Target Details
| UniProt AC | P04629 |
|---|---|
| Gene Symbol | NTRK1 |
| Protein Name | High affinity nerve growth factor receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF13855 (LRR_8) PF16920 (LRRCT_2) PF07714 (PK_Tyr_Ser-Thr) PF18613 (TrkA_TMD) |
Summary
- Multi-target molecules 1,127
- Clinical molecules 52
- Avg pChEMBL 7.65
KEGG Pathways (11)
Associated Diseases (4)
Active Molecules (1,127)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IXPTZPMMOJWPBZ
|
7.8 | IC50 | 2 | — | |
MLXSJDISJFMJES
|
7.8 | IC50 | 2 | — | |
SVIHXEVVNNRVEM
|
7.8 | IC50 | 2 | — | |
XDPZIMBOLIRSMT
|
7.8 | IC50 | 2 | — | |
DIXMBHMNEHPFCX
|
7.8 | IC50 | 12 | — | |
FNUKQFDNWARLGZ
|
7.8 | IC50 | 2 | — | |
HIVVRJXSFJMYEH
|
7.8 | IC50 | 3 | — | |
OEQLJMGIZHYYCW
|
7.8 | IC50 | 3 | — | |
UGWUALPBTGHKQH
|
7.8 | IC50 | 2 | — | |
VDWUFEKTWXEZTN
|
7.8 | IC50 | 3 | — | |
XHKNPVMZBCKSLF
|
7.8 | IC50 | 3 | — | |
CHFWYNNEXACTNW
|
7.8 | IC50 | 2 | — | |
NQAMVBJCWLPNJI
|
7.8 | IC50 | 2 | — | |
PJDOSMIVVUPROI
|
7.8 | IC50 | 2 | — | |
WHPGNGKXSZTMOD
|
7.8 | IC50 | 3 | — | |
GMVQPWCWWLPOQT
|
7.8 | IC50 | 9 | Yes | |
HVJJVFGMNLSTHA
|
7.8 | IC50 | 3 | — | |
FBJDKSAIBPOAQN
|
7.7 | IC50 | 2 | — | |
LYXIOTQYDYQDCB
|
7.7 | IC50 | 2 | — | |
MZKCTWNUCVKGCB
|
7.7 | IC50 | 9 | — | |
PZWKQEQSYRXWEJ
|
7.7 | IC50 | 2 | — | |
UCEDODRINHMTIB
|
7.7 | IC50 | 3 | — | |
UHJMMAFUNGKSLA
|
7.7 | IC50 | 2 | — | |
VSKPQPVBEFIGBJ
|
7.7 | IC50 | 3 | — | |
ZHOXAGNPCZTRBN
|
7.7 | IC50 | 3 | — | |
OXPRNEDRKPNLKW
|
7.7 | IC50 | 3 | — | |
DSSNAGYVGTYAGH
|
7.7 | IC50 | 10 | — | |
LOJQAAWJKRUOCL
|
7.7 | IC50 | 2 | — | |
MVPRWLBKNHWFPM
|
7.7 | IC50 | 6 | — | |
QQIQOMIKWUAMAA
|
7.7 | IC50 | 7 | — | |
WXAPPLXJQZTWJT
|
7.7 | IC50 | 3 | — | |
XVXTUHJPGWZCKO
|
7.7 | IC50 | 2 | — | |
SPGMDULIPMJULM
|
7.7 | IC50 | 2 | — | |
AADXSEVDTNPICQ
|
7.7 | IC50 | 2 | — | |
FUJQPFBKDKKXHX
|
7.7 | IC50 | 3 | — | |
GCYXEGSPUDSZJY
|
7.7 | Ki | 82 | — | |
HXGMCPSJILOUIU
|
7.7 | IC50 | 2 | — | |
PFBAATFKRNWAOG
|
7.7 | IC50 | 3 | — | |
UGEJLCNSVIVALC
|
7.7 | Ki | 41 | — | |
ULHGAQSVFPOUDY
|
7.7 | Ki | 43 | — | |
ULMCFLZUGRSEQA
|
7.7 | Ki | 17 | — | |
VMYCKCWYEIGQOV
|
7.7 | IC50 | 3 | — | |
WLLYMKLGVMLEFL
|
7.7 | IC50 | 2 | — | |
WOKJIIMDDCFJJH
|
7.7 | IC50 | 2 | — | |
AKMHYAGNOVKYER
|
7.7 | IC50 | 3 | — | |
DZAPMAGSEHVBQI
|
7.7 | IC50 | 3 | — | |
HUMIANOGLZOVBP
|
7.7 | IC50 | 2 | — | |
IJEQTEVIXYPEPD
|
7.7 | IC50 | 3 | — | |
KIEKEVDZKHCHOX
|
7.7 | IC50 | 2 | — | |
NNDVLAPMFXYAAS
|
7.7 | IC50 | 3 | — |