Target Details
| UniProt AC | P04629 |
|---|---|
| Gene Symbol | NTRK1 |
| Protein Name | High affinity nerve growth factor receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF13855 (LRR_8) PF16920 (LRRCT_2) PF07714 (PK_Tyr_Ser-Thr) PF18613 (TrkA_TMD) |
Summary
- Multi-target molecules 1,127
- Clinical molecules 52
- Avg pChEMBL 7.65
KEGG Pathways (11)
Associated Diseases (4)
Active Molecules (1,127)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KWZZATFXFXCGHQ
|
10.8 | Kd | 2 | — | |
NRFMLFPXDKIQBF
|
10.5 | Kd | 8 | — | |
TTWJGJUDRLYONZ
|
10.3 | Kd | 6 | — | |
TTWJGJUDRLYONZ
|
10.2 | Kd | 4 | — | |
GNQRZYQSGPWTMY
|
10.1 | Kd | 2 | — | |
ROQYSCDOJUQZFY
|
10.1 | Kd | 2 | — | |
SMKJDFHRUWJNRS
|
10.0 | IC50 | 2 | — | |
HQXVNKKSTUDRSP
|
9.8 | Kd | 2 | — | |
AFTKSWNHMAKIPE
|
9.7 | Kd | 2 | — | |
DRJKEMBRQFSLFC
|
9.7 | IC50 | 3 | — | |
JHUWBOAVDAIILQ
|
9.7 | IC50 | 2 | — | |
JUNWLAORTWKJOM
|
9.7 | IC50 | 3 | — | |
KDCGROMZSUCCMF
|
9.7 | IC50 | 3 | — | |
LKPIGXCNFCFRED
|
9.7 | IC50 | 3 | — | |
PMAXBYMGMQSUFK
|
9.7 | IC50 | 3 | — | |
QGGXHLDONRQJQK
|
9.7 | IC50 | 2 | — | |
QGYZTXJGBDCZHX
|
9.7 | IC50 | 3 | — | |
TVUFMDRGVRGPIS
|
9.7 | IC50 | 3 | — | |
VIEKBHGPZROLOI
|
9.7 | IC50 | 3 | — | |
YLAKIDRGVDYWAA
|
9.7 | IC50 | 2 | — | |
SRWSLWJKGRZRMC
|
9.6 | Kd | 4 | — | |
VGEDWONGQUXJQA
|
9.6 | IC50 | 7 | — | |
DGQKIQCSFPDDDR
|
9.5 | IC50 | 3 | — | |
GJQVPMWSXKFICV
|
9.5 | IC50 | 3 | — | |
GJQVPMWSXKFICV
|
9.5 | IC50 | 3 | — | |
HVRWZFQFSQUILC
|
9.5 | IC50 | 4 | — | |
KQYVFELJSCVCND
|
9.4 | IC50 | 4 | — | |
GVDDEBQJCYQLKV
|
9.4 | IC50 | 3 | — | |
OOFWNPIPNPKKSR
|
9.4 | IC50 | 2 | — | |
YEQLIQZCYJPPOO
|
9.4 | IC50 | 2 | — | |
ZWIVMZNSHMYADK
|
9.4 | IC50 | 3 | — | |
WTGWCKJMZHWOAA
|
9.3 | IC50 | 2 | — | |
BYKOKZMCLVWDCZ
|
9.3 | IC50 | 3 | — | |
GYWAMONQPZXXDB
|
9.3 | IC50 | 2 | — | |
KPAKQPANQHIDII
|
9.3 | IC50 | 2 | — | |
PMTYXROLPZFSKY
|
9.3 | IC50 | 3 | — | |
XJNRYKKXKPGNHH
|
9.3 | IC50 | 2 | — | |
IOYWVCSTQWIERE
|
9.3 | IC50 | 2 | — | |
PKQSRPZFIGJTJF
|
9.3 | IC50 | 2 | — | |
JXLZJPYLDDSEQF
|
9.2 | IC50 | 2 | — | |
VPTLPKOEIZQIAS
|
9.2 | IC50 | 4 | — | |
GPUJXNIEEVLNGE
|
9.2 | IC50 | 2 | — | |
VXKMMMZVPVHQBU
|
9.2 | IC50 | 2 | — | |
GDVDELGPSHNWGV
|
9.2 | IC50 | 4 | — | |
FUHAANUNQWUCBT
|
9.2 | IC50 | 2 | — | |
INXXEGXCIVUCST
|
9.2 | IC50 | 2 | — | |
KVPNOQAXVUMKFJ
|
9.2 | IC50 | 3 | Yes | |
QHFNVZMOKIFBBE
|
9.2 | IC50 | 3 | — | |
RHFCOBKLSNCFAP
|
9.2 | IC50 | 2 | — | |
RHFCOBKLSNCFAP
|
9.2 | IC50 | 2 | — |