Target Details
| UniProt AC | P04629 |
|---|---|
| Gene Symbol | NTRK1 |
| Protein Name | High affinity nerve growth factor receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF13855 (LRR_8) PF16920 (LRRCT_2) PF07714 (PK_Tyr_Ser-Thr) PF18613 (TrkA_TMD) |
Summary
- Multi-target molecules 1,127
- Clinical molecules 52
- Avg pChEMBL 7.65
KEGG Pathways (11)
Associated Diseases (4)
Active Molecules (1,127)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZYIYWAPOCQBZSM
|
7.9 | IC50 | 2 | — | |
QVEBEDUBSUAZSH
|
7.9 | IC50 | 2 | — | |
BNMXHZKBTHOMBT
|
7.9 | IC50 | 3 | — | |
CYMJCVZONIXLKV
|
7.9 | IC50 | 3 | — | |
FAYAUAZLLLJJGH
|
7.9 | IC50 | 36 | Yes | |
NIFOBCJOHDKDIO
|
7.9 | IC50 | 3 | — | |
ZCCPLJOKGAACRT
|
7.9 | Kd | 599 | — | |
DPMQHTABGLRCQK
|
7.9 | IC50 | 5 | — | |
GSRZAXNWBZUUOT
|
7.9 | IC50 | 2 | — | |
IXPTZPMMOJWPBZ
|
7.9 | IC50 | 2 | — | |
RURCYYRVPUXVMX
|
7.9 | IC50 | 2 | — | |
LZJSAQIUAQDIAJ
|
7.9 | IC50 | 2 | — | |
ODVQNAZETSWKTM
|
7.9 | IC50 | 2 | — | |
TZXUJWHUDYHLGV
|
7.9 | IC50 | 2 | — | |
VMUKQRHNARMWLU
|
7.9 | IC50 | 2 | — | |
XKZINYYXWJEYEL
|
7.9 | Ki | 37 | — | |
AGNJXIYEGHWROL
|
7.9 | IC50 | 2 | — | |
FGZBDTYJIFVMCX
|
7.9 | IC50 | 3 | — | |
GEGAHMIBPFSFDY
|
7.9 | IC50 | 3 | — | |
GPVOGAITWLZNLK
|
7.9 | IC50 | 2 | — | |
JWBXEWFBXJNXBU
|
7.9 | IC50 | 4 | — | |
KOZFSFOOLUUIGY
|
7.9 | IC50 | 26 | — | |
KOZFSFOOLUUIGY
|
7.9 | IC50 | 88 | Yes | |
OIBHJHBQKAMDOY
|
7.9 | IC50 | 3 | — | |
VVGBSNRZVJGQFL
|
7.9 | IC50 | 5 | — | |
AVDISIKMHVXATN
|
7.9 | IC50 | 2 | — | |
BGQOUQWQPRPBKN
|
7.9 | IC50 | 7 | — | |
CGCAUJNXCRBIGQ
|
7.9 | IC50 | 2 | — | |
JFSJERWBWSRHJA
|
7.9 | IC50 | 3 | — | |
LIKCNXUVDQCOAH
|
7.8 | IC50 | 3 | — | |
OIZJENLXXROKNH
|
7.8 | IC50 | 3 | — | |
SAAVSPULBSDEOY
|
7.8 | IC50 | 2 | — | |
VSWZVURJMXGYKU
|
7.8 | IC50 | 2 | — | |
ZXXLTAJEIQMHMD
|
7.8 | IC50 | 3 | — | |
JDIGZDKHSLPKGP
|
7.8 | IC50 | 2 | — | |
IPFQMFOPNXOZJB
|
7.8 | IC50 | 2 | — | |
LTWSDRXXRPCLNY
|
7.8 | IC50 | 3 | — | |
REWSLBJUSMBYHR
|
7.8 | IC50 | 3 | — | |
SBVICLYVLJMIDO
|
7.8 | IC50 | 2 | — | |
UGWBYFCYZUIYGV
|
7.8 | IC50 | 2 | — | |
YYCRCMXHHDOWEV
|
7.8 | IC50 | 2 | — | |
PZGCHNDBATUPDX
|
7.8 | IC50 | 2 | — | |
GALVWTFFXPRMQM
|
7.8 | Ki | 20 | — | |
IBCNIGDAKZQAFQ
|
7.8 | IC50 | 2 | — | |
LZFGLNXIDZGIEG
|
7.8 | IC50 | 3 | — | |
ORGAJFAIHVVNPY
|
7.8 | IC50 | 2 | — | |
SICRRVUVAIRMQG
|
7.8 | IC50 | 2 | — | |
VCFDMLBPASGZTP
|
7.8 | Ki | 38 | — | |
XJSFDMGICAWQFS
|
7.8 | Ki | 60 | — | |
DXRCURBJOZPWHE
|
7.8 | IC50 | 2 | — |