Target Details
| UniProt AC | P04585 |
|---|---|
| Gene Symbol | gag-pol |
| Protein Name | Gag-Pol polyprotein |
| Organism | Human immunodeficiency virus type 1 group M subtype B (isolate HXB2) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC) |
Summary
- Multi-target molecules 2,623
- Clinical molecules 3
- Avg pChEMBL 7.89
Top Co-occurrence Targets
- pol 1997 shared
- pol 499 shared
- pol 110 shared
- reverse transcriptase 44 shared
- protease 36 shared
- 18 shared
- CTSD 9 shared
- reverse transcriptase 7 shared
- CTSE 6 shared
- CYP3A4 6 shared
Active Molecules (2,623)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KDXDWVNUODBVJT
|
10.3 | Ki | 2 | — | |
MYLPKRNDNXIKCB
|
10.3 | Ki | 2 | — | |
IOMNHKSPZZFZEP
|
10.3 | Ki | 2 | — | |
PYWNSKWRILMNRI
|
10.3 | Ki | 2 | — | |
UFEKNFOQGIREOW
|
10.3 | Ki | 2 | — | |
VRMCATPXWRGROO
|
10.3 | IC50 | 2 | — | |
CZPUBQYAVIVNEX
|
10.3 | Ki | 2 | — | |
JPWJMZNJZWAWDA
|
10.3 | IC50 | 2 | — | |
ZTHXXPRDWPPMMG
|
10.3 | Ki | 3 | — | |
HFLCERPZYCWLSZ
|
10.2 | Ki | 2 | — | |
HRXLCWSIQGZEGT
|
10.2 | Ki | 2 | — | |
QMZHGXPLZJHFBF
|
10.2 | Ki | 2 | — | |
BVVVLUBDVRWMQM
|
10.2 | Ki | 2 | — | |
CTXMFQMWMNCPNF
|
10.2 | Ki | 2 | — | |
NSBJLKKRNVGNHW
|
10.2 | Ki | 2 | — | |
UGMGBADCLGQMSF
|
10.2 | Ki | 2 | — | |
DOGRITFNUGZZKZ
|
10.2 | Ki | 2 | — | |
FWDLLMHEAFMLAW
|
10.2 | IC50 | 2 | — | |
GVWYIVARRNFICI
|
10.2 | Ki | 2 | — | |
HJBJOSQKBXBTER
|
10.2 | Ki | 2 | — | |
MRVQZDYNHXWYFK
|
10.2 | IC50 | 2 | — | |
PKJPLBXKJRGYRL
|
10.2 | IC50 | 2 | — | |
PKJPLBXKJRGYRL
|
10.2 | IC50 | 2 | — | |
UVPHTIRJUNYMJM
|
10.2 | Ki | 2 | — | |
GWGPTSIQUUQYEQ
|
10.2 | Ki | 2 | — | |
NBQYBSPBXGGPQZ
|
10.2 | Ki | 2 | — | |
NDUNEENBMMFTKS
|
10.2 | Ki | 2 | — | |
PLNSJJUTQRVZIK
|
10.2 | IC50 | 2 | — | |
BKKQECSJRDVDJZ
|
10.2 | Ki | 2 | — | |
MXFDAKCCGMVOPP
|
10.2 | Ki | 2 | — | |
OMUXFMWDWOOQFU
|
10.2 | Ki | 2 | — | |
PAKVCZYVTVITSB
|
10.2 | Ki | 2 | — | |
SAIHLPVEVOOIMK
|
10.2 | Ki | 2 | — | |
PJOMOXITHVFIDP
|
10.2 | Ki | 2 | — | |
XEZWGCBUEIJERI
|
10.2 | Ki | 2 | — | |
ZCKKCLQSZRCWAP
|
10.2 | Ki | 2 | — | |
ZQHWCROOUMKOGV
|
10.2 | Ki | 2 | — | |
NAFWCKJKWJNABK
|
10.2 | Ki | 2 | — | |
SFASRDRWOGHVFO
|
10.2 | Ki | 2 | — | |
PKBPUJCUWPCIQB
|
10.2 | Ki | 2 | — | |
SQFKCAMRRRAISM
|
10.2 | Ki | 2 | — | |
TWYFSQMHPWOVSQ
|
10.2 | Ki | 2 | — | |
VJQAUXZKAOWRNN
|
10.2 | Ki | 2 | — | |
WMTSGCIMPPZQLI
|
10.2 | IC50 | 2 | — | |
FEICASSQSGPGGQ
|
10.1 | Ki | 2 | — | |
SOAFVHMCUQHVNN
|
10.1 | Ki | 2 | — | |
WWTORRPIIMGMSP
|
10.1 | Ki | 2 | — | |
RPQLINAEDRJPQC
|
10.1 | Ki | 2 | — | |
WVKJHIVGBANALA
|
10.1 | Ki | 3 | — | |
GDEOHSJOOBUKGL
|
10.1 | Ki | 2 | — |