Target Details
UniProt ACP04585
Gene Symbolgag-pol
Protein NameGag-Pol polyprotein
OrganismHuman immunodeficiency virus type 1 group M subtype B (isolate HXB2)
Entry Name
Organism Category Pathogen
Pfam Domains PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC)
Summary
  • Multi-target molecules 2,623
  • Clinical molecules 3
  • Avg pChEMBL 7.89
Top Co-occurrence Targets
Active Molecules (2,623)
InChIKey pChEMBL Type Targets Clinical
LUPHHMLWZFHILP 9.3 Ki 2
RXPWCKNSECMTEA 9.3 Ki 2
XXLADDZTQVLRQL 9.3 IC50 2
PKOHXONANBPFJD 9.3 IC50 2
GOVFYIPWKUFSHK 9.3 IC50 2
LUWZWPBFBGGXGY 9.3 Ki 2
QFHSEPSATCMBAS 9.3 IC50 2
WIWAETJMEYEKLK 9.3 IC50 2
WYBXHGHEBRRYPS 9.3 Ki 2
YEIHIAKNVFDXRE 9.3 Ki 2
ARFWEJPKRPPMNX 9.3 IC50 2
GCTCWKNGECMMNZ 9.3 Ki 2
AOMZDQMIOCTPQP 9.3 IC50 2
FBACKGQAIDXNSL 9.3 Ki 2
KEZWGZKGBARAAS 9.3 IC50 2
OXJNORCDTACECD 9.3 Kd 2
ZCQKFPOPDUPHBO 9.3 Ki 2
CGVKYOROKILIOK 9.3 Ki 2
CVQBZPGFVBDMPA 9.3 Ki 2
HPNJYSSQMDYJFF 9.3 IC50 2
HSMOPCIGLSCZAN 9.3 IC50 2
QMFFUYFALTVNOP 9.3 Ki 2
TUKYSJHHBDCNFR 9.3 IC50 2
UDMBCSSLTHHNCD 9.3 Kd 11
UOYZVCHWBOUTTL 9.3 IC50 2
VDVDBLXUHMXJMB 9.3 Ki 2
YLHWBQKQACUIES 9.3 IC50 2
YTGKHEDTLHRZGX 9.3 Ki 2
ZTPYYSCZRHAURY 9.3 IC50 2
ZTPYYSCZRHAURY 9.3 IC50 2
ZTPYYSCZRHAURY 9.3 IC50 2
MXQKEJBEBISBEI 9.3 IC50 2
NIQINMSYVZRSSS 9.3 Ki 2
NTOMRLCGHVNSKO 9.3 Ki 2
HTMNHRZEFBOZIL 9.2 IC50 2
UAUIISPUXGSUCV 9.2 Ki 3
VWTCVPCATZPCSU 9.2 IC50 2
YYTCBCZEWNZXGE 9.2 Ki 2
ANQYWJUUKHEXEZ 9.2 IC50 2
CDZSRMLOVAYORE 9.2 Ki 2
DVZYXCFGZKASRG 9.2 Ki 2
GSZXVWDUELWIJN 9.2 Ki 2
HOUHLOFMBSYNBO 9.2 Ki 2
IFOCKTRSJOLRSQ 9.2 Ki 2
IKULWCUDELLUHH 9.2 Ki 2
IOUDUHWREIAEKP 9.2 IC50 2
KHDJJHQOPWRTEH 9.2 Ki 2
LIENTGAUXNCIDX 9.2 Ki 2
LUOVKNHWLXFGAD 9.2 IC50 2
LUXWCCSCNDRTSF 9.2 IC50 2
2D structure