Target Details
| UniProt AC | P04585 |
|---|---|
| Gene Symbol | gag-pol |
| Protein Name | Gag-Pol polyprotein |
| Organism | Human immunodeficiency virus type 1 group M subtype B (isolate HXB2) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC) |
Summary
- Multi-target molecules 2,623
- Clinical molecules 3
- Avg pChEMBL 7.89
Top Co-occurrence Targets
- pol 1997 shared
- pol 499 shared
- pol 110 shared
- reverse transcriptase 44 shared
- protease 36 shared
- 18 shared
- CTSD 9 shared
- reverse transcriptase 7 shared
- CTSE 6 shared
- CYP3A4 6 shared
Active Molecules (2,623)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HPJIIOAWLFOWEM
|
10.1 | Ki | 2 | — | |
XUJKOFQIVYUCKQ
|
10.1 | Ki | 2 | — | |
LCESHYGFELECTB
|
10.1 | Ki | 2 | — | |
MUULRSITXOVVFK
|
10.1 | IC50 | 3 | — | |
FQPGLEJBVZRHEH
|
10.1 | IC50 | 2 | — | |
KJSCXVXFOAVQHM
|
10.1 | Ki | 2 | — | |
MMUOMMUDZAEDSY
|
10.1 | Ki | 2 | — | |
SNSQMJFLZPJQFY
|
10.1 | IC50 | 2 | — | |
SXPVUUNIEQEZAM
|
10.1 | Ki | 2 | — | |
QVLACFTWGMNBKP
|
10.1 | Ki | 2 | — | |
VXTBMTMRCNWYCK
|
10.1 | Ki | 2 | — | |
HABWGFQXGJRKQW
|
10.1 | Ki | 2 | — | |
HPZHVLWFMURXBI
|
10.1 | Ki | 2 | — | |
LUOOIXNNRYGGEB
|
10.1 | Ki | 2 | — | |
DQWBRZRJSHIBMA
|
10.1 | Ki | 2 | — | |
HLIXOQRYGLWYLS
|
10.1 | Ki | 2 | — | |
KYTKGYRYFOOIRX
|
10.1 | Ki | 2 | — | |
QYYDGLUFMLECTL
|
10.1 | Ki | 2 | — | |
SMBRIZZXTVLKIM
|
10.1 | IC50 | 2 | — | |
VMOXIVNTBGBVFS
|
10.1 | Ki | 2 | — | |
ZFONAWOOOSRORK
|
10.1 | Ki | 2 | — | |
AYFXUKGPCFAPOC
|
10.0 | Ki | 2 | — | |
ARGINUMNBCUKGF
|
10.0 | Ki | 2 | — | |
GGABOCICEXDWLA
|
10.0 | Ki | 2 | — | |
CBKBMLZVZNDFDQ
|
10.0 | Ki | 2 | — | |
DUBLLIBPEZQWQP
|
10.0 | IC50 | 2 | — | |
GDHLTMGXRIRQHJ
|
10.0 | Ki | 2 | — | |
HKAQGSPFDKETKG
|
10.0 | IC50 | 2 | — | |
HKAQGSPFDKETKG
|
10.0 | IC50 | 2 | — | |
HKAQGSPFDKETKG
|
10.0 | IC50 | 2 | — | |
IFTQDGRYVXWWMV
|
10.0 | Ki | 2 | — | |
JWGRPULBGOAZNR
|
10.0 | Ki | 2 | — | |
KQKOIRSEVVSSJU
|
10.0 | Ki | 2 | — | |
MCGUXOJCMTXXSP
|
10.0 | Ki | 2 | — | |
MYUBPZWAEVYXRT
|
10.0 | Ki | 2 | — | |
SGEXQIUVSGWABP
|
10.0 | Ki | 2 | — | |
WOVKOKXRLSYFEP
|
10.0 | Ki | 2 | — | |
YKFONWPAYRGADG
|
10.0 | IC50 | 2 | — | |
YVSHLJNQUPFXTP
|
10.0 | Ki | 2 | — | |
ZCNACGKIKDEZFC
|
10.0 | Kd | 2 | — | |
ZCSGMVSDPDUOEO
|
10.0 | Ki | 2 | — | |
ZZHSDDNNVHINCL
|
10.0 | Ki | 2 | — | |
AIUFCENHONWFHI
|
10.0 | IC50 | 2 | — | |
KDLXYIKRRNIZGK
|
10.0 | IC50 | 2 | — | |
OQLXXEYSDKXFLY
|
10.0 | Ki | 2 | — | |
TYWFTCCQWGMFKY
|
10.0 | Ki | 2 | — | |
WHERZNBVXWXRIV
|
10.0 | IC50 | 2 | — | |
XMZJHJWRJGSPBC
|
10.0 | IC50 | 2 | — | |
YAVCJFGXZDADDF
|
10.0 | IC50 | 2 | — | |
YAXGRNOGUNEIBE
|
9.9 | Ki | 2 | — |