5 | — | |
VRCBGBBYFHLJRE
|
7.3 | IC50 | 5 | — |