Target Details
UniProt ACP04585
Gene Symbolgag-pol
Protein NameGag-Pol polyprotein
OrganismHuman immunodeficiency virus type 1 group M subtype B (isolate HXB2)
Entry Name
Organism Category Pathogen
Pfam Domains PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC)
Summary
  • Multi-target molecules 2,623
  • Clinical molecules 3
  • Avg pChEMBL 7.89
Top Co-occurrence Targets
Active Molecules (2,623)
InChIKey pChEMBL Type Targets Clinical
ADFMHXPVMGVOGF 9.6 Ki 2
BYFQZUPDPUOMAR 9.6 Ki 2
GHONSWTUVKSWOK 9.6 IC50 2
GHONSWTUVKSWOK 9.6 IC50 2
GHONSWTUVKSWOK 9.6 IC50 2
QENQYVYSOVDJNK 9.6 IC50 2
QWFUVXWNTBYMHA 9.6 Ki 2
TZRRVSCDIPHXHN 9.6 Ki 2
UFELAQKNFHLHDW 9.6 IC50 2
UVBAPKJSTSROOR 9.6 Ki 2
YGNMRRZJWHABRJ 9.6 Ki 2
ZJBUCZFZQXPYFC 9.6 IC50 2
ZJBUCZFZQXPYFC 9.6 IC50 2
BGHYHFHFLYFAEU 9.6 Ki 2
FZPJTHVATYWFGZ 9.6 Ki 2
GHBUZSGLSLUJLN 9.6 IC50 2
GHBUZSGLSLUJLN 9.6 IC50 2
PHDPGJPLZABKFA 9.6 IC50 2
QKUZOQWGKMBGSS 9.6 Ki 2
QLFYYBGXVAYDRB 9.6 IC50 2
SUVMGYUHKSTITP 9.6 IC50 2
UKHGTNBNXUQEFN 9.6 Ki 2
GHBUZSGLSLUJLN 9.6 IC50 2
AOLQBHBDLWMQMX 9.6 IC50 2
AOLQBHBDLWMQMX 9.6 IC50 2
AOLQBHBDLWMQMX 9.6 IC50 2
CKRRAJMIYUMXET 9.6 Ki 2
CXDXPJIIEKARJN 9.6 IC50 2
GFVONONAIXMHFG 9.6 Ki 2
FACWTLYMDWLMTA 9.6 Ki 2
FNVKNXUOXYUBDJ 9.6 IC50 2
KYRSNWPSSXSNEP 9.6 Ki 3
QYRBHDADFBLWJR 9.6 Ki 2
UYIDPTWMZFMUKR 9.6 IC50 2
ZMLZLWMYQDSDEB 9.6 Ki 2
CYHCGEKJFIIQML 9.5 IC50 2
CYHCGEKJFIIQML 9.5 IC50 2
CYHCGEKJFIIQML 9.5 IC50 2
PFIHOIVFDOGGJU 9.5 Ki 2
RQSUYZMJIBUYTC 9.5 IC50 2
BHLOBVCFHPPZKS 9.5 Ki 2
BYQUYNCKPYLJOZ 9.5 IC50 2
DFMFLMIHIUQRSX 9.5 IC50 2
FOPJEVCXMWTXGE 9.5 IC50 2
INZGMOIEIWGIQN 9.5 Ki 2
NBTQOOJUNCNMQJ 9.5 IC50 2
NOVVCLRXWROCGF 9.5 Ki 2
PRDAIONOCJACSU 9.5 Ki 2
SGEXQIUVSGWABP 9.5 Ki 2
SKACOTBQIAXUOJ 9.5 Ki 2
2D structure