Target Details
UniProt ACP04585
Gene Symbolgag-pol
Protein NameGag-Pol polyprotein
OrganismHuman immunodeficiency virus type 1 group M subtype B (isolate HXB2)
Entry Name
Organism Category Pathogen
Pfam Domains PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC)
Summary
  • Multi-target molecules 2,623
  • Clinical molecules 3
  • Avg pChEMBL 7.89
Top Co-occurrence Targets
Active Molecules (2,623)
InChIKey pChEMBL Type Targets Clinical
KWVACGKSVFDODQ 9.1 IC50 2
MLGIRVRCUGJSDP 9.1 Ki 2
SAFCQBPFQXDREG 9.1 IC50 2
UEXFBEJFUYIGPH 9.1 Ki 2
UZYMJLJOLJHHQY 9.1 Ki 2
GQXDRKLTUINFRX 9.1 IC50 2
LPLTVUOIANCCLD 9.1 Ki 2
IXGDYFOYTFQOBT 9.1 Ki 2
AYJMRCUOSGDJMG 9.1 Ki 2
JFITYPIRPPCROE 9.1 Ki 2
KCFFFABFDHZEJC 9.1 Ki 2
KKZRCEXYVFUNES 9.1 Ki 2
WCKIUOTZGKZJKC 9.1 Ki 2
LBQQXOLUDHGVFS 9.1 Ki 2
DCJXJZRHLYXSCU 9.1 IC50 2
FPBRNORXTMGALG 9.1 Kd 2
GLKONBHDVMFJNJ 9.1 Ki 2
RSEVSRUJHNNIBW 9.1 IC50 2
YVENLASUPXUYFI 9.1 Ki 2
ZWFXDTZPQGCUFZ 9.1 IC50 2
PRIFHIRAJRKFRJ 9.0 Ki 2
YUSMVPTWXWYLHG 9.0 Ki 2
IGGUZTVFIJYACD 9.0 IC50 2
ZYXJGWBYPOHODT 9.0 IC50 2
CAMSKFMUHQYCNZ 9.0 IC50 2
FACWTLYMDWLMTA 9.0 Ki 2
FXESQGVMUAWWTA 9.0 Ki 2
GBYCHLWJCGXUHJ 9.0 Ki 2
GCBPAPVOMPJQHK 9.0 Ki 9 Yes
JFKIHXVQWVFSNI 9.0 IC50 2
MJIHGBRCJJDHSL 9.0 Ki 2
NKEXROKZQNTBFE 9.0 IC50 2
NLFSULIAFLPDQL 9.0 IC50 2
QDSIURMOHBBWLV 9.0 Ki 2
QIZJJPPKMBIHOW 9.0 Ki 2
QSIYJFPEJMTCCY 9.0 IC50 2
RREBGKCKEYMFSB 9.0 IC50 2
TWONRKIIQCCNQJ 9.0 IC50 2
WMIYXLYUSXGLJD 9.0 Ki 2
XZMDRIWIUCSMJY 9.0 Ki 2
XZMDRIWIUCSMJY 9.0 Ki 2
YPEGMZWYPCFVRN 9.0 IC50 2
YZBQENDDAGQPSE 9.0 Ki 2
ZKAHZOFVRUTLSI 9.0 IC50 2
OVJXCZLLFSJYDS 9.0 IC50 2
CBVCZFGXHXORBI 9.0 Ki 6
BMVNYJXJBDEZBS 9.0 IC50 2
BNGZYPDWYZYMSS 9.0 IC50 2
FIGQLJMXYIMIGW 9.0 IC50 2
HQWLOOZWBNAXSA 9.0 IC50 2
2D structure