Target Details
| UniProt AC | P04585 |
|---|---|
| Gene Symbol | gag-pol |
| Protein Name | Gag-Pol polyprotein |
| Organism | Human immunodeficiency virus type 1 group M subtype B (isolate HXB2) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC) |
Summary
- Multi-target molecules 2,623
- Clinical molecules 3
- Avg pChEMBL 7.89
Top Co-occurrence Targets
- pol 1997 shared
- pol 499 shared
- pol 110 shared
- reverse transcriptase 44 shared
- protease 36 shared
- 18 shared
- CTSD 9 shared
- reverse transcriptase 7 shared
- CTSE 6 shared
- CYP3A4 6 shared
Active Molecules (2,623)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RREYCVXDIYCIMA
|
10.6 | Ki | 2 | — | |
VFYUAUUEVXEJCV
|
10.6 | Ki | 2 | — | |
ZTHXXPRDWPPMMG
|
10.6 | Ki | 3 | — | |
PVRCWMUDFFKIAS
|
10.6 | Ki | 2 | — | |
QDVCOPOXCTUFAE
|
10.5 | Ki | 2 | — | |
WZCSZCGNEYLDGF
|
10.5 | Ki | 2 | — | |
AWXAHWJTZBZGDD
|
10.5 | IC50 | 2 | — | |
DYJSVMWNEYFCMD
|
10.5 | IC50 | 2 | — | |
IWRWYUHCNLAARG
|
10.5 | Ki | 2 | — | |
KBAOMTHUUATJOU
|
10.5 | Ki | 2 | — | |
QQBJVZITBVPJOA
|
10.5 | Ki | 2 | — | |
QSZNPSNWAHVNPD
|
10.5 | Ki | 2 | — | |
STHYWTNVNDGESC
|
10.5 | Ki | 2 | — | |
TWDLOKWTPCLJHI
|
10.5 | Ki | 2 | — | |
WXJFTRVJBDTLCM
|
10.5 | Ki | 2 | — | |
XETIIHXJGVJJAT
|
10.5 | IC50 | 2 | — | |
NTWKGLJNQAZSHF
|
10.5 | Ki | 3 | — | |
RXBWRFDZXRAEJT
|
10.5 | Ki | 2 | — | |
WNBSRRDTYWNYHA
|
10.5 | Ki | 4 | — | |
KGLXFRRLZYLFHH
|
10.5 | Ki | 2 | — | |
GCKOKIJMLAUYIK
|
10.5 | Ki | 2 | — | |
ILUZTGNKABEPFV
|
10.5 | Ki | 2 | — | |
QMNGJVDHBPPPHI
|
10.5 | Ki | 2 | — | |
XRYNUFMTUIJXSU
|
10.5 | Ki | 2 | — | |
PMFZQWVRDGSFAW
|
10.4 | Ki | 2 | — | |
ZKXPPUAKSSRSJN
|
10.4 | Ki | 2 | — | |
KTZXIYPLRZIZDJ
|
10.4 | Ki | 2 | — | |
QNMCBWIGCQHDEC
|
10.4 | Ki | 3 | — | |
YKAFTOZYPINVBL
|
10.4 | Ki | 2 | — | |
CJINWGNBIYXOEZ
|
10.4 | Ki | 2 | — | |
OYLKHGYQDBGESE
|
10.4 | Ki | 2 | — | |
FBTRQCVYUQUHSD
|
10.4 | Ki | 2 | — | |
AAGQNDDFCSYHQM
|
10.4 | Ki | 2 | — | |
FRDXWSPCQJVMNT
|
10.4 | Ki | 2 | — | |
GKDXSQFJDXXEOT
|
10.4 | IC50 | 2 | — | |
KGNBXGDXRKLBII
|
10.4 | Ki | 2 | — | |
OMCGYRQJCQVPHF
|
10.4 | Ki | 2 | — | |
BSDDZYDMOFWADT
|
10.4 | Ki | 2 | — | |
XNMNZSWFRFPRFY
|
10.4 | Ki | 2 | — | |
PNRNVSUAECQBDO
|
10.3 | Ki | 2 | — | |
TWQHRSJOMZMREM
|
10.3 | Ki | 2 | — | |
WENSXXFBLAFVRJ
|
10.3 | Ki | 2 | — | |
VQJIBGNHKRKROK
|
10.3 | Ki | 2 | — | |
HHYBBXBBDLLGIU
|
10.3 | Ki | 2 | — | |
TYXASLSBMBZTJR
|
10.3 | Ki | 2 | — | |
XONGAKBEKSACMN
|
10.3 | Ki | 2 | — | |
QSPGRFMCYWCCTE
|
10.3 | Ki | 2 | — | |
AVKFJGHNZWYFBR
|
10.3 | IC50 | 2 | — | |
BKJDUSXQYYVNMA
|
10.3 | IC50 | 2 | — | |
JPWJMZNJZWAWDA
|
10.3 | IC50 | 2 | — |