Target Details
| UniProt AC | P04628 |
|---|---|
| Gene Symbol | WNT1 |
| Protein Name | Proto-oncogene Wnt-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00110 (wnt) |
Summary
- Multi-target molecules 30
- Clinical molecules 0
- Avg pChEMBL 7.51
KEGG Pathways (17)
- Alzheimer disease
- Basal cell carcinoma
- Breast cancer
- Cadherin signaling
- Chemical carcinogenesis - receptor activation
- Cushing syndrome
- Gastric cancer
- Hepatocellular carcinoma
- Hippo signaling pathway
- Human papillomavirus infection
- Melanogenesis
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Proteoglycans in cancer
- Signaling pathways regulating pluripotency of stem cells
- Wnt signaling pathway
- mTOR signaling pathway
Associated Diseases (2)
Active Molecules (30)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BMTDMPCSMBKKPW
|
9.4 | Kd | 2 | — | |
GUGHZLAJQJKGHH
|
8.5 | IC50 | 2 | — | |
VEGYHVAUPWTKCC
|
8.4 | IC50 | 2 | — | |
XHMCMYNTRDDSMY
|
8.3 | IC50 | 2 | — | |
OLUJPDZZXTUOGS
|
8.2 | IC50 | 2 | — | |
PEEGMHUVHOESOC
|
8.1 | IC50 | 2 | — | |
KGFURJWQBPWTLA
|
7.6 | IC50 | 2 | — | |
HRERMENVFOCZBH
|
7.6 | IC50 | 2 | — | |
VKNDFKHJWONMCW
|
7.5 | IC50 | 2 | — | |
SLDVLHLDCYVDTB
|
7.5 | IC50 | 2 | — | |
XCWMMTANKPXNAA
|
7.5 | IC50 | 2 | — | |
UFCGCLZYGBXDNP
|
7.4 | IC50 | 2 | — | |
QWXGMMPJHDIFKI
|
7.4 | IC50 | 2 | — | |
QQSBPJPTYYIUQB
|
7.4 | IC50 | 2 | — | |
VWPTZVMBSFOJFR
|
7.3 | IC50 | 2 | — | |
PMSDXFRJIMIWMZ
|
7.3 | IC50 | 2 | — | |
YDPWZFPXWFTXNT
|
7.3 | IC50 | 2 | — | |
HVEOEVJLUUUHNZ
|
7.2 | IC50 | 2 | — | |
UEZHKJJFOLPGJG
|
7.2 | IC50 | 2 | — | |
LIXXQBRPVXEVJX
|
7.2 | IC50 | 2 | — | |
OLMDVYFVQFYWFE
|
7.2 | IC50 | 2 | — | |
REZVRRKMWKNZIG
|
7.2 | IC50 | 2 | — | |
SZBCOWYOKDHMCB
|
7.2 | IC50 | 2 | — | |
ZRFQUQSHTMRTPA
|
7.2 | IC50 | 2 | — | |
NDJKPKCOLSTNDX
|
7.1 | IC50 | 2 | — | |
WNKNLOWIRTYXCK
|
7.1 | IC50 | 2 | — | |
BSRXYRKKHONROQ
|
7.0 | IC50 | 2 | — | |
AQRWIEDTFAJEIU
|
7.0 | IC50 | 2 | — | |
FJQLBBOHMPVGMM
|
7.0 | IC50 | 2 | — | |
WUNIOBKOULBZPD
|
6.9 | IC50 | 2 | — |