Target Details
UniProt ACP04585
Gene Symbolgag-pol
Protein NameGag-Pol polyprotein
OrganismHuman immunodeficiency virus type 1 group M subtype B (isolate HXB2)
Entry Name
Organism Category Pathogen
Pfam Domains PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC)
Summary
  • Multi-target molecules 2,623
  • Clinical molecules 3
  • Avg pChEMBL 7.89
Top Co-occurrence Targets
Active Molecules (2,623)
InChIKey pChEMBL Type Targets Clinical
LUXWCCSCNDRTSF 9.2 IC50 2
LUXWCCSCNDRTSF 9.2 IC50 2
MJOXWVYKMFPFPL 9.2 Ki 2
MJOXWVYKMFPFPL 9.2 Ki 2
MYAVIZSWDHVTAO 9.2 Ki 2
NCDNCNXCDXHOMX 9.2 Ki 12
NFRWMVLABDZMDS 9.2 Ki 2
QCJUNBVOLRPXTN 9.2 Ki 2
RQAVEWKEUKIFLD 9.2 Ki 2
WXOMYWCKSSDBHF 9.2 IC50 2
XVHCXIJZLNLRAY 9.2 IC50 2
XWPXFOUWOGRISF 9.2 IC50 2
YBWAJXBCPYCNKK 9.2 Ki 2
YIWOEKZROGXYDW 9.2 IC50 2
FHGXAASKOJAWKN 9.2 IC50 2
HSWCSZNROAIHDJ 9.2 Ki 2
JZXMAVVBPXQVSM 9.2 IC50 2
LGPKDDVYDWPIQK 9.2 IC50 2
ZCVHKZFFSQOZHU 9.2 Ki 2
JYRBGDQPGXEOAA 9.2 IC50 2
RAWLOIRTUZIAJE 9.2 Ki 2
MJOXWVYKMFPFPL 9.2 Ki 2
ZSIOVNJKQAGRBC 9.2 Ki 2
CFGOUUWGBUPZCL 9.2 IC50 2
HOSWQVAUWWIQFR 9.2 Ki 2
KRQUATQFBQPHBE 9.2 IC50 2
NGSRYSDZRCBGIJ 9.2 Ki 2
ZPWRQTPKKQTFGK 9.2 Ki 2
IMGCDQHXXAQTBJ 9.2 IC50 2
NNOFYWJFSHHUJW 9.2 IC50 2
UGSCYOQTKNVPEV 9.2 IC50 2
FITBNCMDDVVHAC 9.2 Ki 2
GSWLEEYHTJFDMI 9.2 Ki 2
IMGCDQHXXAQTBJ 9.2 IC50 2
QDNTXUZUWFKCPF 9.2 IC50 2
REGSUSUQOZCOPY 9.2 Ki 2
UZBJXXZZZVEMND 9.2 IC50 2
GWAFCACQJJTEDY 9.1 Ki 2
IZMLLFHMZHNYNG 9.1 Ki 2
KVSPJLUDFNMXCQ 9.1 IC50 2
KVSPJLUDFNMXCQ 9.1 IC50 2
SFNAMQNOKAGOEZ 9.1 IC50 2
XDASXYHIYMOGQE 9.1 Ki 2
VJCBVESGQNUVSA 9.1 Ki 2
QLKAFUZDAZPRSE 9.1 Ki 2
SSAWLODCPROYGG 9.1 IC50 2
XWDZZONMJRJYLZ 9.1 IC50 2
CANOIEBHYSFNQZ 9.1 IC50 2
MQPXOVRKKPPKFZ 9.1 IC50 2
JTGOXFUSCPOXKE 9.1 Ki 2
2D structure