Target Details
UniProt ACP04585
Gene Symbolgag-pol
Protein NameGag-Pol polyprotein
OrganismHuman immunodeficiency virus type 1 group M subtype B (isolate HXB2)
Entry Name
Organism Category Pathogen
Pfam Domains PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC)
Summary
  • Multi-target molecules 2,623
  • Clinical molecules 3
  • Avg pChEMBL 7.89
Top Co-occurrence Targets
Active Molecules (2,623)
InChIKey pChEMBL Type Targets Clinical
JMNLVMWRVGPARO 9.9 Ki 2
BMUFHJJGKINDQD 9.9 Ki 2
FIUNGTDDQHDHHT 9.9 IC50 2
HVWSACNCBBMPIU 9.9 IC50 2
KNZXQUNBQJDYHJ 9.9 IC50 2
WEOXFVJLLOSYHC 9.9 Ki 2
YCDGAESMEYQMIE 9.9 Ki 2
GHOKUHSKMRQFHB 9.9 Ki 2
JSYUNEPXLBQPTN 9.9 Ki 2
LUPHHMLWZFHILP 9.9 Ki 2
OCVIFOLUOWMFFU 9.9 Ki 2
SKXIDYZBFCDEPH 9.9 Ki 2
WVOSVUDMDYDQMC 9.9 IC50 2
ACHQUDJPGNODSX 9.8 IC50 2
BDLUEJUQSRGZLT 9.8 Ki 2
FYQHJBBCNRLSBW 9.8 IC50 2
HVYNAUPARPIAME 9.8 IC50 2
ITOMYUFMQRFCHM 9.8 Ki 2
JFFVTCOLDQQGTQ 9.8 IC50 2
SGZKFBCCMDSJAH 9.8 IC50 2
VPFBCSZFKQTTKA 9.8 Ki 2
VXCNHQRMEWBANV 9.8 Ki 2
WKRXSHDQEAFLGC 9.8 Ki 2
CMBKNLUUKVNRNH 9.8 Ki 2
CNNKZGRBCPFNKW 9.8 IC50 2
KWIOWBKKSAFPTL 9.8 Ki 2
PIBLAKANIOZAPU 9.8 Ki 2
WPNGOVIGRGIGBK 9.8 IC50 2
AZMMWXVEVKAJAZ 9.8 IC50 2
FBVWDPCOHLLXSB 9.8 Ki 2
IXMOCJVKYIUCEJ 9.8 IC50 2
IXMOCJVKYIUCEJ 9.8 IC50 2
IXMOCJVKYIUCEJ 9.8 IC50 2
NEFNRKCIJRROFR 9.8 Ki 2
RSURGPQKNWGOQG 9.8 IC50 2
TYTLIFJNIMETBZ 9.8 IC50 2
WYBXHGHEBRRYPS 9.8 Ki 2
PFQCUMURCZHTBY 9.8 Ki 3
ZGVUOBCKGRJVSM 9.8 Ki 2
APYLHGQERCKLFK 9.8 IC50 2
CQORGNMKPNEUQR 9.8 Ki 2
JBEBAOJLXPMRIO 9.8 IC50 2
JBEBAOJLXPMRIO 9.8 IC50 2
MWLXVUTUBLGYCG 9.8 Ki 2
MWVDAODXAGANDN 9.8 Ki 2
OFKWXCJKTQUOHD 9.8 Ki 2
QJMAYXGAURCBTD 9.8 Ki 2
BXVIHKICSIIIDC 9.8 IC50 2
AOMZDQMIOCTPQP 9.7 IC50 2
BXVIHKICSIIIDC 9.7 IC50 2
2D structure