Target Details
| UniProt AC | P04629 |
|---|---|
| Gene Symbol | NTRK1 |
| Protein Name | High affinity nerve growth factor receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF13855 (LRR_8) PF16920 (LRRCT_2) PF07714 (PK_Tyr_Ser-Thr) PF18613 (TrkA_TMD) |
Summary
- Multi-target molecules 1,127
- Clinical molecules 52
- Avg pChEMBL 7.65
KEGG Pathways (11)
Associated Diseases (4)
Active Molecules (1,127)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HYHRGQAQGDRQRW
|
7.6 | IC50 | 2 | — | |
JTGBHZLCDFMSGY
|
7.6 | IC50 | 2 | — | |
JXPQCRCHIRKWDH
|
7.6 | IC50 | 3 | — | |
UXQSAGZIRLAKKX
|
7.6 | IC50 | 2 | — | |
XNLDXKJZCGYOAU
|
7.6 | IC50 | 5 | — | |
NBAROHPFFUMFNW
|
7.5 | IC50 | 3 | — | |
PHXJVRSECIGDHY
|
7.5 | IC50 | 59 | — | |
BIJVEGOYPDBWSR
|
7.5 | IC50 | 2 | — | |
CGLJKJPXQBOLMC
|
7.5 | IC50 | 3 | — | |
DHEFBJXZYSKWIF
|
7.5 | IC50 | 2 | — | |
HDMQHDILMFAMEX
|
7.5 | IC50 | 3 | — | |
NLFFJXBANCVTJV
|
7.5 | IC50 | 3 | — | |
NWCVGFXDQDGLSM
|
7.5 | IC50 | 3 | — | |
IHNLQGSBVSZMGR
|
7.5 | IC50 | 3 | — | |
VYTKFXBQPJOMSD
|
7.5 | IC50 | 2 | — | |
AMHUBFWCCMLLCJ
|
7.5 | IC50 | 15 | — | |
AOJFJIKCNFEJMA
|
7.5 | IC50 | 2 | — | |
DLPATUQBJYDVLH
|
7.5 | IC50 | 3 | — | |
IQEIAIXWJHRRRI
|
7.5 | IC50 | 3 | — | |
TVJRDCQUZMGBAB
|
7.5 | IC50 | 13 | — | |
UWXAGMXVWDWRRX
|
7.5 | IC50 | 2 | — | |
JWILUIVAYLRFIY
|
7.5 | IC50 | 14 | — | |
KOCGMVOWSRIEAZ
|
7.5 | IC50 | 2 | — | |
MSWOWUREQODTRO
|
7.5 | IC50 | 11 | — | |
OKICNWNFGLYZRW
|
7.5 | IC50 | 2 | — | |
XKFTZKGMDDZMJI
|
7.5 | IC50 | 8 | Yes | |
XUFRAOMXWJULLM
|
7.5 | IC50 | 2 | — | |
CAHNFGYWMWNXMR
|
7.5 | IC50 | 9 | — | |
CPVWZVNGLWUDCJ
|
7.5 | Kd | 2 | — | |
DYIZMEHLAPKNNN
|
7.5 | IC50 | 3 | — | |
LMFNJXLDISVWLF
|
7.5 | IC50 | 5 | — | |
RAVQVOSIVIEHCN
|
7.5 | IC50 | 3 | — | |
KEMAQYFMSWCNPP
|
7.5 | IC50 | 2 | — | |
HTZHPXKKPOLGTR
|
7.5 | IC50 | 9 | — | |
LYGAZBUPOLXLRE
|
7.5 | IC50 | 2 | — | |
QXACJSRSZMVUQK
|
7.5 | IC50 | 2 | — | |
UUEKSMCPYQPFQV
|
7.5 | IC50 | 2 | — | |
TUPCMOPJDADTAY
|
7.5 | IC50 | 2 | — | |
GVXOANLMUATURP
|
7.5 | IC50 | 2 | — | |
NXSJMRCTGYTSTK
|
7.5 | Kd | 200 | — | |
QHXBWJSQXSYAGG
|
7.5 | IC50 | 16 | — | |
QXQMNBCLKYICGU
|
7.5 | IC50 | 3 | — | |
SAMAJBJTKDGWPS
|
7.5 | IC50 | 2 | — | |
XDWPKPYJLQHIGW
|
7.5 | IC50 | 3 | — | |
XRPNCCIJNVBSFF
|
7.5 | IC50 | 2 | — | |
CUAZXICLJJKGFD
|
7.4 | IC50 | 2 | — | |
PCIMPOMGHFNGMS
|
7.4 | IC50 | 7 | — | |
ZFKQQXLECNVLOF
|
7.4 | IC50 | 7 | — | |
CUAZXICLJJKGFD
|
7.4 | IC50 | 2 | — | |
MMVLETOTGHDVPQ
|
7.4 | IC50 | 7 | — |