Target Details
| UniProt AC | P04629 |
|---|---|
| Gene Symbol | NTRK1 |
| Protein Name | High affinity nerve growth factor receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF13855 (LRR_8) PF16920 (LRRCT_2) PF07714 (PK_Tyr_Ser-Thr) PF18613 (TrkA_TMD) |
Summary
- Multi-target molecules 1,127
- Clinical molecules 52
- Avg pChEMBL 7.65
KEGG Pathways (11)
Associated Diseases (4)
Active Molecules (1,127)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YVDCINMNXNRYMU
|
7.7 | IC50 | 2 | — | |
FULRLUZBOZERKQ
|
7.7 | IC50 | 3 | — | |
HEHIDXMRYPIDIV
|
7.7 | IC50 | 3 | — | |
MVNWGIDWOQYDJB
|
7.7 | IC50 | 3 | — | |
SPBLOIGTOGQHKL
|
7.7 | IC50 | 2 | — | |
SRQQRYTWWRXHKL
|
7.7 | IC50 | 2 | — | |
UBPYILGKFZZVDX
|
7.7 | IC50 | 130 | Yes | |
ZWYZLHQIBDNFFL
|
7.7 | IC50 | 2 | — | |
PDPJLIBDEWXTAI
|
7.7 | IC50 | 2 | — | |
XCCJJNIKWGXTSP
|
7.7 | IC50 | 2 | — | |
DUAIEVYTIKHMGW
|
7.6 | IC50 | 3 | — | |
LSEAQLOYCHTEOK
|
7.6 | IC50 | 10 | — | |
OTXIWIXBZNTJGG
|
7.6 | IC50 | 3 | — | |
PBBRUKZHVDWECM
|
7.6 | IC50 | 3 | — | |
RHGGEGBXSUZHQZ
|
7.6 | IC50 | 3 | — | |
RKRWQXHCILAOQU
|
7.6 | IC50 | 2 | — | |
ZYEIOSXTPZLYKG
|
7.6 | IC50 | 3 | — | |
GAXVYKWKQSGVIF
|
7.6 | IC50 | 2 | — | |
DJYWRQSMWCFDQX
|
7.6 | IC50 | 3 | — | |
IIXWYSCJSQVBQM
|
7.6 | IC50 | 18 | — | |
LASRMRBYBVIFQT
|
7.6 | IC50 | 2 | — | |
PWKWAKJEHNCJDL
|
7.6 | IC50 | 3 | — | |
VXYZCOCRVAQWBG
|
7.6 | IC50 | 15 | — | |
LAJAAZMLLWPYKV
|
7.6 | IC50 | 2 | — | |
KBBXMARUHDVNOM
|
7.6 | IC50 | 2 | — | |
OSVUGUHRKMMBSE
|
7.6 | Kd | 170 | — | |
PKVRKFYLJXIDJS
|
7.6 | IC50 | 3 | — | |
UOOZSMNSBYVUGZ
|
7.6 | Ki | 32 | — | |
VGEDWYCIYWKLHV
|
7.6 | IC50 | 2 | — | |
WZZBNLYBHUDSHF
|
7.6 | IC50 | 3 | — | |
ZCCJKVBTHCOISJ
|
7.6 | Ki | 46 | — | |
VKGDZKKOMMTJBF
|
7.6 | IC50 | 2 | — | |
APPXQUDJLJXULP
|
7.6 | IC50 | 47 | — | |
BXKMPBRSKYRFNY
|
7.6 | IC50 | 2 | — | |
IKJRKNZBCCOIFV
|
7.6 | IC50 | 3 | — | |
JRLOPMVTMMPZMV
|
7.6 | IC50 | 3 | — | |
SBVICLYVLJMIDO
|
7.6 | IC50 | 2 | — | |
UFOSAOVNENJKCZ
|
7.6 | IC50 | 3 | — | |
XCLDJXYOZUVDAT
|
7.6 | IC50 | 2 | — | |
ADHIYNKWKQQREL
|
7.6 | IC50 | 3 | — | |
BNRXMSGHPVYSDK
|
7.6 | IC50 | 24 | — | |
CZZPKZAXQSRAJE
|
7.6 | IC50 | 2 | — | |
DUAIEVYTIKHMGW
|
7.6 | IC50 | 3 | — | |
IGJZBYFJOGZJQO
|
7.6 | IC50 | 3 | — | |
IXPTZPMMOJWPBZ
|
7.6 | IC50 | 2 | — | |
PRZQRZSCFWKYBL
|
7.6 | IC50 | 3 | — | |
YICDYXUSGXQKLK
|
7.6 | IC50 | 2 | — | |
BNXYQBUYYXJKBW
|
7.6 | IC50 | 3 | — | |
DOWWFGLYJNBUSG
|
7.6 | IC50 | 4 | — | |
FGRVKMDGFGXLDX
|
7.6 | IC50 | 5 | — |