Target Details
UniProt ACP04585
Gene Symbolgag-pol
Protein NameGag-Pol polyprotein
OrganismHuman immunodeficiency virus type 1 group M subtype B (isolate HXB2)
Entry Name
Organism Category Pathogen
Pfam Domains PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC)
Summary
  • Multi-target molecules 2,623
  • Clinical molecules 3
  • Avg pChEMBL 7.89
Top Co-occurrence Targets
Active Molecules (2,623)
InChIKey pChEMBL Type Targets Clinical
FYPXVPUOPMHLDN 9.7 Ki 2
FZVFAVNAEOSRRU 9.7 Ki 2
HGLNUSNAKTZJGO 9.7 IC50 2
PYMPNOZOVIYDGG 9.7 Ki 2
UORPPOQBOUNVPY 9.7 IC50 2
AACGEOQWBRCPAI 9.7 IC50 2
BNEUUKYSHWONFU 9.7 IC50 2
BNEUUKYSHWONFU 9.7 IC50 2
BNEUUKYSHWONFU 9.7 IC50 2
JMQRXLDQVOPBLV 9.7 Ki 2
LDGYHSNFNKEYMA 9.7 Ki 2
VWHDFJUUEYKFKE 9.7 Ki 2
YBOQWURBTADCQS 9.7 Ki 2
CVHFWKHAVARIHF 9.7 IC50 2
FYAYMVRGJWVUBF 9.7 Ki 2
MCZPUJMGYKWSIX 9.7 Ki 2
UOHMQWQGAJAUGT 9.7 Ki 2
UPTRZAHECQTLFN 9.7 IC50 2
CWNUTRRUJFJVNU 9.7 Ki 2
GPEVFYOHNNRULA 9.7 IC50 2
MDHGCCCKMXCXRP 9.7 Ki 2
OIGRVBGGQVHPRF 9.7 IC50 2
TZRRVSCDIPHXHN 9.7 IC50 2
UVWWXOZKXJOILJ 9.7 Ki 2
XQHWXGQOXZQZFF 9.7 IC50 2
CUKAUEXJVJXEDL 9.7 Ki 2
HSGWMHCBWWNMPP 9.7 IC50 2
LYXPKYLWOJGHAC 9.7 IC50 2
NIQZVJVTQIZVKW 9.7 IC50 2
TZRRVSCDIPHXHN 9.7 IC50 2
TZRRVSCDIPHXHN 9.7 IC50 2
TZRRVSCDIPHXHN 9.7 IC50 3
DIMZZOUXFBIBDD 9.6 Ki 2
IPITVBZBTYXTRI 9.6 Ki 2
MFSVHROQWVRSOF 9.6 IC50 2
MFSVHROQWVRSOF 9.6 IC50 2
MFSVHROQWVRSOF 9.6 IC50 2
NIQZVJVTQIZVKW 9.6 IC50 2
NSEDEVLFQHAAFP 9.6 Ki 2
QWAXKHKRTORLEM 9.6 IC50 2
ZRLPHWQOZNLOMW 9.6 Ki 3
DOYLRRXQCZFMEN 9.6 Ki 2
HFRPLIKYGJIHRM 9.6 Ki 2
KEXFGVLHSFYUMX 9.6 Ki 2
MJOXWVYKMFPFPL 9.6 Ki 2
MJOXWVYKMFPFPL 9.6 Ki 2
MUEGWYUBGOOONU 9.6 Ki 2
UHTHHESEBZOYNR 9.6 Ki 66 Yes
UKOAHKBCCOTOFZ 9.6 IC50 2
IQDCZKUNYMTBBJ 9.6 Ki 2
2D structure