Target Details
UniProt ACP04585
Gene Symbolgag-pol
Protein NameGag-Pol polyprotein
OrganismHuman immunodeficiency virus type 1 group M subtype B (isolate HXB2)
Entry Name
Organism Category Pathogen
Pfam Domains PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC)
Summary
  • Multi-target molecules 2,623
  • Clinical molecules 3
  • Avg pChEMBL 7.89
Top Co-occurrence Targets
Active Molecules (2,623)
InChIKey pChEMBL Type Targets Clinical
XLBGSVYCWSFTSF 9.5 IC50 2
YWMZEAWUKJYZAL 9.5 Ki 2
ZJBUCZFZQXPYFC 9.5 IC50 2
ZXCLCEUUOMEPJU 9.5 IC50 2
AXRYRYVKAWYZBR 9.5 Kd 6
HHKWKXOCHWLVQU 9.5 Ki 2
MXIJGNJMISLFIE 9.5 IC50 2
XTSOTYHBCMFVQM 9.5 Ki 2
FVPLDCLMENGNJU 9.5 IC50 2
SIZLAJZUXGNMNI 9.5 IC50 2
CBKVXTVDXOQSJH 9.5 Ki 2
BBKUVYHQFBLHIC 9.5 Ki 2
YDOBPQZYAZNHNJ 9.5 Ki 2
HOJASIJITQDJDA 9.5 IC50 2
JZVBSCXBZJRRCG 9.5 IC50 2
UBUFVRJUGFJQSI 9.5 IC50 2
LNHVJOYDAOVTNP 9.4 Ki 2
NTBLOIDJWKXDON 9.4 Ki 2
YCWHOUFNTCROPW 9.4 IC50 2
YQUBCGAUPRDIGJ 9.4 IC50 2
TZRRVSCDIPHXHN 9.4 IC50 2
TZRRVSCDIPHXHN 9.4 Ki 2
ZRCVYOLTPAJSLA 9.4 Ki 2
HFEQKONSPKYSGC 9.4 IC50 2
PHTGQOYLTMJQER 9.4 IC50 2
BOULRXFSMMLNQU 9.4 Ki 2
BOULRXFSMMLNQU 9.4 Ki 2
CIGKLJDIMXPQJJ 9.4 Ki 2
CVQXOSJUWRFKFF 9.4 Ki 2
DEIXMKHNHSPTMM 9.4 Ki 2
DLVWRVNLMLSWAC 9.4 IC50 2
DVMNWHOQQSLWLE 9.4 IC50 2
FMROKUKFSAXFKK 9.4 Ki 2
GIAFMJHKTOLTOT 9.4 Ki 2
JFCQCUMIFWYQLQ 9.4 Ki 2
PCQQCKRYZKOPFN 9.4 IC50 2
QWAXKHKRTORLEM 9.4 Ki 5
SSAWLODCPROYGG 9.4 IC50 2
ZZHSDDNNVHINCL 9.4 Ki 2
QERMHAOACKVOPG 9.4 Ki 2
RYPMMFFNVUMBFD 9.4 Ki 2
UGTCZVWIXZGMAD 9.4 Ki 2
XYGAZPXCXXYIJV 9.4 Ki 2
CBVONKNRKVRZIS 9.4 IC50 2
ZYXJGWBYPOHODT 9.4 IC50 2
IVLGUQXISOUHPG 9.4 Ki 2
ZBAREFVKRAICLD 9.4 Ki 2
LKPGUETYCTUNHI 9.4 IC50 2
XSTOMTIANVBPAN 9.4 IC50 2
IYLCQJSWFWQHCD 9.3 IC50 2
2D structure